3α-Hydroxy-3β-(phenylethynyl)-5β-pregnan-20-ones: Synthesis and Pharmacological Activity of Neuroactive Steroids with High Affinity for GABA A Receptors
Upasani, Ravindra B., Yang, Kevin C., Acosta-Burruel, Manuel, Konkoy, Chris S., McLellan, James A., Woodward, Richard M., Lan, Nancy C., Carter, Richard B., Hawkinson, Jon E.
Published in Journal of medicinal chemistry (03.01.1997)
Published in Journal of medicinal chemistry (03.01.1997)
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Synthesis of N-Substituted 4-(4-Hydroxyphenyl)piperidines, 4-(4-Hydroxybenzyl)piperidines, and (±)-3-(4-Hydroxyphenyl)pyrrolidines: Selective Antagonists at the 1a/2B NMDA Receptor Subtype
Guzikowski, Anthony P, Tamiz, Amir P, Acosta-Burruel, Manuel, Hong-Bae, Soo, Cai, Sui Xiong, Hawkinson, Jon E, Keana, John F. W, Kesten, Suzanne R, Shipp, Christina T, Tran, Minhtam, Whittemore, Edward R, Woodward, Richard M, Wright, Jon L, Zhou, Zhang-Lin
Published in Journal of medicinal chemistry (09.03.2000)
Published in Journal of medicinal chemistry (09.03.2000)
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Synthesis and in vitro activity of 3 beta-substituted-3 alpha-hydroxypregnan-20-ones: Allosteric modulators of the GABA(A) receptor
Hogenkamp, DJ, Tahir, SH, Hawkinson, JE, Upasani, RB, Alauddin, M, Kimbrough, CL, AcostaBurruel, M, Whittemore, ER, Woodward, RM, Lan, NC, Gee, KW, Bolger, MB
Published in Journal of medicinal chemistry (03.01.1997)
Published in Journal of medicinal chemistry (03.01.1997)
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Novel phosphoserine phosphatase inhibitors
Hawkinson, Jon E, Acosta-Burruel, Manuel, Ta, Nahn D, Wood, Paul L
Published in European journal of pharmacology (22.10.1997)
Published in European journal of pharmacology (22.10.1997)
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Journal Article
Synthesis of N- Substituted 4-(4-Hydroxyphenyl)piperidines, 4-(4-Hydroxybenzyl)piperidines, and (±)-3-(4-Hydroxyphenyl)pyrrolidines: Selective Antagonists at the 1 a /2B NMDA Receptor Subtype
Guzikowski, Anthony P., Tamiz, Amir P., Acosta-Burruel, Manuel, Hong-Bae, Soo, Cai, Sui Xiong, Hawkinson, Jon E., Keana, John F. W., Kesten, Suzanne R., Shipp, Christina T., Tran, Minhtam, Whittemore, Edward R., Woodward, Richard M., Wright, Jon L., Zhou, Zhang-Lin
Published in Journal of medicinal chemistry (01.03.2000)
Published in Journal of medicinal chemistry (01.03.2000)
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Substituted 3β-Phenylethynyl Derivatives of 3α-Hydroxy-5α-pregnan-20-one: Remarkably Potent Neuroactive Steroid Modulators of γ-Aminobutyric AcidA Receptors
Jon E. Hawkinson, Manuel Acosta-Burruel, Kevin C. Yang, Derk J. Hogenkamp, Jie-Sheng Chen, Nancy C. Lan, John A. Drewe, Edward R. Whittemore, Richard M. Woodward, Richard B. Carter, Ravindra B. Upasani
Published in The Journal of pharmacology and experimental therapeutics (01.10.1998)
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Published in The Journal of pharmacology and experimental therapeutics (01.10.1998)
Journal Article
3α-Hydroxy-3β-(phenylethynyl)-5β-pregnan-20-ones: Synthesis and Pharmacological Activity of Neuroactive Steroids with High Affinity for GABAA Receptors
Upasani, Ravindra B, Yang, Kevin C, Acosta-Burruel, Manuel, Konkoy, Chris S, McLellan, James A, Woodward, Richard M, Lan, Nancy C, Carter, Richard B, Hawkinson, Jon E
Published in Journal of medicinal chemistry (03.01.1997)
Published in Journal of medicinal chemistry (03.01.1997)
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Steroid inhibition of [3H]SR 95531 binding to the GABAA recognition site
HAWKINSON, J. E, ACOSTA-BURRUEL, M, KIMBROUGH, C. L, GOODNOUGH, D. B, WOOD, P. L
Published in European journal of pharmacology (23.05.1996)
Published in European journal of pharmacology (23.05.1996)
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Journal Article
Synthesis and in Vitro Activity of 3β-Substituted-3α-hydroxypregnan-20-ones: Allosteric Modulators of the GABAA Receptor
Hogenkamp, Derk J, Tahir, S. Hasan, Hawkinson, Jon E, Upasani, Ravi B, Alauddin, Mian, Kimbrough, Catherine L, Acosta-Burruel, Manuel, Whittemore, E. R, Woodward, R. M, Lan, Nancy C, Gee, Kelvin W, Bolger, Michael B
Published in Journal of medicinal chemistry (03.01.1997)
Published in Journal of medicinal chemistry (03.01.1997)
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