Optimization of antimalarial, and anticancer activities of (E)-methyl 2-(7-chloroquinolin-4-ylthio)-3-(4-hydroxyphenyl) acrylate
Romero, Jesús A., Acosta, María E., Gamboa, Neira D., Mijares, Michael R., De Sanctis, Juan B., Charris, Jaime E.
Published in Bioorganic & medicinal chemistry (15.02.2018)
Published in Bioorganic & medicinal chemistry (15.02.2018)
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Synthesis, Antimalarial, Antileishmanial, and Cytotoxicity Activities and Preliminary In Silico ADMET Studies of 2-(7-Chloroquinolin-4-ylamino)ethyl Benzoate Derivatives
Gutiérrez, Joyce E, Ramírez, Hegira, Fernandez-Moreira, Esteban, Acosta, María E, Mijares, Michael R, De Sanctis, Juan Bautista, Gurská, Soňa, Džubák, Petr, Hajdúch, Marián, Labrador-Fagúndez, Liesangerli, Stella, Bruno G, Díaz-Pérez, Luis José, Benaim, Gustavo, Charris, Jaime E
Published in Pharmaceuticals (Basel, Switzerland) (01.12.2023)
Published in Pharmaceuticals (Basel, Switzerland) (01.12.2023)
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Journal Article
Synthesis, β-hematin inhibition studies and antimalarial evaluation of new dehydroxy isoquine derivatives against Plasmodium berghei: A promising antimalarial agent
Valverde, Edgar A., Romero, Angel H., Acosta, María E., Gamboa, Neira, Henriques, Genesis, Rodrigues, Juan R., Ciangherotti, Carlos, López, Simón E.
Published in European journal of medicinal chemistry (25.03.2018)
Published in European journal of medicinal chemistry (25.03.2018)
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Journal Article
Antimalarial, antiproliferative, and apoptotic activity of quinoline-chalcone and quinoline-pyrazoline hybrids. A dual action
Charris, Jaime E., Monasterios, Melina C., Acosta, María E., Rodríguez, Miguel A., Gamboa, Neira D., Martínez, Gricelis P., Rojas, Héctor R., Mijares, Michael R., De Sanctis, Juan B.
Published in Medicinal chemistry research (01.11.2019)
Published in Medicinal chemistry research (01.11.2019)
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Journal Article
Optimization of the synthesis, in silico ADME/Tox profiling studies, and evaluation of the antimalarial activity of (7-chloroquinolin-4-ylthio)alkylbenzoate derivatives
Gutiérrez, Joyce E, Fernandez-Moreira, Esteban, Acosta, María E, Ramírez, Hegira, Charris, Jaime E
Published in Journal of chemical research (01.05.2023)
Published in Journal of chemical research (01.05.2023)
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Journal Article
Synthesis, β-hematin inhibition studies and antimalarial evaluation of dehydroxy isotebuquine derivatives against Plasmodium berghei
Romero, Angel H., Acosta, María E., Gamboa, Neira, Charris, Jaime E., Salazar, José, López, Simón E.
Published in Bioorganic & medicinal chemistry (01.08.2015)
Published in Bioorganic & medicinal chemistry (01.08.2015)
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Analysis of Prevalence and Predictive Factors of Long-Lasting Olfactory and Gustatory Dysfunction in COVID-19 Patients
Callejón-Leblic, María A., Martín-Jiménez, Daniel I., Moreno-Luna, Ramón, Palacios-Garcia, Jose M., Alvarez-Cendrero, Marta, Vizcarra-Melgar, Julissa A., Fernandez-Velez, Carlos, Reyes-Tejero, Isabel M., Maza-Solano, Juan, Gonzalez-Garcia, Jaime, Tena-García, Beatriz, Acosta-Mosquera, María E., Del Cuvillo, Alfonso, Sánchez-Gómez, Serafín
Published in Life (Basel, Switzerland) (17.08.2022)
Published in Life (Basel, Switzerland) (17.08.2022)
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Journal Article
Synthesis, antimalarial, antiproliferative, and apoptotic activities of benzimidazole-5-carboxamide derivatives
Romero, Jesús A., Acosta, María E., Gamboa, Neira D., Mijares, Michael R., De Sanctis, Juan B., Llovera, Ligia J., Charris, Jaime E.
Published in Medicinal chemistry research (01.01.2019)
Published in Medicinal chemistry research (01.01.2019)
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Relationship between serum lipopolysaccharide binding protein levels, disease activity, and clinical characteristics in Paraguayan patients with systemic lupus erythematosus
Losanto, Jhonatan, Langjahr, Patricia, Barrios, Graciela, Paats, Astrid, Acosta de Hetter, María E, de Guillén, Ivalena, Duarte, Margarita, Acosta-Colman, Isabel, Cervera, Ricard
Published in Lupus (01.11.2021)
Published in Lupus (01.11.2021)
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[(7-chloroquinolin-4-yl)amino]acetophenones and their copper(II) derivatives: Synthesis, characterization, computational studies and antimalarial activity
de J Parra, Yonathan, Andueza L, Felix D, Ferrer M, Rosa E, Bruno Colmenarez, Julia, Acosta, María E, Charris, Jaime, Rosenthal, Philip J, Gut, Jiri
Published in EXCLI journal (01.01.2019)
Published in EXCLI journal (01.01.2019)
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Epidemiology of the Cnidarian Physalia physalis stings attended at a health care center in beaches of Adicora, Venezuela
Cazorla-Perfetti, Dalmiro J, Loyo, Jesus, Lugo, Lusneida, Acosta, María E, Morales, Pedro, Haddad, Vidal, Rodriguez-Morales, Alfonso J
Published in Travel medicine and infectious disease (01.09.2012)
Published in Travel medicine and infectious disease (01.09.2012)
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Adaptative Strategies in Gymnocalycium Species (Cactaceae) and the Presence of Ectomycorrhizae Associated with Survival in Arid Environments
Soto Acosta, María E, Perea, Mario, Ruiz, Ana I, Hilal, Mirna, Albornoz, Patricia L, Isla, María I
Published in Plants (Basel) (26.07.2023)
Published in Plants (Basel) (26.07.2023)
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Exposure to severe urban air pollution influences cognitive outcomes, brain volume and systemic inflammation in clinically healthy children
Calderón-Garcidueñas, Lilian, Engle, Randall, Mora-Tiscareño, Antonieta, Styner, Martin, Gómez-Garza, Gilberto, Zhu, Hongtu, Jewells, Valerie, Torres-Jardón, Ricardo, Romero, Lina, Monroy-Acosta, Maria E., Bryant, Christopher, González-González, Luis Oscar, Medina-Cortina, Humberto, D’Angiulli, Amedeo
Published in Brain and cognition (01.12.2011)
Published in Brain and cognition (01.12.2011)
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Synthesis of Trans- and cis-2-acetyl-3-phenyl-3,3a,4,5-tetrahydro-2H-benzo[g] Indazoles: Evaluation as Inhibitors of β-hematin Formation
Aparicio, Daniel A., Lobo, Gricela M., Sánchez, Jennifer L., Monasterios, Melina C., Acosta, María E., De Lima, Lola, Llovera, Ligia J., Ángel, Jorge E., Charris, Jaime E.
Published in Journal of chemical research (01.11.2017)
Published in Journal of chemical research (01.11.2017)
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Journal Article
Synthesis, antimalarial and antileishmanial activity of novel 13-benzyl-15,16-bisnorlabdane derivatives
Salazar, Franklin J., Quintero, Alberto, Gamboa de Dominguezc, Neira, Concepcion, Juan L., Acosta, Maria E., Tropper, Eleonora, Villamizar, Jose E.
Published in Journal of chemical research (01.11.2013)
Published in Journal of chemical research (01.11.2013)
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Identificación de Fusarium oxysporum como agente causal de la podredumbre del pedúnculo de limón en Tucumán (Argentina) y su control
Gabriela M. Fogliata, Cristina V. Martínez, María E. Acosta, María L. Muñoz, L. Daniel Ploper
Published in Revista Industrial y Agrícola de Tucumán (01.12.2018)
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Published in Revista Industrial y Agrícola de Tucumán (01.12.2018)
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Trends in school‐neighbourhood inequalities and youth obesity: Repeated cross‐sectional analyses of the public schools in the state of California
Matsuzaki, Mika, Sanchez‐Vaznaugh, Emma V., Alexovitz, Kelsey, Acosta, Maria E., Sánchez, Brisa N.
Published in Pediatric obesity (01.03.2023)
Published in Pediatric obesity (01.03.2023)
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