Discovery of the Soluble Guanylate Cyclase Stimulator Vericiguat (BAY 1021189) for the Treatment of Chronic Heart Failure
Follmann, Markus, Ackerstaff, Jens, Redlich, Gorden, Wunder, Frank, Lang, Dieter, Kern, Armin, Fey, Peter, Griebenow, Nils, Kroh, Walter, Becker-Pelster, Eva-Maria, Kretschmer, Axel, Geiss, Volker, Li, Volkhart, Straub, Alexander, Mittendorf, Joachim, Jautelat, Rolf, Schirok, Hartmut, Schlemmer, Karl-Heinz, Lustig, Klemens, Gerisch, Michael, Knorr, Andreas, Tinel, Hanna, Mondritzki, Thomas, Trübel, Hubert, Sandner, Peter, Stasch, Johannes-Peter
Published in Journal of medicinal chemistry (22.06.2017)
Published in Journal of medicinal chemistry (22.06.2017)
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Formal total synthesis of (-)-haouamine A
Fuerstner, Alois, Ackerstaff, Jens
Published in Chemical communications (Cambridge, England) (01.01.2008)
Published in Chemical communications (Cambridge, England) (01.01.2008)
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Design and Preclinical Characterization Program toward Asundexian (BAY 2433334), an Oral Factor XIa Inhibitor for the Prevention and Treatment of Thromboembolic Disorders
Roehrig, Susanne, Ackerstaff, Jens, Jiménez Núñez, Eloísa, Teller, Henrik, Ellerbrock, Pascal, Meier, Katharina, Heitmeier, Stefan, Tersteegen, Adrian, Stampfuss, Jan, Lang, Dieter, Schlemmer, Karl-Heinz, Schaefer, Martina, Gericke, Kersten M., Kinzel, Tom, Meibom, Daniel, Schmidt, Martina, Gerdes, Christoph, Follmann, Markus, Hillisch, Alexander
Published in Journal of medicinal chemistry (14.09.2023)
Published in Journal of medicinal chemistry (14.09.2023)
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A versatile protocol for Stille-Migita cross coupling reactions
Fuerstner, Alois, Funel, Jacques-Alexis, Tremblay, Martin, Bouchez, Laure C., Nevado, Cristina, Waser, Mario, Ackerstaff, Jens, Stimson, Christopher C.
Published in Chemical communications (Cambridge, England) (01.01.2008)
Published in Chemical communications (Cambridge, England) (01.01.2008)
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SALTS OF 1-(3-METHYL-2-OXO-2,3-DIHYDRO-1,3-BENZOXAZOL-6-YL)-2,4-DIOXO-3-[(1R)-4-(TRIFLUORMETHYL)-2,3-DIHYDRO-1H-INDEN-1-YL]-1,2,3,4-TETRAHYDROPYRIMIDIN-5-CARBOXYLIC ACID
HINZ MARTIN HOLGER, JESKE MARIO, OLENIK BRITTA, KEIL BIRGIT, FUERSTNER CHANTAL, ACKERSTAFF JENS
Year of Publication 05.07.2016
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Year of Publication 05.07.2016
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치환된 옥소피리딘 유도체
MEIER KATHARINA, ELLERBROCK PASCAL, LANG DIETER, JIMENEZ NUNEZ ELOISA, ROEHRIG SUSANNE, HILLISCH ALEXANDER, STAMPFUSS JAN, MEIBOM DANIEL, HEITMEIER STEFAN, TERSTEEGEN ADRIAN, ACKERSTAFF JENS
Year of Publication 13.03.2018
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Year of Publication 13.03.2018
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아미도-치환된 시클로헥산 유도체
SIEGEL FRANZISKA, LIENAU PHILIP, KOPPITZ MARCUS, BUCHGRABER PHILIPP, BENDER ECKHARD, VON NUSSBAUM FRANZ, LIU NINGSHU, EIS KNUT, SUELZLE DETLEV, BAIRLEIN MICHAELA, LI VOLKHART, ACKERSTAFF JENS, WAGNER SARAH, HOLTON SIMON, HERBERT SIMON ANTHONY
Year of Publication 08.01.2018
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Year of Publication 08.01.2018
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TNKS1 / TNKS2 - AMIDO-SUBSTITUTED AZOLE COMPOUNDS AS INHIBITORS OF TNKS1 AND/OR TNKS2
LIENAU PHILIP, SIEGEL FRANZISKA, GOLZ STEFAN, BENDER ECKHARD, BUCHGRABER PHILIPP, LIU NINGSHU, EIS KNUT, BAUSER MARCUS, SUELZLE DETLEV, BAIRLEIN MICHAELA, ACKERSTAFF JENS, WAGNER SARAH, BASTING DANIEL, HOLTON SIMON, LI VOLKHART MIN JIAN, BALINT JOZSEF
Year of Publication 21.11.2016
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Year of Publication 21.11.2016
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SUBSTITUTED PHENYLALANINE DERIVATIVES
ELLERMANN MANUEL, HILLISCH ALEXANDER, TERJUNG CARSTEN, ROEHN ULRIKE, STRASSBURGER JULIA, GERDES CHRISTOPH, SCHMIDT MARTINA VICTORIA, TERSTEEGEN ADRIAN, SANDMANN STEFFEN, ACKERSTAFF JENS, SPERZEL MICHAEL, WENDT ASTRID, WEBSTER ROBERT ALAN, ROEHRIG SUSANNE, BUCHMUELLER ANJA, HEITMEIER STEFAN, BEYER KRISTIN, SCHAEFER MARTINA
Year of Publication 07.06.2016
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Year of Publication 07.06.2016
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RING-FUSED PYRIMIDINES AND TRIAZINES AND USE THEREOF FOR THE TREATMENT AND/OR PROPHYLAXIS OF CARDIOVASCULAR DISEASES
WUNDER FRANK, REDLICH GORDEN, KNORR ANDREAS, BAERFACKER LARS, LI VOLKHART MIN JIAN, GRIEBENOW NILS, FOLLMANN MARKUS, STASCH JOHANNES PETER, KROH WALTER, ACKERSTAFF JENS
Year of Publication 04.12.2013
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Year of Publication 04.12.2013
Patent
SUBSTITUTED 5-FLUORO-1H-PYRAZOLOPYRIDINES AND USE THEREOF
KNORR ANDREAS, JAUTELAT ROLF, GRIEBENOW NILS, FOLLMANN MARKUS, STASCH JOHANNES PETER, KROH WALTER, SCHLEMMER KARL HEINZ, ACKERSTAFF JENS, BECKER EVA MARIA, WUNDER FRANK, BIERER DONALD, REDLICH GORDEN, HARTMANN ELKE, LI VOLKHART MIN JIAN, MITTENDORF JOACHIM
Year of Publication 22.10.2013
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Year of Publication 22.10.2013
Patent
Versatile Phosphite Ligands Based on Silsesquioxane Backbones
van der Vlugt, Jarl Ivar, Ackerstaff, Jens, Dijkstra, Tessa W., Mills, Allison M., Kooijman, Huub, Spek, Anthony L., Meetsma, Auke, Abbenhuis, Hendrikus C. L., Vogt, Dieter
Published in Advanced synthesis & catalysis (01.03.2004)
Published in Advanced synthesis & catalysis (01.03.2004)
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A Silsesquioxane-Based Diphosphinite Ligand: Synthesis, DFT Study, and Coordination Chemistry
van der Vlugt, Jarl Ivar, Fioroni, Marco, Ackerstaff, Jens, Hanssen, Rob W. J. M, Mills, Allison M, Spek, Anthony L, Meetsma, Auke, Abbenhuis, Hendrikus C. L, Vogt, Dieter
Published in Organometallics (08.12.2003)
Published in Organometallics (08.12.2003)
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SALTS OF 1-(3-METHYL-2-OXO-2,3-DIHYDRO-1,3-BENZOXAZOL-6-YL)-2,4- DIOXO-3-[(1R)-4-(TRIFLUORMETHYL)-2,3-DIHYDRO-1H-INDEN-1-YL)-1,2,3,4- TETRAHYDROPYRIMIDIN-5-CARBOXYLIC ACID
HINZ, MARTIN-HOLGER, FURSTNER, CHANTAL, KEIL, BIRGIT, OLENIK, BRITTA, ACKERSTAFF, JENS, JESKE, MARIO
Year of Publication 29.03.2022
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Year of Publication 29.03.2022
Patent
SALTS OF 1-(3-METHYL-2-OXO-2,3-DIHYDRO-1,3-BENZOXAZOL-6-YL)-2,4-DIOXO-3-[(1R)-4-(TRIFLUORMETHYL)-2,3-DIHYDRO-1H-INDEN-1-YL]-1,2,3,4-TETRAHYDROPYRIMIDIN-5-CARBOXYLIC ACID
HINZ, MARTIN-HOLGER, KEIL, BIRGIT, FURSTNER, CHANTAL, OLENIK, BRITTA, JESKE, MARIO, ACKERSTAFF, JENS
Year of Publication 22.03.2022
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Year of Publication 22.03.2022
Patent
Substituted 5-fluoro-1H-pyrazolopyridines and their use
Wunder, Frank, Redlich, Gorden, Hartmann, Elke, Mittendorf, Joachim, Schlemmer, Karl-Heinz, Becker, Eva-Maria, Bierer, Donald, Griebenow, Nils, Jautelat, Rolf, Follmann, Markus, Kroh, Walter, Li, Volkhart Min-Jian, Stasch, Johannes-Peter, Knorr, Andreas, Ackerstaff, Jens
Year of Publication 20.08.2024
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Year of Publication 20.08.2024
Patent
SUBSTITUTED OXOPYRIDINE DERIVATIVES
ADRIAN TERSTEEGEN, STEFAN HEITMEIER, KATHARINA MEIER, ELOISA JIMENEZ NUNEZ, ALEXANDER HILLISCH, PASCAL ELLERBROCK, DANIEL MEIBOM, SUSANNE ROHRIG, ACKERSTAFF, JENS, DIETER LANG, JAN STAMPFU?
Year of Publication 25.04.2023
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Year of Publication 25.04.2023
Patent