Metabolomic analysis of a selective ABCA1 inducer in obesogenic challenge provides a rationale for therapeutic development
Lewandowski, Cutler T., Khan, Md.Wasim, BenAissa, Manel, Dubrovskyi, Oleksii, Ackerman-Berrier, Martha, LaDu, Mary Jo, Layden, Brian T., Thatcher, Gregory R.J.
Published in EBioMedicine (01.04.2021)
Published in EBioMedicine (01.04.2021)
Get full text
Journal Article
Synthesis, Optimization, and Structure–Activity Relationships of Nicotinamide Phosphoribosyltransferase (NAMPT) Positive Allosteric Modulators (N-PAMs)
Shen, Zhengnan, Ratia, Kiira, Krider, Isabella, Ackerman-Berrier, Martha, Penton, Christopher, Musku, Soumya Reddy, Gordon-Blake, Jesse M., Laham, Megan S., Christie, Nicholas, Ma, Nina, Fu, Jiqiang, Xiong, Rui, Courey, Jenna M., Velma, Ganga Reddy, Thatcher, Gregory R. J.
Published in Journal of medicinal chemistry (28.12.2023)
Published in Journal of medicinal chemistry (28.12.2023)
Get full text
Journal Article
Nonlipogenic ABCA1 Inducers (NLAI) for Alzheimer's Disease Validated in a Mouse Model Expressing Human APOE3/APOE4
Velma, Ganga Reddy, Laham, Megan S, Lewandowski, Cutler, Valencia-Olvera, Ana C, Balu, Deebika, Moore, Annabelle, Ackerman-Berrier, Martha, Rychetsky, Pavel, Penton, Christopher, Musku, Soumya Reddy, Annadurai, Anandhan, Sulaiman, Maha Ibrahim, Ma, Nina, J Thatcher, Gregory R
Published in Journal of medicinal chemistry (12.09.2024)
Published in Journal of medicinal chemistry (12.09.2024)
Get full text
Journal Article
Mechanism of Allosteric Modulation of Nicotinamide Phosphoribosyltransferase to Elevate Cellular NAD
Ratia, Kiira M., Shen, Zhengnan, Gordon-Blake, Jesse, Lee, Hyun, Laham, Megan S., Krider, Isabella S., Christie, Nicholas, Ackerman-Berrier, Martha, Penton, Christopher, Knowles, Natalie G., Musku, Soumya Reddy, Fu, Jiqiang, Velma, Ganga Reddy, Xiong, Rui, Thatcher, Gregory R. J.
Published in Biochemistry (Easton) (21.02.2023)
Published in Biochemistry (Easton) (21.02.2023)
Get full text
Journal Article
Nicotinamide Phosphoribosyltransferase Positive Allosteric Modulators Attenuate Neuronal Oxidative Stress
Gordon-Blake, Jesse, Ratia, Kiira, Weidig, Victoria, Velma, Ganga Reddy, Ackerman-Berrier, Martha, Penton, Christopher, Musku, Soumya Reddy, Alves, Erick T.M., Driver, Tom, Tai, Leon, Thatcher, Gregory R. J.
Published in ACS medicinal chemistry letters (08.02.2024)
Published in ACS medicinal chemistry letters (08.02.2024)
Get full text
Journal Article
The mechanism of nicotinamide phosphoribosyltransferase whereby positive allosteric modulation elevates cellular NAD
Ratia, Kiira M, Shen, Zhengnan, Gordon-Blake, Jesse, Lee, Hyun, Laham, Megan S, Krider, Isabella S, Christie, Nicholas, Ackerman-Berrier, Martha S, Penton, Christopher, Knowles, Natalie G, Soumya Reddy Musku, Fu, Jiqiang, Ganga Reddy Musku, Xiong, Rui, Thatcher, Gregory R J
Published in bioRxiv (22.10.2022)
Published in bioRxiv (22.10.2022)
Get full text
Paper
Efficient Discovery of Inhibitory Ligands for Diverse Targets from a Small Combinatorial Chemical Library of Chimeric Molecules
Thorpe, David S., Edith Chan, A.W., Binnie, Alan, Chen, L.Charlie, Robinson, Anna, Spoonamore, James, Rodwell, David, Wade, Shelly, Wilson, Sydney, Ackerman-Berrier, Martha, Yeoman, Helen, Walle, Stefan, Wu, Qinyuan (Quincey), Wertman, Kenneth F.
Published in Biochemical and biophysical research communications (09.12.1999)
Published in Biochemical and biophysical research communications (09.12.1999)
Get full text
Journal Article
7-SUBSTITUTED AZA-INDAZOLES, COMPOSITIONS CONTAINING SAME, PRODUCTION METHOD AND USE THEREOF
SMRCINA, MARTIN, BJERGARDE, KIRSTEN, SOUAILLE, CATHERINE, ACKERMAN-BERRIER, MARTHA, BACQUE, ERIC, VIVIANI, FABRICE, TABART, MICHEL, RONAN, BAPTISTE, NAIR, ANIL, LEROY, VINCENT, PATEK, MARCEL, DODSON, MARK
Year of Publication 16.04.2014
Get full text
Year of Publication 16.04.2014
Patent
SUBSTITUTED 7-AZAINDAZOLES, COMPOSITIONS CONTAINING THEM, PRODUCTION PROCESS AND USE
MARTHA ACKERMAN-BERRIER, BAPTISTE RONAN, CATHERINE SOUAILLE, MARCEL PATEK, MARTIN SMRCINA, ERIC BACQUE, MICHEL TABART, ANIL NAIR, KRISTEN BJERGARDE, MARK DODSON, FABRICE VIVIANI, VINCENT LEROY
Year of Publication 14.12.2012
Get full text
Year of Publication 14.12.2012
Patent
7-substituted aza-indazoles, compositions containing same, production method and use thereof
SMRCINA, MARTIN, BJERGARDE, KRISTEN, SOUAILLE, CATHERINE, ACKERMAN-BERRIER, MARTHA, VIVIANI, FABRICE, BACQUE, ERIC, TABART, MICHEL, RONAN, BAPTISTE, NAIR, ANIL, LEROY, VINCENT, PATEK, MARCEL, DODSON, MARK
Year of Publication 23.08.2012
Get full text
Year of Publication 23.08.2012
Patent
7-substituted aza-indazoles, compositions containing same, production method and use thereof
Bjergarde, Kirsten, Nair, Anil, Patek, Marcel, Ackerman-Berrier, Martha, Smrcina, Martin, Bacque, Eric, Tabart, Michel, Ronan, Baptiste, Leroy, Vincent, Viviani, Fabrice, Dodson, Mark, Souaille, Catherine
Year of Publication 15.11.2011
Get full text
Year of Publication 15.11.2011
Patent
7-substituted aza-indazoles, compositions containing same, production method and use thereof
BJERGARDE KIRSTEN, ACKERMAN-BERRIER MARTHA, NAIR ANIL, VIVIANI FABRICE, TABART MICHEL, SOUAILLE CATHERINE, SMRCINA MARTIN, BACQUE ERIC, LEROY VINCENT, PATEK MARCEL, RONAN BAPTISTE, DODSON MARK
Year of Publication 15.11.2011
Get full text
Year of Publication 15.11.2011
Patent
7-SUBSTITUTED AZA-INDAZOLES, COMPOSITION CONTAINING SAME, PRODUCTION METHOD AND USE THEREOF
BJERGARDE KIRSTEN, ACKERMAN-BERRIER MARTHA, NAIR ANIL, VIVIANI FABRICE, TABART MICHEL, SOUAILLE CATHERINE, SMRCINA MARTIN, BACQUE ERIC, LEROY VINCENT, PATEK MARCEL, RONAN BAPTISTE, DODSON MARK
Year of Publication 10.05.2011
Get full text
Year of Publication 10.05.2011
Patent
7-substituted aza-indazoles, compositions containing same, production method and use thereof
SMRCINA, MARTIN, BJERGARDE, KRISTEN, SOUAILLE, CATHERINE, ACKERMAN-BERRIER, MARTHA, BACQUE, ERIC, VIVIANI, FABRICE, TABART, MICHEL, RONAN, BAPTISTE, NAIR, ANIL, LEROY, VINCENT, PATEK, MARCEL, DODSON, MARK
Year of Publication 31.03.2011
Get full text
Year of Publication 31.03.2011
Patent
7- AZA- INDAZOLES SUSTITUIDOS, COMPOSICIONES QUE LOS CONTIENEN, PROCEDIMIENTO DE FABRICACION Y SU UTILIZACION
MARTHA ACKERMAN-BERRIER, BAPTISTE RONAN, CATHERINE SOUAILLE, MARCEL PATEK, MARTIN SMRCINA, ANIL NAIR, KRISTEN BJERGARDE, ERIC BAQUE, MARK DODSON, MICHAEL TABART, VINCENT LEROY, FABRICE VIVIANI
Year of Publication 09.11.2010
Get full text
Year of Publication 09.11.2010
Patent
7-substituted aza-indazoles, compositions containing same, production method and use thereof
SMRCINA, MARTIN, BJERGARDE, KIRSTEN, SOUAILLE, CATHERINE, ACKERMAN-BERRIER, MARTHA, BACQUE, ERIC, VIVIANI, FABRICE, TABART, MICHEL, RONAN, BAPTISTE, NAIR, ANIL, LEROY, VINCENT, PATEK, MARCEL, DODSON, MARK
Year of Publication 25.11.2009
Get full text
Year of Publication 25.11.2009
Patent
7-SUBSTITUTED AZA-INDAZOLES, COMPOSITIONS CONTAINING SAME, PRODUCTION METHOD AND USE THEREOF
SMRCINA, MARTIN, BJERGARDE, KIRSTEN, SOUAILLE, CATHERINE, ACKERMAN-BERRIER, MARTHA, BACQUE, ERIC, VIVIANI, FABRICE, TABART, MICHEL, RONAN, BAPTISTE, NAIR, ANIL, LEROY, VINCENT, PATEK, MARCEL, DODSON, MARK
Year of Publication 21.08.2009
Get full text
Year of Publication 21.08.2009
Patent
7-SUBSTITUTED AZA-INDAZOLES, COMPOSITIONS CONTAINING SAME, PRODUCTION METHOD AND USE THEREOF
DODSON,MARK, PATEK,MARCEL, BACQUE,ERIC, SOUAILLE,CATHERINE, RONAN,BAPTISTE, VIVIANI,FABRICE, LEROY,VINCENT, SMRCINA,MARTIN, NAIR,ANIL, BJERGARDE,KIRSTEN, TABART,MICHEL, ACKERMAN-BERRIER,MARTHA
Year of Publication 14.07.2009
Get full text
Year of Publication 14.07.2009
Patent
7-SUBSTITUTED AZA-INDAZOLES, COMPOSITIONS CONTAINING SAME, PRODUCTION METHOD AND USE THEREOF
SMRCINA, MARTIN, BJERGARDE, KIRSTEN, SOUAILLE, CATHERINE, ACKERMAN-BERRIER, MARTHA, BACQUE, ERIC, VIVIANI, FABRICE, TABART, MICHEL, RONAN, BAPTISTE, NAIR, ANIL, LEROY, VINCENT, PATEK, MARCEL, DODSON, MARK
Year of Publication 22.09.2015
Get full text
Year of Publication 22.09.2015
Patent
7-Substituted Aza-Indazoles, Compositions Containing Same, Production Method and Use Thereof
BJERGARDE KIRSTEN, ACKERMAN-BERRIER MARTHA, NAIR ANIL, VIVIANI FABRICE, TABART MICHEL, SOUAILLE CATHERINE, SMRCINA MARTIN, BACQUE ERIC, LEROY VINCENT, PATEK MARCEL, RONAN BAPTISTE, DODSON MARK
Year of Publication 31.07.2008
Get full text
Year of Publication 31.07.2008
Patent