Two-Photon “Caging” Groups: Effect of Position Isomery on the Photorelease Properties of Aminoquinoline-Derived Photolabile Protecting Groups
Tran, Christine, Gallavardin, Thibault, Petit, Morgane, Slimi, Riadh, Dhimane, Hamid, Blanchard-Desce, Mireille, Acher, Francine C, Ogden, David, Dalko, Peter I
Published in Organic letters (06.02.2015)
Published in Organic letters (06.02.2015)
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Substitution Effect on the One- and Two-photon Sensitivity of DMAQ “Caging” Groups
Petit, Morgane, Tran, Christine, Roger, Thomas, Gallavardin, Thibault, Dhimane, Hamid, Palma-Cerda, Francisco, Blanchard-Desce, Mireille, Acher, Francine C, Ogden, David, Dalko, Peter I
Published in Organic letters (21.12.2012)
Published in Organic letters (21.12.2012)
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Molecular determinants of agonist selectivity in glutamate-gated chloride channels which likely explain the agonist selectivity of the vertebrate glycine and GABAA-ρ receptors
Blarre, Thomas, Bertrand, Hugues-Olivier, Acher, Francine C, Kehoe, JacSue
Published in PloS one (26.09.2014)
Published in PloS one (26.09.2014)
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l-(+)-2-Amino-4-thiophosphonobutyric Acid (l-thioAP4), a New Potent Agonist of Group III Metabotropic Glutamate Receptors: Increased Distal Acidity Affords Enhanced Potency
Selvam, Chelliah, Goudet, Cyril, Oueslati, Nadia, Pin, Jean-Philippe, Acher, Francine C
Published in Journal of medicinal chemistry (20.09.2007)
Published in Journal of medicinal chemistry (20.09.2007)
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Design, Synthesis, Pharmacology, and In Silico Studies of (1 S ,2 S ,3 S )-2-(( S )-Amino(carboxy)methyl)-3-(carboxymethyl)cyclopropane-1-carboxylic Acid (LBG30300): A Picomolar Potency Subtype-Selective mGlu 2 Receptor Agonist
Liu, Na, Eshak, Floriane, Malhaire, Fanny, Brabet, Isabelle, Prézeau, Laurent, Renard, Emma, Pin, Jean-Philippe, Acher, Francine C, Staudt, Markus, Bunch, Lennart
Published in Journal of medicinal chemistry (25.01.2024)
Published in Journal of medicinal chemistry (25.01.2024)
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Metabotropic glutamate receptor orthosteric ligands and their binding sites
Acher, Francine C., Cabayé, Alexandre, Eshak, Floriane, Goupil-Lamy, Anne, Pin, Jean-Philippe
Published in Neuropharmacology (15.02.2022)
Published in Neuropharmacology (15.02.2022)
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Design, Synthesis, Pharmacology, and In Silico Studies of (1S,2S,3S)‑2-((S)‑Amino(carboxy)methyl)-3-(carboxymethyl)cyclopropane-1-carboxylic Acid (LBG30300): A Picomolar Potency Subtype-Selective mGlu2 Receptor Agonist
Liu, Na, Eshak, Floriane, Malhaire, Fanny, Brabet, Isabelle, Prézeau, Laurent, Renard, Emma, Pin, Jean-Philippe, Acher, Francine C., Staudt, Markus, Bunch, Lennart
Published in Journal of medicinal chemistry (25.01.2024)
Published in Journal of medicinal chemistry (25.01.2024)
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Epitope Identification of an mGlu5 Receptor Nanobody Using Physics-Based Molecular Modeling and Deep Learning Techniques
Eshak, Floriane, Pion, Léo, Scholler, Pauline, Nevoltris, Damien, Chames, Patrick, Rondard, Philippe, Pin, Jean-Philippe, Acher, Francine C., Goupil-Lamy, Anne
Published in Journal of chemical information and modeling (10.06.2024)
Published in Journal of chemical information and modeling (10.06.2024)
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Novel Inhibitory Site Revealed by XAP044 Mode of Action on the Metabotropic Glutamate 7 Receptor Venus Flytrap Domain
Cristiano, Nunzia, Cabayé, Alexandre, Brabet, Isabelle, Glatthar, Ralf, Tora, Amelie, Goudet, Cyril, Bertrand, Hugues-Olivier, Goupil-Lamy, Anne, Flor, Peter J., Pin, Jean-Philippe, McCort-Tranchepain, Isabelle, Acher, Francine C.
Published in Journal of medicinal chemistry (25.07.2024)
Published in Journal of medicinal chemistry (25.07.2024)
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Asc-1 Transporter (SLC7A10): Homology Models And Molecular Dynamics Insights Into The First Steps Of The Transport Mechanism
Mikou, Afaf, Cabayé, Alexandre, Goupil, Anne, Bertrand, Hugues-Olivier, Mothet, Jean-Pierre, Acher, Francine C.
Published in Scientific reports (28.02.2020)
Published in Scientific reports (28.02.2020)
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Amino Acids Bearing Aromatic or Heteroaromatic Substituents as a New Class of Ligands for the Lysosomal Sialic Acid Transporter Sialin
Dubois, Lilian, Pietrancosta, Nicolas, Cabaye, Alexandre, Fanget, Isabelle, Debacker, Cécile, Gilormini, Pierre-André, Dansette, Patrick M, Dairou, Julien, Biot, Christophe, Froissart, Roseline, Goupil-Lamy, Anne, Bertrand, Hugues-Olivier, Acher, Francine C, McCort-Tranchepain, Isabelle, Gasnier, Bruno, Anne, Christine
Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
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Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites
Selvam, Chelliah, Lemasson, Isabelle A, Brabet, Isabelle, Oueslati, Nadia, Karaman, Berin, Cabaye, Alexandre, Tora, Amélie S, Commare, Bruno, Courtiol, Tiphanie, Cesarini, Sara, McCort-Tranchepain, Isabelle, Rigault, Delphine, Mony, Laetitia, Bessiron, Thomas, McLean, Heather, Leroux, Frédéric R, Colobert, Françoise, Daniel, Hervé, Goupil-Lamy, Anne, Bertrand, Hugues-Olivier, Goudet, Cyril, Pin, Jean-Philippe, Acher, Francine C
Published in Journal of medicinal chemistry (08.03.2018)
Published in Journal of medicinal chemistry (08.03.2018)
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A Virtual Screening Hit Reveals New Possibilities for Developing Group III Metabotropic Glutamate Receptor Agonists
Selvam, Chelliah, Oueslati, Nadia, Lemasson, Isabelle A, Brabet, Isabelle, Rigault, Delphine, Courtiol, Tiphanie, Cesarini, Sara, Triballeau, Nicolas, Bertrand, Hugues-Olivier, Goudet, Cyril, Pin, Jean-Philippe, Acher, Francine C
Published in Journal of medicinal chemistry (08.04.2010)
Published in Journal of medicinal chemistry (08.04.2010)
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The antipsychotic-like effects of the mGlu group III orthosteric agonist, LSP1-2111, involves 5-HT1A signalling
Wierońska, Joanna M., Acher, Francine C., Sławińska, Anna, Gruca, Piotr, Łasoń-Tyburkiewicz, Magdalena, Papp, Mariusz, Pilc, Andrzej
Published in Psychopharmacology (01.06.2013)
Published in Psychopharmacology (01.06.2013)
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Design, synthesis and biological evaluation of small-azo-dyes as potent Vesicular Glutamate Transporters inhibitors
Favre-Besse, Franck-Cyril, Poirel, Odile, Bersot, Tiphaine, Kim-Grellier, Elodie, Daumas, Stephanie, El Mestikawy, Salah, Acher, Francine C., Pietrancosta, Nicolas
Published in European journal of medicinal chemistry (06.05.2014)
Published in European journal of medicinal chemistry (06.05.2014)
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