Synthetic and Receptor Signaling Explorations of the Mitragyna Alkaloids: Mitragynine as an Atypical Molecular Framework for Opioid Receptor Modulators
Kruegel, Andrew C, Gassaway, Madalee M, Kapoor, Abhijeet, Váradi, András, Majumdar, Susruta, Filizola, Marta, Javitch, Jonathan A, Sames, Dalibor
Published in Journal of the American Chemical Society (01.06.2016)
Published in Journal of the American Chemical Society (01.06.2016)
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Journal Article
Molecular mechanism of setron-mediated inhibition of full-length 5-HT3A receptor
Basak, Sandip, Gicheru, Yvonne, Kapoor, Abhijeet, Mayer, Megan L., Filizola, Marta, Chakrapani, Sudha
Published in Nature communications (19.07.2019)
Published in Nature communications (19.07.2019)
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Journal Article
Clinical development times for innovative drugs
Brown, Dean G., Wobst, Heike J., Kapoor, Abhijeet, Kenna, Leslie A., Southall, Noel
Published in Nature reviews. Drug discovery (01.11.2022)
Published in Nature reviews. Drug discovery (01.11.2022)
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Journal Article
Structure-based characterization of novel TRPV5 inhibitors
Hughes, Taylor Et, Del Rosario, John Smith, Kapoor, Abhijeet, Yazici, Aysenur Torun, Yudin, Yevgen, Fluck, 3rd, Edwin C, Filizola, Marta, Rohacs, Tibor, Moiseenkova-Bell, Vera Y
Published in eLife (25.10.2019)
Published in eLife (25.10.2019)
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Journal Article
Clinical development times for innovative drugs
Brown, Dean G, Wobst, Heike J, Kapoor, Abhijeet, Kenna, Leslie A, Southall, Noel
Published in Nature reviews. Drug discovery (01.11.2022)
Published in Nature reviews. Drug discovery (01.11.2022)
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Journal Article
Phenotype plasticity and altered sensitivity to chemotherapeutic agents in aggressive prostate cancer cells
Paxson, Allan I, Chang, Loren H, Gard, Jaime M C, Harryman, William L, Nelson, Colin S, Salmon, Stella B, Marr, Kendra D, Wachsmuth, Leah M, Ramanathan, Anita, Ran, Jing, Kapoor, Abhijeet, Marugan, Juan J, Henderson, Mark J, Sanchez, Tino W, Cress, Anne E
Published in Frontiers in cell and developmental biology (2023)
Published in Frontiers in cell and developmental biology (2023)
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Journal Article
Differential dynamics of RAS isoforms in GDP- and GTP-bound states
Kapoor, Abhijeet, Travesset, Alex
Published in Proteins, structure, function, and bioinformatics (01.06.2015)
Published in Proteins, structure, function, and bioinformatics (01.06.2015)
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Journal Article
Membrane recognition and substrate binding mechanism of PIP4Kγ kinase from molecular simulations
Kapoor, Abhijeet, Henderson, Mark J., Marugan, Juan, Southall, Noel
Published in Biophysical journal (11.02.2022)
Published in Biophysical journal (11.02.2022)
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Journal Article
Identification of a peptide that disrupts hADA3-E6 interaction with implications in HPV induced cancer therapy
Chand, Vaibhav, Kapoor, Abhijeet, Kundu, Suman, Nag, Alo
Published in Life sciences (1973) (01.01.2022)
Published in Life sciences (1973) (01.01.2022)
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Journal Article
Folding and stability of helical bundle proteins from coarse-grained models
Kapoor, Abhijeet, Travesset, Alex
Published in Proteins, structure, function, and bioinformatics (01.07.2013)
Published in Proteins, structure, function, and bioinformatics (01.07.2013)
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Journal Article
Structural elucidation of RXFP2 allosteric agonist (compound-6641) binding: A computational and experimental approach
Kapoor, Abhijeet, Esteban-Lopez, Maria, Wilson, Kenneth J., Agoulnik, Alexander I., Henderson, Mark J., Marugan, Juan J.
Published in Biophysical journal (08.02.2024)
Published in Biophysical journal (08.02.2024)
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Journal Article
Dynamic and Kinetic Elements of µ-Opioid Receptor Functional Selectivity
Kapoor, Abhijeet, Martinez-Rosell, Gerard, Provasi, Davide, de Fabritiis, Gianni, Filizola, Marta
Published in Scientific reports (12.09.2017)
Published in Scientific reports (12.09.2017)
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Journal Article