Loading…
Loading…
Monoselective Histone Deacetylase 6 PROTAC Degrader Shows In Vivo Tractability
Garcha, Harsimran K., Olaoye, Olasunkanmi O., Sedighi, Abootaleb, Pölöske, Daniel, Hariri, Pearla, Yu, Wenlong, Abdallah, Diaaeldin I., Moriggl, Richard, de Araujo, Elvin D., Gunning, Patrick T.
Published in Journal of medicinal chemistry (27.03.2025)
Published in Journal of medicinal chemistry (27.03.2025)
Get full text
Journal Article
Loading…
Microwave-assisted synthesis of pomalidomide building blocks for rapid PROTAC and molecular glue development
Abdallah, Diaaeldin I, Israelian, Johan, Hasan, Lina S, Patel, Naman H, Keillor, Jeffrey W, Wright, Timothy B, Saqib, Bilal, de Araujo, Elvin D, Gunning, Patrick T
Published in Chemical communications (Cambridge, England) (19.03.2025)
Published in Chemical communications (Cambridge, England) (19.03.2025)
Get full text
Journal Article
Loading…
Hyperactive STAT5 hijacks T cell receptor signaling and drives immature T cell acute lymphoblastic leukemia
Suske, Tobias, Sorger, Helena, Manhart, Gabriele, Ruge, Frank, Prutsch, Nicole, Zimmerman, Mark W., Eder, Thomas, Abdallah, Diaaeldin I., Maurer, Barbara, Wagner, Christina, Schönefeldt, Susann, Spirk, Katrin, Pichler, Alexander, Pemovska, Tea, Schweicker, Carmen, Pölöske, Daniel, Hubanic, Emina, Jungherz, Dennis, Müller, Tony Andreas, Aung, Myint Myat Khine, Orlova, Anna, Pham, Ha Thi Thanh, Zimmel, Kerstin, Krausgruber, Thomas, Bock, Christoph, Müller, Mathias, Dahlhoff, Maik, Boersma, Auke, Rülicke, Thomas, Fleck, Roman, de Araujo, Elvin Dominic, Gunning, Patrick Thomas, Aittokallio, Tero, Mustjoki, Satu, Sanda, Takaomi, Hartmann, Sylvia, Grebien, Florian, Hoermann, Gregor, Haferlach, Torsten, Staber, Philipp Bernhard, Neubauer, Heidi Anne, Look, Alfred Thomas, Herling, Marco, Moriggl, Richard
Published in The Journal of clinical investigation (15.04.2024)
Published in The Journal of clinical investigation (15.04.2024)
Get full text
Journal Article
Loading…
Dual specific STAT3/5 degraders effectively block acute myeloid leukemia and natural killer/T cell lymphoma
Pölöske, Daniel, Sorger, Helena, Schönbichler, Anna, Araujo, Elvin D., Neubauer, Heidi A., Orlova, Anna, Timonen, Sanna H., Abdallah, Diaaeldin I., Ianevski, Aleksandr, Kuusanmäki, Heikki, Surbek, Marta, Heyes, Elisabeth, Eder, Thomas, Wagner, Christina, Suske, Tobias, Metzelder, Martin L., Bergmann, Michael, Dahlhoff, Maik, Grebien, Florian, Fleck, Roman, Pirker, Christine, Berger, Walter, Hadzijusufovic, Emir, Sperr, Wolfgang R., Kenner, Lukas, Valent, Peter, Aittokallio, Tero, Herling, Marco, Mustjoki, Satu, Gunning, Patrick T., Moriggl, Richard
Published in HemaSphere (01.12.2024)
Published in HemaSphere (01.12.2024)
Get full text
Journal Article
Loading…
Small molecule STAT3/5 inhibitors exhibit therapeutic potential in acute myeloid leukemia and extra-nodal natural killer/T cell lymphoma
Pölöske, Daniel, Sorger, Helena, Schönbichler, Anna, de Araujo, Elvin D., Neubauer, Heidi A., Orlova, Anna, Timonen, Sanna H., Abdallah, Diaaeldin I., Ianevski, Aleksandr, Kuusanmäki, Heikki, Surbek, Marta, Wagner, Christina, Suske, Tobias, Metzelder, Martin L., Bergmann, Michael, Dahlhoff, Maik, Grebien, Florian, Fleck, Roman, Pirker, Christine, Berger, Walter, Hadzijusufovic, Emir, Sperr, Wolfgang R., Kenner, Lukas, Valent, Peter, Aittokallio, Tero, Herling, Marco, Mustjoki, Satu, Gunning, Patrick T., Moriggl, Richard
Published in bioRxiv (16.10.2023)
Published in bioRxiv (16.10.2023)
Get full text
Paper