Design and synthesis of some thiazolyl and thiadiazolyl derivatives of antipyrine as potential non-acidic anti-inflammatory, analgesic and antimicrobial agents
Rostom, Sherif A.F., El-Ashmawy, Ibrahim M., Abd El Razik, Heba A., Badr, Mona H., Ashour, Hayam M.A.
Published in Bioorganic & medicinal chemistry (15.01.2009)
Published in Bioorganic & medicinal chemistry (15.01.2009)
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Azole antimicrobial pharmacophore-based tetrazoles: Synthesis and biological evaluation as potential antimicrobial and anticonvulsant agents
Rostom, Sherif A.F., Ashour, Hayam M.A., Razik, Heba A. Abd El, Fattah, Abd El Fattah H. Abd El, El-Din, Nagwa N.
Published in Bioorganic & medicinal chemistry (15.03.2009)
Published in Bioorganic & medicinal chemistry (15.03.2009)
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New heterocyclic hybrids of pyrazole and its bioisosteres: Design, synthesis and biological evaluation as dual acting antimalarial-antileishmanial agents
Bekhit, Adnan A., Hassan, Ahmed M.M., Abd El Razik, Heba A., El-Miligy, Mostafa M.M., El-Agroudy, Eman J., Bekhit, Alaa El-Din A.
Published in European journal of medicinal chemistry (13.04.2015)
Published in European journal of medicinal chemistry (13.04.2015)
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Pyrazoles containing thiophene, thienopyrimidine and thienotriazolopyrimidine as COX-2 selective inhibitors: Design, synthesis, in vivo anti-inflammatory activity, docking and in silico chemo-informatic studies
El-Shoukrofy, Mai S., Abd El Razik, Heba A., AboulWafa, Omaima M., Bayad, Aida E., El-Ashmawy, Ibrahim M.
Published in Bioorganic chemistry (01.04.2019)
Published in Bioorganic chemistry (01.04.2019)
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New pyrimidines and triazolopyrimidines as antiproliferative and antioxidants with cyclooxygenase-1/2 inhibitory potential
Omar, Ashraf M, Abd El Razik, Heba A, Hazzaa, Aly A, El-Attar, Maryam Az, El Demellawy, Maha A, Abdel Wahab, Abeer E, El Hawash, Soad Am
Published in Future medicinal chemistry (01.07.2019)
Published in Future medicinal chemistry (01.07.2019)
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Synthesis and biological evaluation of purine-pyrazole hybrids incorporating thiazole, thiazolidinone or rhodanine moiety as 15-LOX inhibitors endowed with anticancer and antioxidant potential
Afifi, Ola S., Shaaban, Omaima G., Abd El Razik, Heba A., Shams El-Dine, Shams El-Dine A., Ashour, Fawzia A., El-Tombary, Alaa A., Abu-Serie, Marwa M.
Published in Bioorganic chemistry (01.06.2019)
Published in Bioorganic chemistry (01.06.2019)
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Journal Article
Benzodioxole–Pyrazole Hybrids as Anti‐Inflammatory and Analgesic Agents with COX‐1,2/5‐LOX Inhibition and Antioxidant Potential
Abd El Razik, Heba A., Badr, Mona H., Atta, Attia H., Mouneir, Samar M., Abu‐Serie, Marwa M.
Published in Archiv der Pharmazie (Weinheim) (01.05.2017)
Published in Archiv der Pharmazie (Weinheim) (01.05.2017)
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Identification of new 5-(2,6-dichlorophenyl)-3-oxo-2,3-dihydro-5H-thiazolo[3,2-a]pyrimidine-7-carboxylic acids as p38α MAPK inhibitors: Design, synthesis, antitumor evaluation, molecular docking and in silico studies
El-Wakil, Marwa H., El-Dershaby, Hadeel A., Ghazallah, Rasha A., El-Yazbi, Amira F., Abd El-Razik, Heba A., Soliman, Farid S.G.
Published in Bioorganic chemistry (01.04.2024)
Published in Bioorganic chemistry (01.04.2024)
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New thieno[3,2-d]pyrimidine-based derivatives: Design, synthesis and biological evaluation as antiproliferative agents, EGFR and ARO inhibitors inducing apoptosis in breast cancer cells
Farghaly, Ahmed M., AboulWafa, Omaima M., Baghdadi, Hoda H., Abd El Razik, Heba A., Sedra, Samir M.Y., Shamaa, Marium M.
Published in Bioorganic chemistry (01.10.2021)
Published in Bioorganic chemistry (01.10.2021)
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Structure-based development of novel triazoles and related thiazolotriazoles as anticancer agents and Cdc25A/B phosphatase inhibitors. Synthesis, in vitro biological evaluation, molecular docking and in silico ADME-T studies
Rostom, Sherif A.F., Badr, Mona H., Abd El Razik, Heba A., Ashour, Hayam M.A.
Published in European journal of medicinal chemistry (20.10.2017)
Published in European journal of medicinal chemistry (20.10.2017)
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Journal Article
Synthesis of new pyrazolo[3,4‐d]pyrimidine derivatives and evaluation of their anti‐inflammatory and anticancer activities
Abd El Razik, Heba A., Mroueh, Mohamad, Faour, Wissam H., Shebaby, Wassim N., Daher, Costantine F., Ashour, Hayam M. A., Ragab, Hanan M.
Published in Chemical biology & drug design (01.07.2017)
Published in Chemical biology & drug design (01.07.2017)
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Synthesis and biological evaluation of new oxadiazoline-substituted naphthalenyl acetates as anticancer agents
Chaaban, Ibrahim, El Khawass, El Sayeda M., Abd El Razik, Heba A., El Salamouni, Nehad S., Redondo-Horcajo, Mariano, Barasoain, Isabel, Díaz, J. Fernando, Yli-Kauhaluoma, Jari, Moreira, Vânia M.
Published in European journal of medicinal chemistry (24.11.2014)
Published in European journal of medicinal chemistry (24.11.2014)
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Journal Article
Purines and triazolo[4,3-e]purines containing pyrazole moiety as potential anticancer and antioxidant agents
Shaaban, Omaima G, Abd El Razik, Heba A, A Shams El-Dine, Shams El-Dine, Ashour, Fawzia A, El-Tombary, Alaa A, Afifi, Ola S, Abu-Serie, Marwa M
Published in Future medicinal chemistry (01.06.2018)
Published in Future medicinal chemistry (01.06.2018)
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Journal Article
Synthesis of Some Pyrazolines and Pyrimidines Derived from Polymethoxy Chalcones as Anticancer and Antimicrobial Agents
Rostom, Sherif A.F., Badr, Mona H., Abd El Razik, Heba A., Ashour, Hayam M.A., Abdel Wahab, Abeer E.
Published in Archiv der Pharmazie (Weinheim) (01.09.2011)
Published in Archiv der Pharmazie (Weinheim) (01.09.2011)
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Journal Article
Synthesis and Anti-Proliferative Activity of Sulfanyltriazolylnaphthalenols and Sulfanyltriazolylnaphthalene-1,4-diones
Chaaban, Ibrahim, El Khawass, El Sayeda M., Abd El Razik, Heba A., El Salamouni, Nehad S., Redondo-Horcajo, Mariano, Barasoain, Isabel, Díaz, José Fernando, Yli-Kauhaluoma, Jari, Moreira, Vânia M.
Published in Archiv der Pharmazie (Weinheim) (01.09.2016)
Published in Archiv der Pharmazie (Weinheim) (01.09.2016)
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