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Published in Bioorganic & medicinal chemistry letters (15.03.2014)
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An inhibitor of Bcl-2 family proteins induces regression of solid tumours
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Published in ACS medicinal chemistry letters (08.10.2020)
Published in ACS medicinal chemistry letters (08.10.2020)
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Year of Publication 10.09.2020
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Year of Publication 27.08.2020
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Year of Publication 13.02.2020
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8-CARBAMOYL-2-(2,3-DISUBSTITUTED PYRID-6-YL)-1,2,3,4-TETRAHYDROISOQUINOLINE DERIVATIVES AS APOPTOSIS-INDUCING AGENTS FOR TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES
GEORGE DOHERTY, TAO ZHI-FU, SONG XIAOHONG, ANDREW SOUERS, AARON R KUNZER, LE WANG, XILU WANG, ANDREW JUDD, TODD M HANSEN, SULLIVAN GERARD M, ROBIN FREY, WENDT MICHAEL D, MILAN BRUNCKO
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Year of Publication 02.11.2017
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APOPTOSIS INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES
GEORGE DOHERTY, GERARD SULLIVAN, TAO ZHI-FU, STEVEN ELMORE, SONG XIAOHONG, LAURA HEXAMER, AARON R KUNZER, LE WANG, MICHAEL WENDT, LISA HASVOLD, XILU WANG, TODD M HANSEN, ROBERT MANTEI, ANDREW J SOUERS, DING HONG, GARY T WANG, MILAN BRUNCKO
Year of Publication 06.09.2018
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Year of Publication 06.09.2018
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Discovery of A-1331852, a First-in-Class, Potent, and Orally-Bioavailable BCL-X-L Inhibitor
Wang, Le, Doherty, George A., Judd, Andrew S., Tao, Zhi-Fu, Hansen, T. Matthew, Frey, Robin R., Song, Xiaohong, Bruncko, Milan, Kunzer, Aaron R., Wang, Xilu, Wendt, Michael D., Flygare, John A., Catron, Nathaniel D., Judge, Russell A., Park, Chang H., Shekhar, Shashank, Phillips, Darren C., Nimmer, Paul, Smith, Morey L., Tahir, Stephen K., Xiao, Yu, Xue, John, Zhang, Haichao, Le, Phuong N., Mitten, Michael J., Boghaert, Erwin R., Gao, Wenqing, Kovar, Peter, Choo, Edna F., Diaz, Dolores, Fairbrother, Wayne J., Elmore, Steven W., Sampath, Deepak, Leverson, Joel D., Souers, Andrew James
Published in ACS medicinal chemistry letters (08.10.2020)
Published in ACS medicinal chemistry letters (08.10.2020)
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Year of Publication 30.03.2017
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APOPTOSIS INDUCING AGENTS FOR TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES
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Year of Publication 09.03.2017
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Year of Publication 09.03.2017
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SULFONE AMIDE DERIVATIVE AS BCL-2-SELECTIVE APOPTOSIS INDUCING AGENT FOR TREATMENT OF CANCER AND IMMUNE DISEASE
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Year of Publication 16.07.2015
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Year of Publication 16.07.2015
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APOPTOSIS-INDUCING AGENTS FOR TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES
GEORGE DOHERTY, GERARD SULLIVAN, TAO ZHI-FU, STEVEN ELMORE, SONG XIAOHONG, LAURA HEXAMER, AARON R KUNZER, LE WANG, MICHAEL WENDT, LISA HASVOLD, XILU WANG, TODD M HANSEN, ROBERT MANTEI, ANDREW J SOUERS, DING HONG, GARY T WANG, MILAN BRUNCKO
Year of Publication 18.06.2015
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Year of Publication 18.06.2015
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APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES
WILLIAM J MCCLELLAN, GERARD M SULLIVAN, ROBERT A MANTEI, STEVEN W ELMORE, TAO ZHI-FU, PETER EDWARD CZABOTAR, DAI YUJIA, SONG XIAOHONG, LAURA HEXAMER, GUILLAUME LAURENT LESSENE, PARK CHEOL-MIN, PETER MALCOLM COLMAN, AARON R KUNZER, LE WANG, LISA HASVOLD, XILU WANG, ANDREW M PETROS, CHANG H PARK, ANDREW J SOUERS, WENDT MICHAEL D, DING HONG, GARY T WANG, GEORGE A DOHERTY, MILAN BRUNCKO
Year of Publication 11.06.2015
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Year of Publication 11.06.2015
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