Donepezil-Based Central Acetylcholinesterase Inhibitors by Means of a “Bio-Oxidizable” Prodrug Strategy: Design, Synthesis, and in Vitro Biological Evaluation
Peauger, Ludovic, Azzouz, Rabah, Gembus, Vincent, Ţînţaş, Mihaela-Liliana, Sopková-de Oliveira Santos, Jana, Bohn, Pierre, Papamicaël, Cyril, Levacher, Vincent
Published in Journal of medicinal chemistry (13.07.2017)
Published in Journal of medicinal chemistry (13.07.2017)
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Journal Article
Design, Synthesis, and In Vitro Biological Activities of a Bio-Oxidizable Prodrug to Deliver Both ChEs and DYRK1A Inhibitors for AD Therapy
Barré, Anaïs, Azzouz, Rabah, Gembus, Vincent, Papamicaël, Cyril, Levacher, Vincent
Published in Molecules (Basel, Switzerland) (01.04.2019)
Published in Molecules (Basel, Switzerland) (01.04.2019)
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Journal Article
Efficient Conversion of Epoxides into Carbonates with CO2 and a Single Organocatalyst: Laboratory and Kilogram-Scale Experiments
Azzouz, Rabah, Moreno, Viviana Contreras, Herasme-Grullon, Clara, Levacher, Vincent, Estel, Lionel, Ledoux, Alain, Derrouiche, Salim, Marsais, Francis, Bischoff, Laurent
Published in Synlett (24.01.2020)
Published in Synlett (24.01.2020)
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Novel donepezil-like N-benzylpyridinium salt derivatives as AChE inhibitors and their corresponding dihydropyridine “bio-oxidizable” prodrugs: Synthesis, biological evaluation and structure-activity relationship
Azzouz, Rabah, Peauger, Ludovic, Gembus, Vincent, Ţînţaş, Mihaela-Liliana, Sopková-de Oliveira Santos, Jana, Papamicaël, Cyril, Levacher, Vincent
Published in European journal of medicinal chemistry (10.02.2018)
Published in European journal of medicinal chemistry (10.02.2018)
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Journal Article
Access to Highly Enantioenriched Donepezil-like 1,4-Dihydropyridines as Promising Anti-Alzheimer Prodrug Candidates via Enantioselective Tsuji Allylation and Organocatalytic Aza-Ene-Type Domino Reactions
Ţînţaş, Mihaela-Liliana, Azzouz, Rabah, Peauger, Ludovic, Gembus, Vincent, Petit, Emilie, Bailly, Laëtitia, Papamicaël, Cyril, Levacher, Vincent
Published in Journal of organic chemistry (19.07.2018)
Published in Journal of organic chemistry (19.07.2018)
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Journal Article
Access to Highly Enantioenriched Donepezil-like 1,4-Dihydropyridines as Promising Anti-Alzheimer Prodrug Candidates via Enantioselective Tsuji Allylation and Organocatalytic Aza-Ene-Type Domino Reactions
Ţînţaş, Mihaela-Liliana, Azzouz, Rabah, Peauger, Ludovic, Gembus, Vincent, Petit, Emilie, Bailly, Laetitia, Papamicaël, Cyril, Levacher, Vincent
Published in Journal of organic chemistry (07.09.2018)
Published in Journal of organic chemistry (07.09.2018)
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Journal Article
Synthesis of new F-18-radiolabeled silicon-based nitroimidazole compounds
Joyard, Yoann, Azzouz, Rabah, Bischoff, Laurent, Papamicael, Cyril, Labar, Daniel, Bol, Anne, Bol, Vanessa, Vera, Pierre, Gregoire, Vincent, Levacher, Vincent, Bohn, Pierre
Published in Bioorganic & medicinal chemistry (01.07.2013)
Published in Bioorganic & medicinal chemistry (01.07.2013)
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Journal Article
Design of silicon-based misonidazole analogues and (18)F-radiolabelling
Bohn, Pierre, Deyine, Abdallah, Azzouz, Rabah, Bailly, Laetitia, Fiol-Petit, Catherine, Bischoff, Laurent, Fruit, Corinne, Marsais, Francis, Vera, Pierre
Published in Nuclear medicine and biology (01.11.2009)
Published in Nuclear medicine and biology (01.11.2009)
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Journal Article
Synthesis of new 18F-radiolabeled silicon-based nitroimidazole compounds
Joyard, Yoann, Azzouz, Rabah, Bischoff, Laurent, Papamicaël, Cyril, Labar, Daniel, Bol, Anne, Bol, Vanessa, Vera, Pierre, Grégoire, Vincent, Levacher, Vincent, Bohn, Pierre
Published in Bioorganic & medicinal chemistry (01.07.2013)
Published in Bioorganic & medicinal chemistry (01.07.2013)
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Journal Article
O-tetrahydropyran-2-yloxy (O-THP) as an ortho-directing group in the lithiation of pyridines
Azzouz, Rabah, Bischoff, Laurent, Fruit, Corinne, Marsais, Francis
Published in Synlett (01.08.2006)
Published in Synlett (01.08.2006)
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Aminomethylation of lithiated nicotinamide: access to new pyridolactams
Prieur, Emilie, Azzouz, Rabah, Deguest, Geoffrey, Fruit, Corinne, Bischoff, Laurent, Marsais, Francis
Published in Tetrahedron letters (01.01.2008)
Published in Tetrahedron letters (01.01.2008)
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Journal Article
Design of silicon-based misonidazole analogues and 18F-radiolabelling
Bohn, Pierre, Deyine, Abdallah, Azzouz, Rabah, Bailly, Laetitia, Fiol-Petit, Catherine, Bischoff, Laurent, Fruit, Corinne, Marsais, Francis, Vera, Pierre
Published in Nuclear medicine and biology (01.11.2009)
Published in Nuclear medicine and biology (01.11.2009)
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Journal Article
Design of silicon-based misonidazole analogues and18 F-radiolabelling
Bohn, Pierre, Deyine, Abdallah, Azzouz, Rabah, Bailly, Laetitia, Fiol-Petit, Catherine, Bischoff, Laurent, Fruit, Corinne, Marsais, Francis, Vera, Pierre
Published in Nuclear medicine and biology (2009)
Published in Nuclear medicine and biology (2009)
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Journal Article
VALORISATION DU CO2
LEDOUX, ALAIN, ESTEL, LIONEL, CONTRERAS MORENO, VIVIANA, DERROUICHE, SALIM, BISCHOFF, LAURENT, AZZOUZ, RABAH, LEVACHER, VINCENT, MARSAIS, FRANCIS
Year of Publication 13.07.2018
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Year of Publication 13.07.2018
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