TMC278, a Next-Generation Nonnucleoside Reverse Transcriptase Inhibitor (NNRTI), Active against Wild-Type and NNRTI-Resistant HIV-1
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Published in Antimicrobial Agents and Chemotherapy (01.02.2010)
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Resistance profile of etravirine: combined analysis of baseline genotypic and phenotypic data from the randomized, controlled Phase III clinical studies
VINGERHOETS, Johan, TAMBUYZER, Lotke, AZIJN, Hilde, HOOGSTOEL, Annemie, NIJS, Steven, PEETERS, Monika, DE BETHUNE, Marie-Pierre, DE SMEDT, Goedele, WOODFALL, Brian, PICCHIO, Gastón
Published in AIDS (London) (20.02.2010)
Published in AIDS (London) (20.02.2010)
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TMC114, a Novel Human Immunodeficiency Virus Type 1 Protease Inhibitor Active against Protease Inhibitor-Resistant Viruses, Including a Broad Range of Clinical Isolates
DE MEYER, Sandra, AZIJN, Hilde, SURLERAUX, Dominique, JOCHMANS, Dirk, TAHRI, Abdellah, PAUWELS, Rudi, WIGERINCK, Piet, DE BETHUNE, Marie-Pierre
Published in Antimicrobial Agents and Chemotherapy (01.06.2005)
Published in Antimicrobial Agents and Chemotherapy (01.06.2005)
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TMC125 Displays a High Genetic Barrier to the Development of Resistance: Evidence from In Vitro Selection Experiments
VINGERHOETS, Johan, AZIJN, Hilde, FRANSEN, Els, DE BAERE, Inky, SMEULDERS, Liesbet, JOCHMANS, Dirk, ANDRIES, Koen, PAUWELS, Rudi, DE BETHUNE, Marie-Pierre
Published in Journal of Virology (01.10.2005)
Published in Journal of Virology (01.10.2005)
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TMC125, a Novel Next-Generation Nonnucleoside Reverse Transcriptase Inhibitor Active against Nonnucleoside Reverse Transcriptase Inhibitor-Resistant Human Immunodeficiency Virus Type 1
ANDRIES, Koen, AZIJN, Hilde, DE BETHUNE, Marie-Pierre, THIELEMANS, Theo, LUDOVICI, Donald, KUKLA, Michael, HEERES, Jan, JANSSEN, Paul, DE CORTE, Bart, VINGERHOETS, Johan, PAUWELS, Rudi
Published in Antimicrobial Agents and Chemotherapy (01.12.2004)
Published in Antimicrobial Agents and Chemotherapy (01.12.2004)
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Discovery and Selection of TMC114, a Next Generation HIV-1 Protease Inhibitor
Surleraux, Dominique L. N. G, Tahri, Abdellah, Verschueren, Wim G, Pille, Geert M. E, de Kock, Herman A, Jonckers, Tim H. M, Peeters, Anik, De Meyer, Sandra, Azijn, Hilde, Pauwels, Rudi, de Bethune, Marie-Pierre, King, Nancy M, Prabu-Jeyabalan, Moses, Schiffer, Celia A, Wigerinck, Piet B. T. P
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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Connection Domain Mutations in HIV-1 Reverse Transcriptase Do Not Impact Etravirine Susceptibility and Virologic Responses to Etravirine-Containing Regimens
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Published in Antimicrobial Agents and Chemotherapy (01.06.2011)
Published in Antimicrobial Agents and Chemotherapy (01.06.2011)
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A Rapid Method for Simultaneous Detection of Phenotypic Resistance to Inhibitors of Protease and Reverse Transcriptase in Recombinant Human Immunodeficiency Virus Type 1 Isolates from Patients Treated with Antiretroviral Drugs
HERTOGS, K, DE BETHUNE, M.-P, PEETERS, F, STASZEWSKI, S, CONANT, M, BLOOR, S, KEMP, S, LARDER, B, PAUWELS, R, MILLER, V, IVENS, T, SCHEL, P, VAN CAUWENBERGE, A, VAN DEN EYNDE, C, VAN GERWEN, V, AZIJN, H, VAN HOUTTE, M
Published in Antimicrobial Agents and Chemotherapy (01.02.1998)
Published in Antimicrobial Agents and Chemotherapy (01.02.1998)
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Compilation and prevalence of mutations associated with resistance to non-nucleoside reverse transcriptase inhibitors
TAMBUYZER, Lotke, AZIJN, Hilde, RIMSKY, Laurence T, VINGERHOETS, Johan, LECOCQ, Pierre, KRAUS, Guenter, PICCHIO, Gaston, DE BETHUNE, Marie-Pierre
Published in Antiviral therapy (2009)
Published in Antiviral therapy (2009)
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Characterization of genotypic and phenotypic changes in HIV-1-infected patients with virologic failure on an etravirine-containing regimen in the DUET-1 and DUET-2 clinical studies
Tambuyzer, Lotke, Vingerhoets, Johan, Azijn, Hilde, Daems, Bjorn, Nijs, Steven, de Béthune, Marie-Pierre, Picchio, Gastón
Published in AIDS research and human retroviruses (01.11.2010)
Published in AIDS research and human retroviruses (01.11.2010)
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Etravirine limits the emergence of darunavir and other protease inhibitor resistance-associated mutations in the DUET trials
PEETERS, Monika, VINGERHOETS, Johan, TAMBUYZER, Lotke, AZIJN, Hilde, HILL, Andrew, DE MEYER, Sandra, PICCHIO, Gaston
Published in AIDS (London) (27.03.2010)
Published in AIDS (London) (27.03.2010)
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Evolution of anti-HIV drug candidates. Part 3: diarylpyrimidine (DAPY) analogues
Ludovici, Donald W., De Corte, Bart L., Kukla, Michael J., Ye, Hong, Ho, Chih Y., Lichtenstein, Mark A., Kavash, Robert W., Andries, Koen, de Béthune, Marie-Pierre, Azijn, Hilde, Pauwels, Rudi, Lewi, Paul J., Heeres, Jan, Koymans, Lucien M.H., de Jonge, Marc R., Van Aken, Koen J.A., Daeyaert, Frederik F.D., Das, Kalyan, Arnold, Edward, Janssen, Paul A.J.
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
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Design of HIV-1 Protease Inhibitors Active on Multidrug-Resistant Virus
Surleraux, Dominique L. N. G, de Kock, Herman A, Verschueren, Wim G, Pille, Geert M. E, Maes, Louis J. R, Peeters, Anik, Vendeville, Sandrine, De Meyer, Sandra, Azijn, Hilde, Pauwels, Rudi, de Bethune, Marie-Pierre, King, Nancy M, Prabu-Jeyabalan, Moses, Schiffer, Celia A, Wigerinck, Piet B. T. P
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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Short communication: activity of etravirine on different HIV type 1 subtypes: in vitro susceptibility in treatment-naive patients and week 48 pooled DUET study data
Vingerhoets, Johan, Azijn, Hilde, Tambuyzer, Lotke, Dierynck, Inge, De Meyer, Sandra, Rimsky, Laurence, Nijs, Steven, De Smedt, Goedele, de Béthune, Marie-Pierre, Picchio, Gaston
Published in AIDS research and human retroviruses (01.06.2010)
Published in AIDS research and human retroviruses (01.06.2010)
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Design, Synthesis, and SAR of a Novel Pyrazinone Series with Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitory Activity
Heeres, Jan, de Jonge, Marc R, Koymans, Lucien M. H, Daeyaert, Frits F. D, Vinkers, Maarten, Van Aken, Koen J. A, Arnold, Eddy, Das, Kalyan, Kilonda, Amuri, Hoornaert, Georges J, Compernolle, Frans, Cegla, Marek, Azzam, Rasha A, Andries, Koen, de Béthune, Marie-Pierre, Azijn, Hilde, Pauwels, Rudi, Lewi, Paul J, Janssen, Paul A. J
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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Evolution of anti-HIV drug candidates. Part 2 : Diaryltriazine (DATA) analogues
LUDOVICI, Donald W, KAVASH, Robert W, MOEREELS, Henry E. L, HEERES, Jan, KOYMANS, Lucien M. H, DE JONGE, Marc R, VAN AKEN, Koen J. A, DAEYAERT, Frederik F. D, LEWI, Paul J, DAS, Kalyan, ARNOLD, Edward, JANSSEN, Paul A. J, KUKLA, Michael J, HO, Chih Y, HONG YE, DE CORTE, Bart L, ANDRIES, Koen, DE BETHUNE, Marie-Pierre, AZIJN, Hilde, PAUWELS, Rudi
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
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Evolution of anti-HIV drug candidates. Part 1: From α-Anilinophenylacetamide (α-APA) to imidoyl thiourea (ITU)
Ludovici, Donald W., Kukla, Michael J., Grous, Philip G., Krishnan, Suma, Andries, Koen, de Béthune, Marie-Pierre, Azijn, Hilde, Pauwels, Rudi, De Clercq, Erik, Arnold, Edward, Janssen, Paul A.J.
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
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Evolution of Anti-HIV Drug CandidatesPart 2: Diaryltriazine (DATA) Analogues
Ludovici, Donald W., Kavash, Robert W., Kukla, Michael J., Ho, Chih Y., Ye, Hong, De Corte, Bart L., Andries, Koen, de Béthune, Marie-Pierre, Azijn, Hilde, Pauwels, Rudi, Moereels, Henry E.L., Heeres, Jan, Koymans, Lucien M.H., de Jonge, Marc R., Van Aken, Koen J.A., Daeyaert, Frederik F.D., J. Lewi, Paul, Das, Kalyan, Arnold, Edward, Janssen, Paul A.J.
Published in Bioorganic & medicinal chemistry letters (01.09.2001)
Published in Bioorganic & medicinal chemistry letters (01.09.2001)
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Automated techniques in biotechnology
Pauwels, Rudi, Azijn, Hilde, de Béthune, Marie-Pierre, Claeys, Carine, Hertogs, Kurt
Published in Current opinion in biotechnology (1995)
Published in Current opinion in biotechnology (1995)
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