Design and evaluation of pyrazolopyrimidines as KCNQ channel modulators
Osuma, Augustine T., Xu, Xiangdong, Wang, Zhi, Van Camp, Jennifer A., Freiberg, Gail M.
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Published in Bioorganic & medicinal chemistry letters (01.10.2019)
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The HPK1 Inhibitor A‑745 Verifies the Potential of Modulating T Cell Kinase Signaling for Immunotherapy
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Published in ACS chemical biology (18.03.2022)
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A scalable approach to diaminopyrazoles using flow chemistry
Wilson, Noel S., Osuma, Augustine T., Camp, Jennifer A.Van, Xu, Xiangdong
Published in Tetrahedron letters (22.08.2012)
Published in Tetrahedron letters (22.08.2012)
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Porphyrins with Exocyclic Rings. 13. Synthesis and Spectroscopic Characterization of Highly Modified Porphyrin Chromophores with Fused Acenaphthylene and Benzothiadiazole Rings
Lash, Timothy D, Chandrasekar, Pushpa, Osuma, Augustine T, Chaney, Sun T, Spence, John D
Published in Journal of organic chemistry (13.11.1998)
Published in Journal of organic chemistry (13.11.1998)
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Journal Article
ChemInform Abstract: A Scalable Approach to Diaminopyrazoles Using Flow Chemistry
Wilson, Noel S., Osuma, Augustine T., Van Camp, Jennifer A., Xu, Xiangdong
Published in ChemInform (27.11.2012)
Published in ChemInform (27.11.2012)
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The efficient synthesis of (3R,4R,5R)-3-amino-4,5-dimethyl-octanoic acid, a chiral β-amino acid with potent affinity for the α2δ protein
Zhang, Ji, Blazecka, Peter G., Pflum, Derek A., Bozelak, Joseph, Vrieze, Derek, Colbry, Norman L., Hoge, Garrett, Boyles, David C., Samas, Brian, Curran, Timothy T., Osuma, Augustine T., Johnson, Paul, Kesten, Suzanne, Schwarz, Jacob B., Goodman, Annise, Plummer, Mark, Akin, Anne, Huang, Yun, Lovdahl, Michael, Thorpe, Andrew J.
Published in Tetrahedron letters (18.03.2009)
Published in Tetrahedron letters (18.03.2009)
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Journal Article
The efficient synthesis of (3R,4R,5R)-3-amino-4,5-dimethyl-octanoic acid, a chiral beta-amino acid with potent affinity for the alpha(2)delta protein
Zhang, Ji, Blazecka, Peter G., Pflum, Derek A., Bozelak, Joseph, Vrieze, Derek, Colbry, Norman L., Hoge, Garrett, Boyles, David C., Samas, Brian, Curran, Timothy T., Osuma, Augustine T., Johnson, Paul, Kesten, Suzanne, Schwarz, Jacob B., Goodman, Annise, Plummer, Mark, Akin, Anne, Huang, Yun, Lovdahl, Michael, Thorpe, Andrew J.
Published in Tetrahedron letters (18.03.2009)
Published in Tetrahedron letters (18.03.2009)
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Journal Article
The efficient synthesis of (3 R,4 R,5 R)-3-amino-4,5-dimethyl-octanoic acid, a chiral β-amino acid with potent affinity for the α 2δ protein
Zhang, Ji, Blazecka, Peter G., Pflum, Derek A., Bozelak, Joseph, Vrieze, Derek, Colbry, Norman L., Hoge, Garrett, Boyles, David C., Samas, Brian, Curran, Timothy T., Osuma, Augustine T., Johnson, Paul, Kesten, Suzanne, Schwarz, Jacob B., Goodman, Annise, Plummer, Mark, Akin, Anne, Huang, Yun, Lovdahl, Michael, Thorpe, Andrew J.
Published in Tetrahedron letters (2009)
Published in Tetrahedron letters (2009)
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Journal Article
Porphyrins with Exocyclic Rings. 13. 1 Synthesis and Spectroscopic Characterization of Highly Modified Porphyrin Chromophores with Fused Acenaphthylene and Benzothiadiazole Rings
Lash, Timothy D., Chandrasekar, Pushpa, Osuma, Augustine T., Chaney, Sun T., Spence, John D.
Published in Journal of organic chemistry (01.11.1998)
Published in Journal of organic chemistry (01.11.1998)
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INDAZOLONES AS MODULATORS OF TNF SIGNALING
Dietrich, Justin D, Kinsman, David, Friedman, Michael, Ihle, David, Vasudevan, Anil, Burchat, Andrew, Mullen, Kelly, Osuma, Augustine T, Wilson, Noel S, Breinlinger, Eric C
Year of Publication 02.08.2018
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Year of Publication 02.08.2018
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TRICYCLIC MODULATORS OF TNF SIGNALING
Dietrich, Justin D, Frank, Kristine E, Cox, Phil B, Vasudevan, Anil, Osuma, Augustine T, Li, Huan-Qui, Longenecker, Kenton L, Wilson, Noel S, Breinlinger, Eric C, Friedman, Michael M, Rowley, Ann Marie
Year of Publication 28.06.2018
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Year of Publication 28.06.2018
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Tricyclic modulators of TNF signaling
Dietrich, Justin D, Frank, Kristine E, Gomtsyan, Arthur, Dombrowski, Amanda W, Schmidt, Robert, Breinlinger, Eric C, Friedman, Michael M, Cox, Phil B, Vasudevan, Anil, Osuma, Augustine T, Daanen, Jerome, Li, Huan-Qui, Longenecker, Kenton L, Wilson, Noel S, Rowley, Ann Marie, Djuric, Stevan
Year of Publication 23.04.2019
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Year of Publication 23.04.2019
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NAMPT INHIBITORS
SORENSEN, BRYAN, SWEIS, RAMZI F, CLARK, RICHARD F, LONGENECKER, KENTON, OSUMA, AUGUSTINE T, HEYMAN, HOWARD R, JUDD, ANDY, PLUISHCHEV, MARINA A, FREY, ROBIN, HANSEN, TODD M, CURTIN, MICHAEL L, DOHERTY, GEORGE, MICHAELIDES, MICHAEL R
Year of Publication 30.08.2017
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Year of Publication 30.08.2017
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Sorensen Bryan, Judd Andrew, Heyman Howard R, Pliushchev Marina, Osuma Augustine T, Hansen Todd, Doherty George, Curtin Michael L, Michaelides Michael, Clark Richard F, Sweis Ramzi, Frey Robin, Longenecker Kenton
Year of Publication 18.05.2017
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Year of Publication 18.05.2017
Patent
NAMPT INHIBITORS
HEYMAN HOWARD R, JUDD ANDREW, HANSEN TODD, MICHAELIDES MICHAEL, DOHERTY GEORGE, SORENSEN BRYAN, LONGENECKER KENTON, FREY ROBIN, CURTIN MICHAEL L, SWEIS RAMZI, OSUMA AUGUSTINE T, CLARK RICHARD F, PLIUSHCHEV MARINA
Year of Publication 30.06.2016
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Year of Publication 30.06.2016
Patent
NAMPT INHIBITORS
HEYMAN HOWARD R, JUDD ANDREW, HANSEN TODD, MICHAELIDES MICHAEL, DOHERTY GEORGE, SORENSEN BRYAN, LONGENECKER KENTON, FREY ROBIN, CURTIN MICHAEL L, SWEIS RAMZI, OSUMA AUGUSTINE T, CLARK RICHARD F, PLIUSHCHEV MARINA
Year of Publication 30.06.2016
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Year of Publication 30.06.2016
Patent
NAMPT INHIBITORS NAMPT
SORENSEN, BRYAN, CLARK, RICHARD F, SWEIS, RAMZI F, LONGENECKER, KENTON, OSUMA, AUGUSTINE T, HEYMAN, HOWARD R, PLIUSHCHEV, MARINA A, JUDD, ANDY, FREY, ROBIN, HANSEN, TODD M, CURTIN, MICHAEL L, DOHERTY, GEORGE, MICHAELIDES, MICHAEL R
Year of Publication 04.03.2016
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Year of Publication 04.03.2016
Patent
NAMPT INHIBITORS NAMPT
SORENSEN, BRYAN, CLARK, RICHARD F, SWEIS, RAMZI F, LONGENECKER, KENTON, OSUMA, AUGUSTINE T, HEYMAN, HOWARD R, PLIUSHCHEV, MARINA A, JUDD, ANDY, FREY, ROBIN, HANSEN, TODD M, CURTIN, MICHAEL L, DOHERTY, GEORGE, MICHAELIDES, MICHAEL R
Year of Publication 26.02.2016
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Year of Publication 26.02.2016
Patent
NAMPT inhibitors
HEYMAN HOWARD R, HANSEN TODD M, MICHAELIDES MICHAEL R, DOHERTY GEORGE, SWEIS RAMZI F, SORENSEN BRYAN, LONGENECKER KENTON, FREY ROBIN, CURTIN MICHAEL L, JUDD ANDY, OSUMA AUGUSTINE T, PLIUSHCHEV MARINA A, CLARK RICHARD F
Year of Publication 24.11.2015
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Year of Publication 24.11.2015
Patent