Small molecule inhibition of cGAS reduces interferon expression in primary macrophages from autoimmune mice
Vincent, Jessica, Adura, Carolina, Gao, Pu, Luz, Antonio, Lama, Lodoe, Asano, Yasutomi, Okamoto, Rei, Imaeda, Toshihiro, Aida, Jumpei, Rothamel, Katherine, Gogakos, Tasos, Steinberg, Joshua, Reasoner, Seth, Aso, Kazuyoshi, Tuschl, Thomas, Patel, Dinshaw J., Glickman, J. Fraser, Ascano, Manuel
Published in Nature communications (29.09.2017)
Published in Nature communications (29.09.2017)
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Rejuvenation of mucosal immunosenescence by adipose tissue-derived mesenchymal stem cells
Tsuruhara, Akitoshi, Aso, Kazuyoshi, Tokuhara, Daisuke, Ohori, Junichiro, Kawabata, Masaki, Kurono, Yuichi, McGhee, Jerry R, Fujihashi, Kohtaro
Published in International immunology (01.01.2017)
Published in International immunology (01.01.2017)
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Design and synthesis of 1-(1-benzothiophen-7-yl)-1H-pyrazole, a novel series of G protein-coupled receptor 52 (GPR52) agonists
Nakahata, Takashi, Tokumaru, Kazuyuki, Ito, Yoshiteru, Ishii, Naoki, Setoh, Masaki, Shimizu, Yuji, Harasawa, Toshiya, Aoyama, Kazunobu, Hamada, Teruki, Kori, Masakuni, Aso, Kazuyoshi
Published in Bioorganic & medicinal chemistry (01.05.2018)
Published in Bioorganic & medicinal chemistry (01.05.2018)
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Journal Article
Adipose-Derived Mesenchymal Stem Cells Restore Impaired Mucosal Immune Responses in Aged Mice
Aso, Kazuyoshi, Tsuruhara, Akitoshi, Takagaki, Kentaro, Oki, Katsuyuki, Ota, Megumi, Nose, Yasuhiro, Tanemura, Hideki, Urushihata, Naoki, Sasanuma, Jinichi, Sano, Masayuki, Hirano, Atsuyuki, Aso, Rio, McGhee, Jerry R, Fujihashi, Kohtaro
Published in PloS one (03.02.2016)
Published in PloS one (03.02.2016)
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Publisher Correction: Small molecule inhibition of cGAS reduces interferon expression in primary macrophages from autoimmune mice
Vincent, Jessica, Adura, Carolina, Gao, Pu, Luz, Antonio, Lama, Lodoe, Asano, Yasutomi, Okamoto, Rei, Imaeda, Toshihiro, Aida, Jumpei, Rothamel, Katherine, Gogakos, Tasos, Steinberg, Joshua, Reasoner, Seth, Aso, Kazuyoshi, Tuschl, Thomas, Patel, Dinshaw J., Glickman, J. Fraser, Ascano, Manuel
Published in Nature communications (23.11.2017)
Published in Nature communications (23.11.2017)
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Chemical structure-guided design of dynapyrazoles, cell-permeable dynein inhibitors with a unique mode of action
Steinman, Jonathan B, Santarossa, Cristina C, Miller, Rand M, Yu, Lola S, Serpinskaya, Anna S, Furukawa, Hideki, Morimoto, Sachie, Tanaka, Yuta, Nishitani, Mitsuyoshi, Asano, Moriteru, Zalyte, Ruta, Ondrus, Alison E, Johnson, Alex G, Ye, Fan, Nachury, Maxence V, Fukase, Yoshiyuki, Aso, Kazuyoshi, Foley, Michael A, Gelfand, Vladimir I, Chen, James K, Carter, Andrew P, Kapoor, Tarun M
Published in eLife (19.05.2017)
Published in eLife (19.05.2017)
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Potential roles of CCR5(+) CCR6(+) dendritic cells induced by nasal ovalbumin plus Flt3 ligand expressing adenovirus for mucosal IgA responses
Fukuyama, Yoshiko, Tokuhara, Daisuke, Sekine, Shinichi, Aso, Kazuyoshi, Kataoka, Kosuke, Davydova, Julia, Yamamoto, Masato, Gilbert, Rebekah S, Tokuhara, Yuka, Fujihashi, Keiko, Kunisawa, Jun, Yuki, Yoshikazu, Kiyono, Hiroshi, McGhee, Jerry R, Fujihashi, Kohtaro
Published in PloS one (02.04.2013)
Published in PloS one (02.04.2013)
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Journal Article
Intractable Absence Seizures in Hyperinsulinism-Hyperammonemia Syndrome
Nakano, Kousuke, MD, Kobayashi, Katsuhiro, MD, Okano, Yoshiyuki, MD, Aso, Kazuyoshi, MD, Ohtsuka, Yoko, MD
Published in Pediatric neurology (01.08.2012)
Published in Pediatric neurology (01.08.2012)
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Melanin-concentrating hormone receptor 1 antagonists: Synthesis, structure–activity relationship, docking studies, and biological evaluation of 2,3,4,5-tetrahydro-1H-3-benzazepine derivatives
Kasai, Shizuo, Kamaura, Masahiro, Kamata, Makoto, Aso, Kazuyoshi, Ogino, Hitomi, Nakano, Yoshihide, Watanabe, Kaoru, Kaisho, Tomoko, Tawada, Michiko, Nagisa, Yasutaka, Takekawa, Shiro, Kato, Koki, Suzuki, Nobuhiro, Ishihara, Yuji
Published in Bioorganic & medicinal chemistry (01.11.2011)
Published in Bioorganic & medicinal chemistry (01.11.2011)
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A Molecular Mucosal Adjuvant To Enhance Immunity Against Pneumococcal Infection In The Elderly
Fukuyama, Yoshiko, Ikeda, Yorihiko, Ohori, Junichiro, Sugita, Gen, Aso, Kazuyoshi, Fujihashi, Keiko, Briles, David E, McGhee, Jerry R, Fujihashi, Kohtaro
Published in Immune network (01.02.2015)
Published in Immune network (01.02.2015)
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Journal Article
Spectrum of glutamate dehydrogenase mutations in Japanese patients with congenital hyperinsulinism and hyperammonemia syndrome
Aso, Kazuyoshi, Okano, Yoshiyuki, Takeda, Taisuke, Sakamoto, Osamu, Ban, Kyoko, Iida, Kazumi, Yamano, Tsunekazu, Shintaku, Haruo
Published in Osaka City medical journal (01.06.2011)
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Published in Osaka City medical journal (01.06.2011)
Journal Article
A Molecular Mucosal Adjuvant To Enhance Immunity Against Pneumococcal Infection In The Elderly
Fukuyama, Yoshiko, Ikeda, Yorihiko, Ohori, Junichiro, Sugita, Gen, Aso, Kazuyoshi, Fujihashi, Keiko, Briles, David E, McGhee, Jerry R, Fujihashi, Kohtaro
Published in Immune network (2015)
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Published in Immune network (2015)
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Identification of a novel series of potent and selective CCR6 inhibitors as biological probes
Tawaraishi, Taisuke, Sakauchi, Nobuki, Hidaka, Kousuke, Yoshikawa, Kyoko, Okui, Toshitake, Kuno, Haruhiko, Chisaki, Ikumi, Aso, Kazuyoshi
Published in Bioorganic & medicinal chemistry letters (01.10.2018)
Published in Bioorganic & medicinal chemistry letters (01.10.2018)
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Design, synthesis, and pharmacological evaluation of 4-azolyl-benzamide derivatives as novel GPR52 agonists
Tokumaru, Kazuyuki, Ito, Yoshiteru, Nomura, Izumi, Nakahata, Takashi, Shimizu, Yuji, Kurimoto, Emi, Aoyama, Kazunobu, Aso, Kazuyoshi
Published in Bioorganic & medicinal chemistry (15.06.2017)
Published in Bioorganic & medicinal chemistry (15.06.2017)
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Biochemical and structural analysis of the interaction between β-amyloid and fibrinogen
Zamolodchikov, Daria, Berk-Rauch, Hanna E., Oren, Deena A., Stor, Daniel S., Singh, Pradeep K., Kawasaki, Masanori, Aso, Kazuyoshi, Strickland, Sidney, Ahn, Hyung Jin
Published in Blood (25.08.2016)
Published in Blood (25.08.2016)
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Antimalarial proteasome inhibitor reveals collateral sensitivity from intersubunit interactions and fitness cost of resistance
Kirkman, Laura A., Zhan, Wenhu, Visone, Joseph, Dziedziech, Alexis, Singh, Pradeep K., Fan, Hao, Tong, Xinran, Bruzual, Igor, Hara, Ryoma, Kawasaki, Masanori, Imaeda, Toshihiro, Okamoto, Rei, Sato, Kenjiro, Michino, Mayako, Alvaro, Elena Fernandez, Guiang, Liselle F., Sanz, Laura, Mota, Daniel J., Govindasamy, Kavitha, Wang, Rong, Ling, Yan, Tumwebaze, Patrick K., Sukenick, George, Shi, Lei, Vendome, Jeremie, Bhanot, Purnima, Rosenthal, Philip J., Aso, Kazuyoshi, Foley, Michael A., Cooper, Roland A., Kafsack, Bjorn, Doggett, J. Stone, Nathan, Carl F., Lin, Gang
Published in Proceedings of the National Academy of Sciences - PNAS (17.07.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (17.07.2018)
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Discovery of 1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazoles as novel class of corticotropin releasing factor 1 receptor antagonists
Kojima, Takuto, Mochizuki, Michiyo, Takai, Takafumi, Hoashi, Yasutaka, Morimoto, Sachie, Seto, Masaki, Nakamura, Minoru, Kobayashi, Katsumi, Sako, Yuu, Tanaka, Maiko, Kanzaki, Naoyuki, Kosugi, Yohei, Yano, Takahiko, Aso, Kazuyoshi
Published in Bioorganic & medicinal chemistry (15.05.2018)
Published in Bioorganic & medicinal chemistry (15.05.2018)
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Design, Synthesis, and Optimization of Macrocyclic Peptides as Species-Selective Antimalaria Proteasome Inhibitors
Zhang, Hao, Ginn, John, Zhan, Wenhu, Liu, Yi J., Leung, Annie, Toita, Akinori, Okamoto, Rei, Wong, Tzu-Tshin, Imaeda, Toshihiro, Hara, Ryoma, Yukawa, Takafumi, Michino, Mayako, Vendome, Jeremie, Beuming, Thijs, Sato, Kenjiro, Aso, Kazuyoshi, Meinke, Peter T., Nathan, Carl F., Kirkman, Laura A., Lin, Gang
Published in Journal of medicinal chemistry (14.07.2022)
Published in Journal of medicinal chemistry (14.07.2022)
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