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Published in Nature communications (21.05.2019)
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Small molecule inhibition of cGAS reduces interferon expression in primary macrophages from autoimmune mice
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Published in Nature communications (29.09.2017)
Published in Nature communications (29.09.2017)
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Discovery of an Orally Bioavailable, Brain-Penetrating, in Vivo Active Phosphodiesterase 2A Inhibitor Lead Series for the Treatment of Cognitive Disorders
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Published in Journal of medicinal chemistry (28.09.2017)
Published in Journal of medicinal chemistry (28.09.2017)
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Publisher Correction: Small molecule inhibition of cGAS reduces interferon expression in primary macrophages from autoimmune mice
Vincent, Jessica, Adura, Carolina, Gao, Pu, Luz, Antonio, Lama, Lodoe, Asano, Yasutomi, Okamoto, Rei, Imaeda, Toshihiro, Aida, Jumpei, Rothamel, Katherine, Gogakos, Tasos, Steinberg, Joshua, Reasoner, Seth, Aso, Kazuyoshi, Tuschl, Thomas, Patel, Dinshaw J, Glickman, J Fraser, Ascano, Manuel
Published in Nature communications (23.11.2017)
Published in Nature communications (23.11.2017)
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Discovery, synthesis and biological evaluation of isoquinolones as novel and highly selective JNK inhibitors ( 2)
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Published in Bioorganic & medicinal chemistry (15.04.2008)
Published in Bioorganic & medicinal chemistry (15.04.2008)
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The first asymmetric synthesis of a dopamine D1 agonist, dihydrexidine, employing asymmetric conjugate addition technology
Asano, Yasutomi, Yamashita, Mitsuaki, Nagai, Kazushige, Kuriyama, Masami, Yamada, Ken-ichi, Tomioka, Kiyoshi
Published in Tetrahedron letters (26.11.2001)
Published in Tetrahedron letters (26.11.2001)
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Pharmacological characterization of synthetic serine palmitoyltransferase inhibitors by biochemical and cellular analyses
Adachi, Ryutaro, Asano, Yasutomi, Ogawa, Kazumasa, Oonishi, Motomi, Tanaka, Yukiya, Kawamoto, Tomohiro
Published in Biochemical and biophysical research communications (18.03.2018)
Published in Biochemical and biophysical research communications (18.03.2018)
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THE CHIRAL LIGAND-CATALYZED ENANTIOSELECTIVE CONJUGATE ADDITION OF ORGANOLITHIUM TO BHA ENOATE
ASANO, Yasutomi, IIDA, Akira, TOMIOKA, Kiyoshi
Published in Chemical & pharmaceutical bulletin (01.01.1998)
Published in Chemical & pharmaceutical bulletin (01.01.1998)
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Antitumor activity of a novel and orally available inhibitor of serine palmitoyltransferase
Yaguchi, Masahiro, Shibata, Sachio, Satomi, Yoshinori, Hirayama, Megumi, Adachi, Ryutaro, Asano, Yasutomi, Kojima, Takuto, Hirata, Yasuhiro, Mizutani, Akio, Kiba, Atsushi, Sagiya, Yoji
Published in Biochemical and biophysical research communications (11.03.2017)
Published in Biochemical and biophysical research communications (11.03.2017)
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Discovery of novel serine palmitoyltransferase inhibitors as cancer therapeutic agents
Kojima, Takuto, Asano, Yasutomi, Kurasawa, Osamu, Hirata, Yasuhiro, Iwamura, Naoki, Wong, Tzu-Tshin, Saito, Bunnai, Tanaka, Yuta, Arai, Ryosuke, Yonemori, Kazuko, Miyamoto, Yasufumi, Sagiya, Yoji, Yaguchi, Masahiro, Shibata, Sachio, Mizutani, Akio, Sano, Osamu, Adachi, Ryutaro, Satomi, Yoshinori, Hirayama, Megumi, Aoyama, Kazunobu, Hiura, Yuto, Kiba, Atsushi, Kitamura, Shuji, Imamura, Shinichi
Published in Bioorganic & medicinal chemistry (15.05.2018)
Published in Bioorganic & medicinal chemistry (15.05.2018)
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Identification of Novel, Potent, and Orally Available GCN2 Inhibitors with Type I Half Binding Mode
Fujimoto, Jun, Kurasawa, Osamu, Takagi, Terufumi, Liu, Xin, Banno, Hiroshi, Kojima, Takuto, Asano, Yasutomi, Nakamura, Akito, Nambu, Tadahiro, Hata, Akito, Ishii, Tsuyoshi, Sameshima, Tomoya, Debori, Yasuyuki, Miyamoto, Maki, Klein, Michael G, Tjhen, Richard, Sang, Bi-Ching, Levin, Irena, Lane, Scott Weston, Snell, Gyorgy P, Li, Ke, Kefala, Georgia, Hoffman, Isaac D, Ding, Steve C, Cary, Douglas R, Mizojiri, Ryo
Published in ACS medicinal chemistry letters (10.10.2019)
Published in ACS medicinal chemistry letters (10.10.2019)
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HETEROCYCLIC COMPOUND
ASANO, Yasutomi, SASAKI, Shinobu, SETO, Masaki, ANDO, Haruhi, TAKAMI, Kazuaki
Year of Publication 02.04.2020
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Year of Publication 02.04.2020
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Discovery, synthesis and biological evaluation of isoquinolones as novel and highly selective JNK inhibitors ( 1)
Asano, Yasutomi, Kitamura, Shuji, Ohra, Taiichi, Aso, Kazuyoshi, Igata, Hideki, Tamura, Tomoko, Kawamoto, Tomohiro, Tanaka, Toshimasa, Sogabe, Satoshi, Matsumoto, Shin-ichi, Yamaguchi, Masashi, Kimura, Hiroyuki, Itoh, Fumio
Published in Bioorganic & medicinal chemistry (15.04.2008)
Published in Bioorganic & medicinal chemistry (15.04.2008)
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CONDENSED-CYCLIC COMPOUND
ASANO, Yasutomi, SASAKI, Shinobu, SETO, Masaki, ANDO, Haruhi, KITAMURA, Shuji, SATO, Ayumu, TAKAMI, Kazuaki, MAEZAKI, Hironobu, SWANN, Steve L
Year of Publication 02.04.2020
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Year of Publication 02.04.2020
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Enantioselective Hydrogen Atom Transfer Reactions: Synthesis of N-Acyl-α-Amino Acid Esters
Sibi, Mukund P., Asano, Yasutomi, Sausker, Justin B.
Published in Angewandte Chemie (International ed.) (01.04.2001)
Published in Angewandte Chemie (International ed.) (01.04.2001)
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LIU XIN, KOJIMA TAKUTO, TAKAGI TERUFUMI, KURASAWA OSAMU, FUJIMOTO JUN, BANNO HIROSHI, ASANO YASUTOMI, CARY DOUGLAS ROBERT
Year of Publication 08.04.2019
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Year of Publication 08.04.2019
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HETEROCYCLIC COMPOUND
ASANO, Yasutomi, FUJIMOTO, Jun, BANNO, Hiroshi, KOJIMA, Takuto, LIU, Xin, KURASAWA, Osamu, TAKAGI, Terufumi, CARY, Douglas Robert
Year of Publication 15.02.2018
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Year of Publication 15.02.2018
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