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Published in EMBO molecular medicine (01.06.2018)
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Published in Bioorganic & medicinal chemistry (01.07.2017)
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Published in eLife (19.05.2017)
Published in eLife (19.05.2017)
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Design and Synthesis of Potent Inhibitor of Apoptosis (IAP) Proteins Antagonists Bearing an Octahydropyrrolo[1,2‑a]pyrazine Scaffold as a Novel Proline Mimetic
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Published in Journal of medicinal chemistry (14.02.2013)
Published in Journal of medicinal chemistry (14.02.2013)
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Published in Bioorganic & medicinal chemistry (15.09.2013)
Published in Bioorganic & medicinal chemistry (15.09.2013)
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Synthetic Studies toward GKK1032s, Novel Antibiotic Antitumor Agents: Enantioselective Synthesis of the Fully Elaborated Tricyclic Core via an Intramolecular Diels−Alder Cycloaddition
Asano, Moriteru, Inoue, Munenori, Watanabe, Kazuhiro, Abe, Hideki, Katoh, Tadashi
Published in Journal of organic chemistry (01.09.2006)
Published in Journal of organic chemistry (01.09.2006)
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The identification and pharmacological evaluation of potent, selective and orally available ACC1 inhibitor
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Published in Bioorganic & medicinal chemistry letters (01.12.2019)
Published in Bioorganic & medicinal chemistry letters (01.12.2019)
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Design and synthesis of a novel 1H-pyrrolo[3,2-b]pyridine-3-carboxamide derivative as an orally available ACC1 inhibitor
Mizojiri, Ryo, Nii, Noriyuki, Asano, Moriteru, Sasaki, Masako, Satoh, Yoshihiko, Yamamoto, Yukiko, Sumi, Hiroyuki, Maezaki, Hironobu
Published in Bioorganic & medicinal chemistry (15.06.2019)
Published in Bioorganic & medicinal chemistry (15.06.2019)
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Synthesis and biological evaluation of novel selective androgen receptor modulators (SARM-s) Part Ill: Discovery of 4-(5-oxopyrrolidine-1-yl) benzonitrile derivative 2f as a clinical candidate
Aikawa, Katsuji, Asano, Moriteru, Ono, Koji, Habuka, Noriyuki, Yano, Jason, Wilson, Keith, Fujita, Hisashi, Kandori, Hitoshi, Hara, Takahito, Morimoto, Megumi, Santou, Takashi, Yamaoka, Masuo, Nakayama, Masaharu, Hasuoka, Atsushi
Published in Bioorganic & medicinal chemistry (01.07.2017)
Published in Bioorganic & medicinal chemistry (01.07.2017)
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Discovery of Novel Selective Acetyl-CoA Carboxylase (ACC) 1 Inhibitors
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Published in Journal of medicinal chemistry (08.02.2018)
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Synthesis and biological evaluation of novel selective androgen receptor modulators (SARMs). Part II: Optimization of 4-(pyrrolidin-1-yl)benzonitrile derivatives
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Published in Bioorganic & medicinal chemistry letters (01.05.2017)
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