Selexipag: An Oral and Selective IP Prostacyclin Receptor Agonist for the Treatment of Pulmonary Arterial Hypertension
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Published in Journal of medicinal chemistry (24.09.2015)
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NS-187, a potent and selective dual Bcr-Abl/Lyn tyrosine kinase inhibitor, is a novel agent for imatinib-resistant leukemia
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Published in Blood (01.12.2005)
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2-{4-[(5,6-Diphenylpyrazin-2-yl)(isopropyl)amino]butoxy}-N-(methylsulfonyl)acetamide (NS-304), an Orally Available and Long-Acting Prostacyclin Receptor Agonist Prodrug
Kuwano, Keiichi, Hashino, Asami, Asaki, Tetsuo, Hamamoto, Taisuke, Yamada, Tetsuhiro, Okubo, Kaori, Kuwabara, Kenji
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Published in The Journal of pharmacology and experimental therapeutics (01.09.2007)
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NS-187 (INNO-406), a Bcr-Abl/Lyn Dual Tyrosine Kinase Inhibitor
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Book Review
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Design and synthesis of 3-substituted benzamide derivatives as Bcr-Abl kinase inhibitors
Asaki, Tetsuo, Sugiyama, Yukiteru, Hamamoto, Taisuke, Higashioka, Masaya, Umehara, Masato, Naito, Haruna, Niwa, Tomoko
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
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Structure–activity studies on 1,3-dioxane-2-carboxylic acid derivatives, a novel class of subtype-selective peroxisome proliferator-activated receptor α (PPARα) agonists
Asaki, Tetsuo, Aoki, Tomiyoshi, Hamamoto, Taisuke, Sugiyama, Yukiteru, Ohmachi, Shinji, Kuwabara, Kenji, Murakami, Kohji, Todo, Makoto
Published in Bioorganic & medicinal chemistry (15.01.2008)
Published in Bioorganic & medicinal chemistry (15.01.2008)
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Structural factors contributing to the Abl/Lyn dual inhibitory activity of 3-substituted benzamide derivatives
Horio, Tatsuya, Hamasaki, Tomohiro, Inoue, Toshihiko, Wakayama, Tatsushi, Itou, Shinsaku, Naito, Haruna, Asaki, Tetsuo, Hayase, Hiroki, Niwa, Tomoko
Published in Bioorganic & medicinal chemistry letters (15.05.2007)
Published in Bioorganic & medicinal chemistry letters (15.05.2007)
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Discovery of a novel class of 1,3-dioxane-2-carboxylic acid derivatives as subtype-selective peroxisome proliferator-activated receptor α (PPARα) agonists
Aoki, Tomiyoshi, Asaki, Tetsuo, Hamamoto, Taisuke, Sugiyama, Yukiteru, Ohmachi, Shinji, Kuwabara, Kenji, Murakami, Kohji, Todo, Makoto
Published in Bioorganic & medicinal chemistry (15.03.2008)
Published in Bioorganic & medicinal chemistry (15.03.2008)
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Structure–activity relationship study on the 6-membered heteroaromatic ring system of diphenylpyrazine-type prostacyclin receptor agonists
Asaki, Tetsuo, Hamamoto, Taisuke, Sugiyama, Yukiteru, Kuwano, Keiichi, Kuwabara, Kenji, Niwa, Tomoko
Published in Bioorganic & medicinal chemistry (01.12.2007)
Published in Bioorganic & medicinal chemistry (01.12.2007)
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Journal Article
2-[4-[(5,6-diphenylpyrazin-2-yl)(isopropyl)amino]butoxy]-N-(methylsulfonyl)acetamide (NS-304), an orally available and long-acting prostacyclin receptor agonist prodrug
Kuwano, Keiichi, Hashino, Asami, Asaki, Tetsuo, Hamamoto, Taisuke, Yamada, Tetsuhiro, Okubo, Kaori, Kuwabara, Kenji
Published in The Journal of pharmacology and experimental therapeutics (01.09.2007)
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Published in The Journal of pharmacology and experimental therapeutics (01.09.2007)
Journal Article
Structure-activity studies on 1,3-dioxane-2-carboxylic acid derivatives, a novel class of subtype-selective peroxisome proliferator-activated receptor a (PPARa) agonists
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Published in Bioorganic & medicinal chemistry (2008)
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Published in Bioorganic & medicinal chemistry (2008)
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Structural factors contributing to the Al/Lyn dual inhibitory activity of 3-substituted benzamide derivatives
HORIO, Tatsuya, HAMASAKI, Tomohiro, INOUE, Toshihiko, WAKAYAMA, Tatsushi, ITOU, Shinsaku, NAITO, Haruna, ASAKI, Tetsuo, HAYASE, Hiroki, NIWA, Tomoko
Published in Bioorganic & medicinal chemistry letters (2007)
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Published in Bioorganic & medicinal chemistry letters (2007)
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