Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 1. Synthesis and Structure−Activity Relationship of a Class of Human Immunodeficiency Virus type 1 Integrase Inhibitors
Pasquini, Serena, Mugnaini, Claudia, Tintori, Cristina, Botta, Maurizio, Trejos, Alejandro, Arvela, Riina K, Larhed, Mats, Witvrouw, Myriam, Michiels, Martine, Christ, Frauke, Debyser, Zeger, Corelli, Federico
Published in Journal of medicinal chemistry (28.08.2008)
Published in Journal of medicinal chemistry (28.08.2008)
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Journal Article
Highly Regioselective Internal Heck Arylation of Hydroxyalkyl Vinyl Ethers by Aryl Halides in Water
Arvela, Riina K, Pasquini, Serena, Larhed, Mats
Published in Journal of organic chemistry (17.08.2007)
Published in Journal of organic chemistry (17.08.2007)
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Synthesis, X-ray Analysis, and Biological Evaluation of a New Class of Stereopure Lactam-Based HIV-1 Protease Inhibitors
Wu, Xiongyu, Öhrngren, Per, Joshi, Advait A, Trejos, Alejandro, Persson, Magnus, Arvela, Riina K, Wallberg, Hans, Vrang, Lotta, Rosenquist, Åsa, Samuelsson, Bertil B, Unge, Johan, Larhed, Mats
Published in Journal of medicinal chemistry (22.03.2012)
Published in Journal of medicinal chemistry (22.03.2012)
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Rapid cyanation of aryl iodides in water using microwave promotion
Arvela, RK, Leadbeater, NE, Torenius, HM, Tye, H
Published in Organic & biomolecular chemistry (07.04.2003)
Published in Organic & biomolecular chemistry (07.04.2003)
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Journal Article
Investigations on the 4-quinolone-3-carboxylic acid motif. 1. Synthesis-activity relationship of a class of human immunodeficiency virus type 1 integrase inhibitors
Pasquini, Serena, Mugnaini, Claudia, Tintori, Cristina, Botta, Maurizio, Trejos, Alejandro, Arvela, Riina K., Larhed, Mats, Witvrouw, Myriam, Michiels, Martine, Christ, Frauke, Debyser, Zeger, Corelli, Federico
Published in Journal of medicinal chemistry (28.08.2008)
Published in Journal of medicinal chemistry (28.08.2008)
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Journal Article
PHARMACOLOGICALLY ACTIVE QUINAZOLINEDIONE DERIVATIVES
HOGLUND IISA, HIETANEN ARI, VESALAINEN ANNIINA, PRUSIS PETERIS, ARVELA RIINA, HEIKKINEN TERHI, TORMAKANGAS OLLI
Year of Publication 06.01.2017
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Year of Publication 06.01.2017
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N-PROP-2-YNYL CARBOXAMIDE DERIVATIVES AND THEIR USE AS TRPA1 ANTAGONISTS
SALO HARRI, HOLM PATRIK, ROSLUND MATTIAS, PRUSIS PETERIS, ARVELA RIINA, HEIKKINEN TERHI
Year of Publication 08.06.2015
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Year of Publication 08.06.2015
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N-PROP-2-YNYL CARBOXAMIDE DERIVATIVES AND THEIR USE AS TRPA1 ANTAGONISTS
HEIKKINEN, TERHI, PRUSIS, PETERIS, HOLM, PATRIK, SALO, HARRI, ROSLUND, MATTIAS, ARVELA, RIINA
Year of Publication 28.10.2021
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Year of Publication 28.10.2021
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N-PROP-2-YNYL CARBOXAMIDE DERIVATIVES AND THEIR USE AS TRPA1 ANTAGONISTS
HEIKKINEN, TERHI, PRUSIS, PETERIS, HOLM, PATRIK, SALO, HARRI, ROSLUND, MATTIAS, ARVELA, RIINA
Year of Publication 10.11.2020
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Year of Publication 10.11.2020
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N-prop-2-ynyl carboxamide derivatives and their use as trpa1 antagonists
Roslund, Mattias, Salo, Harri, Heikkinen, Terhi, Holm, Patrik, Arvela, Riina, Prusis, Peteris
Year of Publication 27.07.2018
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Year of Publication 27.07.2018
Patent
N-PROP-2-YNYL CARBOXAMIDE DERIVATIVES AND THEIR USE AS TRPA1 ANTAGONISTS
HEIKKINEN, Terhi, SALO, Harri, ROSLUND, Mattias, ARVELA, Riina, HOLM, Patrik, PRUSIS, Peteris
Year of Publication 28.02.2018
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Year of Publication 28.02.2018
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