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In Vitro Intrinsic Clearance-Based Optimization of N 3-Phenylpyrazinones as Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

In Vitro Intrinsic Clearance-Based Optimization of N 3-Phenylpyrazinones as Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

by Hartz, Richard A, Ahuja, Vijay T, Rafalski, Maria, Schmitz, William D, Brenner, Allison B, Denhart, Derek J, Ditta, Jonathan L, Deskus, Jeffrey A, Yue, Eddy W, Arvanitis, Argyrios G, Lelas, Snjezana, Li, Yu-Wen, Molski, Thaddeus F, Wong, Harvey, Grace, James E, Lentz, Kimberley A, Li, Jianqing, Lodge, Nicholas J, Zaczek, Robert, Combs, Andrew P, Olson, Richard E, Mattson, Ronald J, Bronson, Joanne J, Macor, John E
Published in Journal of medicinal chemistry (23.07.2009)

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Synthesis and evaluation of 2-anilino-3-phenylsulfonyl-6-methylpyridines as corticotropin-releasing factor1 receptor ligands

Synthesis and evaluation of 2-anilino-3-phenylsulfonyl-6-methylpyridines as corticotropin-releasing factor1 receptor ligands

by HARTZ, Richard A, ARVANITIS, Argyrios G, ARNOLD, Charles, RESCINITO, Joseph P, HUNG, Kimberly L, GE ZHANG, WONG, Harvey, LANGLEY, David R, GILLIGAN, Paul J, TRAINOR, George L
Published in Bioorganic & medicinal chemistry letters (15.02.2006)

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Synthesis, Structure−Activity Relationships, and In Vivo Evaluation of N 3-Phenylpyrazinones as Novel Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

Synthesis, Structure−Activity Relationships, and In Vivo Evaluation of N 3-Phenylpyrazinones as Novel Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

by Hartz, Richard A, Ahuja, Vijay T, Arvanitis, Argyrios G, Rafalski, Maria, Yue, Eddy W, Denhart, Derek J, Schmitz, William D, Ditta, Jonathan L, Deskus, Jeffrey A, Brenner, Allison B, Hobbs, Frank W, Payne, Joseph, Lelas, Snjezana, Li, Yu-Wen, Molski, Thaddeus F, Mattson, Gail K, Peng, Yong, Wong, Harvey, Grace, James E, Lentz, Kimberley A, Qian-Cutrone, Jingfang, Zhuo, Xiaoliang, Shu, Yue-Zhong, Lodge, Nicholas J, Zaczek, Robert, Combs, Andrew P, Olson, Richard E, Bronson, Joanne J, Mattson, Ronald J, Macor, John E
Published in Journal of medicinal chemistry (23.07.2009)

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Synthesis and structure–activity relationships of pyrido[3,2-b]pyrazin-3(4H)-ones and pteridin-7(8H)-ones as corticotropin-releasing factor-1 receptor antagonists

Synthesis and structure–activity relationships of pyrido[3,2-b]pyrazin-3(4H)-ones and pteridin-7(8H)-ones as corticotropin-releasing factor-1 receptor antagonists

by Dzierba, Carolyn D., Sielecki, Thais M., Arvanitis, Argyrios G., Galka, Amy, Johnson, Tricia L., Takvorian, Amy G., Rafalski, Maria, Kasireddy-Polam, Padmaja, Vig, Shikha, Dasgupta, Bireshwar, Zhang, Ge, Molski, Thaddeus F., Wong, Harvey, Zaczek, Robert C., Lodge, Nicholas J., Combs, Andrew P., Gilligan, Paul J., Trainor, George L., Bronson, Joanne J., Macor, John E.
Published in Bioorganic & medicinal chemistry letters (01.08.2012)

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3-4-7-23--4--1--1--3- HYDROXYL KETO AND GLUCURONIDE DERIVATIVES OF 3-4-7H-PYRROLO[23-D]PYRIMIDIN-4-YL-1H-PYRAZOL-1-YL-3-CYCLOPENTYLPROPANENITRILE

3-4-7-23--4--1--1--3- HYDROXYL KETO AND GLUCURONIDE DERIVATIVES OF 3-4-7H-PYRROLO[23-D]PYRIMIDIN-4-YL-1H-PYRAZOL-1-YL-3-CYCLOPENTYLPROPANENITRILE

by LI MEI, NEDZA FRANK M, SHILLING ADAM, SHEPARD STACEY, GALYA LAURINE G, RODGERS JAMES D, ARVANITIS ARGYRIOS G
Year of Publication 27.11.2018

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Patent

HYDROXYL, KETO, AND GLUCURONIDE DERIVATIVES OF 3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROPANENITRILE

HYDROXYL, KETO, AND GLUCURONIDE DERIVATIVES OF 3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROPANENITRILE

by LEE MAY, FRANK M NEDZA, SHEPARD STACEY, ADAM SHILLING, LAURINE G GALYA, RODGERS JAMES D, ARVANITIS ARGYRIOS G
Year of Publication 28.12.2017

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Patent

3-4-7-23--4--1--1--3- HYDROXYL KETO AND GLUCURONIDE DERIVATIVES OF 3-4-7H-PYRROLO[23-D]PYRIMIDIN-4-YL-1H-PYRAZOL-1-YL-3-CYCLOPENTYLPROPANENITRILE

3-4-7-23--4--1--1--3- HYDROXYL KETO AND GLUCURONIDE DERIVATIVES OF 3-4-7H-PYRROLO[23-D]PYRIMIDIN-4-YL-1H-PYRAZOL-1-YL-3-CYCLOPENTYLPROPANENITRILE

by LI MEI, NEDZA FRANK M, SHILLING ADAM, SHEPARD STACEY, GALYA LAURINE G, RODGERS JAMES D, ARVANITIS ARGYRIOS G
Year of Publication 29.08.2017

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Patent

HYDROXYL, KETO, AND GLUCURONIDE DERIVATIVES OF 3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROPANENITRILE

HYDROXYL, KETO, AND GLUCURONIDE DERIVATIVES OF 3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROPANENITRILE

by LEE MAY, FRANK M NEDZA, SHEPARD STACEY, ADAM SHILLING, LAURINE G GALYA, RODGERS JAMES D, ARVANITIS ARGYRIOS G
Year of Publication 21.04.2016

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Patent

Imidazo[4,5- b]pyridines as corticotropin releasing factor receptor ligands

Imidazo[4,5- b]pyridines as corticotropin releasing factor receptor ligands

by Arvanitis, Argyrios G., Rescinito, Joseph T., Arnold, Charles R., Wilde, Richard G., Cain, Gary A., Sun, Jung Hui, Yan, Jia-Sheng, Teleha, Christopher A., Fitzgerald, Lawrence W., McElroy, John, Zaczek, Robert, Hartig, Paul R., Grossman, Scott, Arneric, Stephen P., Gilligan, Paul J., Olson, Richard E., Robertson, David W.
Published in Bioorganic & medicinal chemistry letters (06.01.2003)

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Journal Article

CRF Ligands via suzuki and negishi couplings of 3-pyridyl boronic acids or halides with 2-benzyloxy-4-chloro-3-nitropyridine

CRF Ligands via suzuki and negishi couplings of 3-pyridyl boronic acids or halides with 2-benzyloxy-4-chloro-3-nitropyridine

by Arvanitis, Argyrios G., Arnold, Charles R., Fitzgerald, Lawrence W., Frietze, William E., Olson, Richard E., Gilligan, Paul J., Robertson, David W.
Published in Bioorganic & medicinal chemistry letters (20.01.2003)

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Journal Article

HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINE AND PYRROLO[2,3-b]PYRIMIDINE AS JANUS KINASE INHIBITORS

HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINE AND PYRROLO[2,3-b]PYRIMIDINE AS JANUS KINASE INHIBITORS

by JALLURI RAVI KUMAR, RAFALSKI MARIA, FALAHATPISHEH NIKOO, STORACE LOUIS, MADUSKUIE THOMAS P, SHEPARD STACEY, FRIDMAN JORDAN S, VADDI KRISHNA, WANG HAISHENG, RODGERS JAMES D, ARVANITIS ARGYRIOS G
Year of Publication 05.11.2015

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Patent

METABOLITES OF THE JANUS KINASE INHIBITOR (R)-3-(4-(7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROPANENITRILE

METABOLITES OF THE JANUS KINASE INHIBITOR (R)-3-(4-(7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROPANENITRILE

by SHI JACK GUOEN, RODGERS JAMES D, ARVANITIS ARGYRIOS G
Year of Publication 11.05.2010

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Patent

Imidazo[4,5- c]pyridines as corticotropin releasing factor receptor ligands

Imidazo[4,5- c]pyridines as corticotropin releasing factor receptor ligands

by Arvanitis, Argyrios G., Rescinito, Joseph T., Arnold, Charles R., Wilde, Richard G., Fitzgerald, Lawrence W., Zaczek, Robert, Hartig, Paul R., Grossman, Scott, Arneric, Stephen P., Gilligan, Paul J., Olson, Richard E., Robertson, David W.
Published in Bioorganic & medicinal chemistry letters (06.01.2003)

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Journal Article

HYDROXYL, KETO, AND GLUCURONIDE DERIVATIVES OF 3-(4-(7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROPANENITRILE

HYDROXYL, KETO, AND GLUCURONIDE DERIVATIVES OF 3-(4-(7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROPANENITRILE

by LI MEI, NEDZA FRANK M, SHILLING ADAM, SHEPARD STACEY, GALYA LAURINE G, RODGERS JAMES D, ARVANITIS ARGYRIOS G
Year of Publication 18.09.2012

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Patent

N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-D]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-D]PYRIMIDINES AS JANUS KINASE INHIBITORS

N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-D]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-D]PYRIMIDINES AS JANUS KINASE INHIBITORS

by STORACE LOUIS, SHEPARD STACEY, FOLMER BEVERLY, SHAO LIXIN, ZHU WENYU, WANG HAISHENG, RODGERS JAMES D, ARVANITIS ARGYRIOS G, GLENN JOSEPH P
Year of Publication 12.04.2012

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Patent

Corrections to In Vitro Intrinsic Clearance-Based Optimization of N 3-Phenylpyrazinones as Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

Corrections to In Vitro Intrinsic Clearance-Based Optimization of N 3-Phenylpyrazinones as Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

by Hartz, Richard A., Ahuja, Vijay T., Rafalski, Maria, Schmitz, William D., Brenner, Allison B., Denhart, Derek J., Ditta, Jonathan L., Deskus, Jeffrey A., Yue, Eddy W., Arvanitis, Argyrios G., Lelas, Snjezana, Li, Yu-Wen, Molski, Thaddeus F., Wong, Harvey, Grace, James E., Lentz, Kimberley A., Li, Jianqing, Lodge, Nicholas J., Zaczek, Robert, Combs, Andrew P., Olson, Richard E., Mattson, Ronald J., Bronson, Joanne J., Macor, John E.
Published in Journal of medicinal chemistry (24.09.2009)

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Journal Article

In Vitro Intrinsic Clearance-Based Optimization of N3-Phenylpyrazinones as Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

In Vitro Intrinsic Clearance-Based Optimization of N3-Phenylpyrazinones as Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

by HARTZ, Richard A, AHUJA, Vijay T, LELAS, Snjezana, LI, Yu-Wen, MOLSKI, Thaddeus F, WONG, Harvey, GRACE, James E, LENTZ, Kimberley A, JIANQING LI, LODGE, Nicholas J, ZACZEK, Robert, COMBS, Andrew P, RAFALSKI, Maria, OLSON, Richard E, MATTSON, Ronald J, BRONSON, Joanne J, MACOR, John E, SCHMITZ, William D, BRENTER, Allison B, DENHART, Derek J, DITTA, Jonathan L, DESKUS, Jeffrey A, YUE, Eddy W, ARVANITIS, Argyrios G
Published in Journal of medicinal chemistry (23.07.2009)

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Journal Article

Synthesis, Structure—Activity Relationships, and In Vivo Evaluation of N3-Phenylpyrazinones as Novel Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

Synthesis, Structure—Activity Relationships, and In Vivo Evaluation of N3-Phenylpyrazinones as Novel Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

by HARTZ, Richard A, AHUJA, Vijay T, HOBBS, Frank W, PAYNE, Joseph, LELAS, Snjezana, LI, Yu-Wen, MOLSKI, Thaddeus F, MATTSON, Gail K, YONG PENG, WONG, Harvey, GRACE, James E, LENTZ, Kimberley A, ARVANITIS, Argyrios G, QIAN-CUTRONE, Jingfang, XIAOLIANG ZHUO, SHU, Yue-Zhong, LODGER, Nicholas J, ZACZEK, Robert, COMBS, Andrew P, OLSON, Richard E, BRONSON, Joanne J, MATTSON, Ronald J, MACOR, John E, RAFALSKI, Maria, YUE, Eddy W, DENHART, Derek J, SCHMITZ, William D, DITTA, Jonathan L, DESKUS, Jeffrey A, BRENNER, Allison B
Published in Journal of medicinal chemistry (23.07.2009)

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Synthesis and evaluation of 2-anilino-3-phenylsulfonyl-6-methylpyridines as corticotropin-releasing factor sub(1) receptor ligands

Synthesis and evaluation of 2-anilino-3-phenylsulfonyl-6-methylpyridines as corticotropin-releasing factor sub(1) receptor ligands

by Hartz, Richard A, Arvanitis, Argyrios G, Arnold, Charles, Rescinito, Joseph P, Hung, Kimberly L, Zhang, Ge, Wong, Harvey, Langley, David R, Gilligan, Paul J, Trainor, George L
Published in Bioorganic & medicinal chemistry letters (01.02.2006)

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Journal Article

Synthesis and evaluation of 2-anilino-3-phenylsulfonyl-6-methylpyridines as corticotropin-releasing factor 1 receptor ligands

Synthesis and evaluation of 2-anilino-3-phenylsulfonyl-6-methylpyridines as corticotropin-releasing factor 1 receptor ligands

by Hartz, Richard A., Arvanitis, Argyrios G., Arnold, Charles, Rescinito, Joseph P., Hung, Kimberly L., Zhang, Ge, Wong, Harvey, Langley, David R., Gilligan, Paul J., Trainor, George L.
Published in Bioorganic & medicinal chemistry letters (2006)

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