Search Results - "ARMOUR, Duncan" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Maraviroc (UK-427,857), a Potent, Orally Bioavailable, and Selective Small-Molecule Inhibitor of Chemokine Receptor CCR5 with Broad-Spectrum Anti-Human Immunodeficiency Virus Type 1 Activity

Maraviroc (UK-427,857), a Potent, Orally Bioavailable, and Selective Small-Molecule Inhibitor of Chemokine Receptor CCR5 with Broad-Spectrum Anti-Human Immunodeficiency Virus Type 1 Activity

by DORR, Patrick, WESTBY, Mike, WEBSTER, Rob, ARMOUR, Duncan, PRICE, David, STAMMEN, Blanda, WOOD, Anthony, PERROS, Manos, DOBBS, Susan, GRIFFIN, Paul, IRVINE, Becky, MACARTNEY, Malcolm, MORI, Julie, RICKETT, Graham, SMITH-BURCHNELL, Caroline, NAPIER, Carolyn
Published in Antimicrobial Agents and Chemotherapy (01.11.2005)

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Journal Article

The Discovery of the CCR5 Receptor Antagonist, UK-427,857, A New Agent for the Treatment of HIV Infection and AIDS

The Discovery of the CCR5 Receptor Antagonist, UK-427,857, A New Agent for the Treatment of HIV Infection and AIDS

by Wood, Anthony, Armour, Duncan
Published in Progress in Medicinal Chemistry (2005)

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Book Chapter Journal Article

Overcoming hERG affinity in the discovery of maraviroc; a CCR5 antagonist for the treatment of HIV

Overcoming hERG affinity in the discovery of maraviroc; a CCR5 antagonist for the treatment of HIV

by Price, David A, Armour, Duncan, de Groot, Marcel, Leishman, Derek, Napier, Carolyn, Perros, Manos, Stammen, Blanda L, Wood, Anthony
Published in Current topics in medicinal chemistry (01.09.2008)

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Journal Article

The Discovery of CCR5 Receptor Antagonists for the Treatment of HIV Infection: Hit-to-Lead Studies

The Discovery of CCR5 Receptor Antagonists for the Treatment of HIV Infection: Hit-to-Lead Studies

by Armour, Duncan, de Groot, Marcel J., Edwards, Martin, Perros, Manos, Price, David A., Stammen, Blanda L., Wood, Anthony
Published in ChemMedChem (10.07.2006)

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Journal Article

Enantioselective Synthesis of 3,6-Dihydro-1H-pyridin-2-ones: Unexpected Regioselectivity in the Palladium-Catalyzed Decarboxylative Carbonylation of 5-Vinyloxazolidin-2-ones

Enantioselective Synthesis of 3,6-Dihydro-1H-pyridin-2-ones: Unexpected Regioselectivity in the Palladium-Catalyzed Decarboxylative Carbonylation of 5-Vinyloxazolidin-2-ones

by Knight, Julian G, Ainge, Simon W, Harm, Andrew M, Harwood, Simon J, Maughan, Haydn I, Armour, Duncan R, Hollinshead, David M, Jaxa-Chamiec, Albert A
Published in Journal of the American Chemical Society (29.03.2000)

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Journal Article

The Discovery of Tropane-derived CCR5 Receptor Antagonists

The Discovery of Tropane-derived CCR5 Receptor Antagonists

by Armour, Duncan R., De Groot, Marcel J., Price, David A., Stammen, Blanda L. C., Wood, Anthony, Perros, Manos, Burt, Catherine
Published in Chemical biology & drug design (01.04.2006)

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Journal Article

Discovery of 1,5-Benzodiazepines with Peripheral Cholecystokinin (CCK-A) Receptor Agonist Activity. 1. Optimization of the Agonist “Trigger”

Discovery of 1,5-Benzodiazepines with Peripheral Cholecystokinin (CCK-A) Receptor Agonist Activity. 1. Optimization of the Agonist “Trigger”

by Aquino, Christopher J, Armour, Duncan R, Berman, Judd M, Birkemo, Larry S, Carr, Robin A. E, Croom, Dallas K, Dezube, Milana, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, Head, Julie E, Hirst, Gavin C, James, Michael K, Johnson, Michael F, Miller, Laurence J, Queen, Kennedy L, Rimele, Thomas J, Smith, David N, Sugg, Elizabeth E
Published in Journal of medicinal chemistry (19.01.1996)

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Journal Article

Discovery of an Orally Bioavailable NK1 Receptor Antagonist, (2S,3S)-(2-Methoxy-5-tetrazol-1-ylbenzyl)(2-phenylpiperidin-3-yl)amine (GR203040), with Potent Antiemetic Activity

Discovery of an Orally Bioavailable NK1 Receptor Antagonist, (2S,3S)-(2-Methoxy-5-tetrazol-1-ylbenzyl)(2-phenylpiperidin-3-yl)amine (GR203040), with Potent Antiemetic Activity

by Ward, Peter, Armour, Duncan R, Bays, David E, Evans, Brian, Giblin, Gerard M. P, Heron, Nicola, Hubbard, Tania, Liang, Kai, Middlemiss, David
Published in Journal of medicinal chemistry (01.12.1995)

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Journal Article

Overcoming HERG affinity in the discovery of the CCR5 antagonist maraviroc

Overcoming HERG affinity in the discovery of the CCR5 antagonist maraviroc

by Price, David A., Armour, Duncan, de Groot, Marcel, Leishman, Derek, Napier, Carolyn, Perros, Manos, Stammen, Blanda L., Wood, Anthony
Published in Bioorganic & medicinal chemistry letters (01.09.2006)

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Journal Article

Synthesis and applications of tert-alkoxysiloxane linkers in solid-phase chemistry

Synthesis and applications of tert-alkoxysiloxane linkers in solid-phase chemistry

by Meloni, Marco M., White, Peter D., Armour, Duncan, Brown, Richard C.D.
Published in Tetrahedron (08.01.2007)

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Journal Article

Novel silyl linkers for solid-phase synthesis

Novel silyl linkers for solid-phase synthesis

by Meloni, Marco M., Brown, R.C.D., White, Peter D., Armour, Duncan
Published in Tetrahedron letters (19.08.2002)

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Journal Article

Research Letter: The Discovery of Tropane-derived CCR5 Receptor Antagonists

Research Letter: The Discovery of Tropane-derived CCR5 Receptor Antagonists

by Armour, Duncan R, de Groot, Marcel J, Price, David A, Stammen, Blanda LC, Wood, Anthony, Perros, Manos, Burt, Catherine
Published in Chemical biology & drug design (01.04.2006)

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Journal Article

Enantioselective Synthesis of 3,6-Dihydro-1 H -pyridin-2-ones: Unexpected Regioselectivity in the Palladium-Catalyzed Decarboxylative Carbonylation of 5-Vinyloxazolidin-2-ones

Enantioselective Synthesis of 3,6-Dihydro-1 H -pyridin-2-ones: Unexpected Regioselectivity in the Palladium-Catalyzed Decarboxylative Carbonylation of 5-Vinyloxazolidin-2-ones

by Knight, Julian G., Ainge, Simon W., Harm, Andrew M., Harwood, Simon J., Maughan, Haydn I., Armour, Duncan R., Hollinshead, David M., Jaxa-Chamiec, Albert A.
Published in Journal of the American Chemical Society (01.03.2000)

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Journal Article

CCR5 modulators

CCR5 modulators

by ARMOUR DUNCAN R
Year of Publication 29.04.2009

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Patent

AZABICYCLOALKANES AS CCR5 MODULATORS

AZABICYCLOALKANES AS CCR5 MODULATORS

by Price, David Anthony, Wood, Anthony, Edwards, Martin Paul, Armour, Duncan Robert, Perros, Manoussos, Stammen, Blanda Luzia Christa
Year of Publication 26.01.2018

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Patent

AZABICYCLOALKANES AS CCR5 MODULATORS

AZABICYCLOALKANES AS CCR5 MODULATORS

by Price, David Anthony, Wood, Anthony, Edwards, Martin Paul, Armour, Duncan Robert, Perros, Manoussos, Stammen, Blanda Luzia Christa
Year of Publication 03.11.2017

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Patent

AZABICYCLOALKANES AS CCR5 MODULATORS, PHARMACEUTICAL COMPOSITIONS COMPRISING THEREOF AND THEIR USE

AZABICYCLOALKANES AS CCR5 MODULATORS, PHARMACEUTICAL COMPOSITIONS COMPRISING THEREOF AND THEIR USE

by EDWARDS, MARTIN PAUL, PRICE, DAVID ANTHONY, PERROS, MANOUSSOS, ARMOUR, DUNCAN ROBERT, STAMMEN, BLANDA LUZIA CHRISTA, WOOD, ANTHONY
Year of Publication 28.05.2013

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Patent

AZABICYCLOALKANES AS CCR5 MODULATORS

AZABICYCLOALKANES AS CCR5 MODULATORS

by WOOD, Anthony, PERROS, Manoussos, STAMMEN, Blanda, Luzia, Christa, ARMOUR, Duncan, Robert, PRICE, David, Anthony, EDWARDS, Martin, Paul
Year of Publication 10.10.2011

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Patent

AZABICYCLOALKANES AS CCR5 MODULATORS

AZABICYCLOALKANES AS CCR5 MODULATORS

by WOOD ANTHONY, PERROS MANOUSSOS, PRICE DAVID ANTHONY, EDWARDS MARTIN PAUL, ARMOUR DUNCAN ROBERT, STAMMEN BLANDA LUZIA C
Year of Publication 31.08.2011

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Patent

Azabicycloalkan som CCR5-modulatorer

Azabicycloalkan som CCR5-modulatorer

by EDWARDS, MARTIN PAUL, PRICE, DAVID ANTHONY, PERROS, MANOUSSOS, ARMOUR, DUNCAN ROBERT, STAMMEN, BLANDA LUZIA C, WOOD, ANTHONY
Year of Publication 27.06.2011

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Patent

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