Sulfinimidate Esters as an Electrophilic Sulfinimidoyl Motif Source: Synthesis of N‑Protected Sulfilimines from Grignard Reagents
Andresini, Michael, Spennacchio, Mauro, Colella, Marco, Losito, Gianluca, Aramini, Andrea, Degennaro, Leonardo, Luisi, Renzo
Published in Organic letters (03.09.2021)
Published in Organic letters (03.09.2021)
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Journal Article
N−N Bond Formation Using an Iodonitrene as an Umpolung of Ammonia: Straightforward and Chemoselective Synthesis of Hydrazinium Salts
Tota, Arianna, Colella, Marco, Carlucci, Claudia, Aramini, Andrea, Clarkson, Guy, Degennaro, Leonardo, Bull, James A., Luisi, Renzo
Published in Advanced synthesis & catalysis (05.01.2021)
Published in Advanced synthesis & catalysis (05.01.2021)
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Journal Article
A new synthetic dual agonist of GPR120/GPR40 induces GLP-1 secretion and improves glucose homeostasis in mice
Bianchini, Gianluca, Nigro, Cecilia, Sirico, Anna, Novelli, Rubina, Prevenzano, Immacolata, Miele, Claudia, Beguinot, Francesco, Aramini, Andrea
Published in Biomedicine & pharmacotherapy (01.07.2021)
Published in Biomedicine & pharmacotherapy (01.07.2021)
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Journal Article
Paclitaxel binds and activates C5aR1: A new potential therapeutic target for the prevention of chemotherapy-induced peripheral neuropathy and hypersensitivity reactions
Brandolini, Laura, d'Angelo, Michele, Novelli, Rubina, Castelli, Vanessa, Giorgio, Cristina, Sirico, Anna, Cocchiaro, Pasquale, D'Egidio, Francesco, Benedetti, Elisabetta, Cristiano, Claudia, Bugatti, Antonella, Ruocco, Anna, Amendola, Pier Giorgio, Talarico, Carmine, Manelfi, Candida, Iaconis, Daniela, Beccari, Andrea, Quadros, Andreza U, Cunha, Thiago M, Caruso, Arnaldo, Russo, Roberto, Cimini, Annamaria, Aramini, Andrea, Allegretti, Marcello
Published in Cell death & disease (25.05.2022)
Published in Cell death & disease (25.05.2022)
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Journal Article
Branched-Chain Amino Acids and Di-Alanine Supplementation in Aged Mice: A Translational Study on Sarcopenia
Mantuano, Paola, Boccanegra, Brigida, Bianchini, Gianluca, Cappellari, Ornella, Tulimiero, Lisamaura, Conte, Elena, Cirmi, Santa, Sanarica, Francesca, De Bellis, Michela, Mele, Antonietta, Liantonio, Antonella, Allegretti, Marcello, Aramini, Andrea, De Luca, Annamaria
Published in Nutrients (09.01.2023)
Published in Nutrients (09.01.2023)
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Journal Article
Intranasal delivery of NGF rescues hearing impairment in aged SAMP8 mice
Castelli, Vanessa, d’Angelo, Michele, Zazzeroni, Francesca, Vecchiotti, Davide, Alesse, Edoardo, Capece, Daria, Brandolini, Laura, Cattani, Franca, Aramini, Andrea, Allegretti, Marcello, Cimini, Annamaria
Published in Cell death & disease (13.09.2023)
Published in Cell death & disease (13.09.2023)
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Journal Article
Intravitreal Administration of rhNGF Enhances Regenerative Processes in a Zebrafish Model of Retinal Degeneration
Cocchiaro, Pasquale, Di Donato, Vincenzo, Rubbini, Davide, Mastropasqua, Rodolfo, Allegretti, Marcello, Mantelli, Flavio, Aramini, Andrea, Brandolini, Laura
Published in Frontiers in pharmacology (07.03.2022)
Published in Frontiers in pharmacology (07.03.2022)
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Journal Article
Ketoprofen, lysine and gabapentin co-crystal magnifies synergistic efficacy and tolerability of the constituent drugs: Pre-clinical evidences towards an innovative therapeutic approach for neuroinflammatory pain
Aramini, Andrea, Bianchini, Gianluca, Lillini, Samuele, Tomassetti, Mara, Pacchiarotti, Niccolò, Canestrari, Daniele, Cocchiaro, Pasquale, Novelli, Rubina, Dragani, Maria Concetta, Palmerio, Ferdinando, Mattioli, Simone, Bordignon, Simone, d’Angelo, Michele, Castelli, Vanessa, d’Egidio, Francesco, Maione, Sabatino, Luongo, Livio, Boccella, Serena, Cimini, Annamaria, Brandolini, Laura, Chierotti, Michele Remo, Allegretti, Marcello
Published in Biomedicine & pharmacotherapy (01.07.2023)
Published in Biomedicine & pharmacotherapy (01.07.2023)
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Journal Article
Ketoprofen lysine salt has a better gastrointestinal and renal tolerability than ketoprofen acid: A comparative tolerability study in the Beagle dog
Novelli, Rubina, Aramini, Andrea, Boccella, Serena, Bagnasco, Michela, Cattani, Franca, Ferrari, Mauro Paolo, Goisis, Giovanni, Minnella, Enrico Maria, Allegretti, Marcello, Pace, Virgilio
Published in Biomedicine & pharmacotherapy (01.09.2022)
Published in Biomedicine & pharmacotherapy (01.09.2022)
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Journal Article
Inhibition of osteoclast activity by complement regulation with DF3016A, a novel small-molecular-weight C5aR inhibitor
D’Angelo, Rosa, Mangini, Maria, Fonderico, Jole, Fulle, Stefania, Mayo, Emilia, Aramini, Andrea, Mariggiò, Stefania
Published in Biomedicine & pharmacotherapy (01.03.2020)
Published in Biomedicine & pharmacotherapy (01.03.2020)
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Journal Article
Unexpected Salt/Cocrystal Polymorphism of the Ketoprofen–Lysine System: Discovery of a New Ketoprofen–l-Lysine Salt Polymorph with Different Physicochemical and Pharmacokinetic Properties
Aramini, Andrea, Bianchini, Gianluca, Lillini, Samuele, Bordignon, Simone, Tomassetti, Mara, Novelli, Rubina, Mattioli, Simone, Lvova, Larisa, Paolesse, Roberto, Chierotti, Michele Remo, Allegretti, Marcello
Published in Pharmaceuticals (Basel, Switzerland) (10.06.2021)
Published in Pharmaceuticals (Basel, Switzerland) (10.06.2021)
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Journal Article
Branched-chain amino acids and L-alanine supplementation ameliorate calcium dyshomeostasis in sarcopenia: New insights for nutritional interventions
Conte, Elena, Mantuano, Paola, Boccanegra, Brigida, Imbrici, Paola, Dinoi, Giorgia, Lenti, Roberta, Cappellari, Ornella, Cappetta, Donato, De Angelis, Antonella, Berrino, Liberato, Gordish-Dressman, Heather, Bianchini, Gianluca, Aramini, Andrea, Allegretti, Marcello, Liantonio, Antonella, De Luca, Annamaria
Published in Frontiers in pharmacology (19.06.2024)
Published in Frontiers in pharmacology (19.06.2024)
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Journal Article
Ergogenic Effect of BCAAs and L-Alanine Supplementation: Proof-of-Concept Study in a Murine Model of Physiological Exercise
Mantuano, Paola, Bianchini, Gianluca, Cappellari, Ornella, Boccanegra, Brigida, Conte, Elena, Sanarica, Francesca, Mele, Antonietta, Camerino, Giulia M, Brandolini, Laura, Allegretti, Marcello, De Bellis, Michela, Aramini, Andrea, De Luca, Annamaria
Published in Nutrients (30.07.2020)
Published in Nutrients (30.07.2020)
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Journal Article
Targeting the minor pocket of C5aR for the rational design of an oral allosteric inhibitor for inflammatory and neuropathic pain relief
Moriconi, Alessio, Cunha, Thiago M., Souza, Guilherme R., Lopes, Alexandre H., Cunha, Fernando Q., Carneiro, Victor L., Pinto, Larissa G., Brandolini, Laura, Aramini, Andrea, Bizzarri, Cinzia, Bianchini, Gianluca, Beccari, Andrea R., Fanton, Marco, Bruno, Agostino, Costantino, Gabriele, Bertini, Riccardo, Galliera, Emanuela, Locati, Massimo, Ferreira, Sérgio H., Teixeira, Mauro M., Allegretti, Marcello
Published in Proceedings of the National Academy of Sciences - PNAS (25.11.2014)
Published in Proceedings of the National Academy of Sciences - PNAS (25.11.2014)
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Journal Article
Inflammation-Independent Antinociceptive Effects of DF2755A, a CXCR1/2 Selective Inhibitor: A New Potential Therapeutic Treatment for Peripheral Neuropathy Associated to Non-Ulcerative Interstitial Cystitis/Bladder Pain Syndrome
Brandolini, Laura, Aramini, Andrea, Bianchini, Gianluca, Ruocco, Anna, Bertini, Riccardo, Novelli, Rubina, Angelico, Patrizia, Valsecchi, Anna Elisa, Russo, Roberto, Castelli, Vanessa, Cimini, Annamaria, Allegretti, Marcello
Published in Frontiers in pharmacology (28.04.2022)
Published in Frontiers in pharmacology (28.04.2022)
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Journal Article
Emerging Role of C5 Complement Pathway in Peripheral Neuropathies: Current Treatments and Future Perspectives
Giorgio, Cristina, Zippoli, Mara, Cocchiaro, Pasquale, Castelli, Vanessa, Varrassi, Giustino, Aramini, Andrea, Allegretti, Marcello, Brandolini, Laura, Cesta, Maria Candida
Published in Biomedicines (07.04.2021)
Published in Biomedicines (07.04.2021)
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Journal Article
Catalyst-Free Synthesis of Polysubstituted 5-Acylamino-1,3-Thiazoles via Hantzsch Cyclization of α-Chloroglycinates
Tomassetti, Mara, Lupidi, Gabriele, Piermattei, Pamela, Rossi, Federico V, Lillini, Samuele, Bianchini, Gianluca, Aramini, Andrea, Ciufolini, Marco A, Marcantoni, Enrico
Published in Molecules (Basel, Switzerland) (25.10.2019)
Published in Molecules (Basel, Switzerland) (25.10.2019)
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Journal Article
Combination Drug Therapy for the Management of Chronic Neuropathic Pain
Boccella, Serena, De Filippis, Lidia, Giorgio, Cristina, Brandolini, Laura, Jones, Meghan, Novelli, Rubina, Amorizzo, Ezio, Leoni, Matteo Luigi Giuseppe, Terranova, Gaetano, Maione, Sabatino, Luongo, Livio, Leone, Manuela, Allegretti, Marcello, Minnella, Enrico Maria, Aramini, Andrea
Published in Biomolecules (Basel, Switzerland) (01.12.2023)
Published in Biomolecules (Basel, Switzerland) (01.12.2023)
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Journal Article
The role of C5a-C5aR1 axis in bone pathophysiology: A mini-review
Ruocco, Anna, Sirico, Anna, Novelli, Rubina, Iannelli, Silvia, Van Breda, Shane Vontelin, Kyburz, Diego, Hasler, Paul, Aramini, Andrea, Amendola, Pier Giorgio
Published in Frontiers in cell and developmental biology (08.08.2022)
Published in Frontiers in cell and developmental biology (08.08.2022)
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Journal Article
1,3-Dibromo-1,1-difluoro-2-propanone as a Useful Synthon for a Chemoselective Preparation of 4‑Bromodifluoromethyl Thiazoles
Colella, Marco, Musci, Pantaleo, Carlucci, Claudia, Lillini, Samuele, Tomassetti, Mara, Aramini, Andrea, Degennaro, Leonardo, Luisi, Renzo
Published in ACS omega (30.11.2018)
Published in ACS omega (30.11.2018)
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