A Novel Single-Site Mutation in the Catalytic Domain of Protoporphyrinogen Oxidase IX (PPO) Confers Resistance to PPO-Inhibiting Herbicides
Rangani, Gulab, Salas-Perez, Reiofeli A, Aponte, Raphael A, Knapp, Michael, Craig, Ian R, Mietzner, Thomas, Langaro, Ana Claudia, Noguera, Matheus M, Porri, Aimone, Roma-Burgos, Nilda
Published in Frontiers in plant science (15.05.2019)
Published in Frontiers in plant science (15.05.2019)
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Journal Article
new amino acid substitution (Ala-205-Phe) in acetolactate synthase (ALS) confers broad spectrum resistance to ALS-inhibiting herbicides
Brosnan, James T, Vargas, Jose J, Breeden, Gregory K, Grier, Logan, Aponte, Raphael A, Tresch, Stefan, Laforest, Martin
Published in Planta (01.01.2016)
Published in Planta (01.01.2016)
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Antimalarial Inhibitors Targeting Serine Hydroxymethyltransferase (SHMT) with in Vivo Efficacy and Analysis of their Binding Mode Based on X‑ray Cocrystal Structures
Schwertz, Geoffrey, Witschel, Matthias C, Rottmann, Matthias, Bonnert, Roger, Leartsakulpanich, Ubolsree, Chitnumsub, Penchit, Jaruwat, Aritsara, Ittarat, Wanwipa, Schäfer, Anja, Aponte, Raphael A, Charman, Susan A, White, Karen L, Kundu, Abhijit, Sadhukhan, Surajit, Lloyd, Mel, Freiberg, Gail M, Srikumaran, Myron, Siggel, Marc, Zwyssig, Adrian, Chaiyen, Pimchai, Diederich, François
Published in Journal of medicinal chemistry (22.06.2017)
Published in Journal of medicinal chemistry (22.06.2017)
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Potent Inhibitors of Plasmodial Serine Hydroxymethyltransferase (SHMT) Featuring a Spirocyclic Scaffold
Schwertz, Geoffrey, Witschel, Matthias C., Rottmann, Matthias, Leartsakulpanich, Ubolsree, Chitnumsub, Penchit, Jaruwat, Aritsara, Amornwatcharapong, Watcharee, Ittarat, Wanwipa, Schäfer, Anja, Aponte, Raphael A., Trapp, Nils, Chaiyen, Pimchai, Diederich, François
Published in ChemMedChem (08.05.2018)
Published in ChemMedChem (08.05.2018)
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Conformational Aspects in the Design of Inhibitors for Serine Hydroxymethyltransferase (SHMT): Biphenyl, Aryl Sulfonamide, and Aryl Sulfone Motifs
Schwertz, Geoffrey, Frei, Michelle S., Witschel, Matthias C., Rottmann, Matthias, Leartsakulpanich, Ubolsree, Chitnumsub, Penchit, Jaruwat, Aritsara, Ittarat, Wanwipa, Schäfer, Anja, Aponte, Raphael A., Trapp, Nils, Mark, Kerstin, Chaiyen, Pimchai, Diederich, François
Published in Chemistry : a European journal (12.10.2017)
Published in Chemistry : a European journal (12.10.2017)
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Fine Tuning of a Biological Machine: DnaK Gains Improved Chaperone Activity by Altered Allosteric Communication and Substrate Binding
Schweizer, Regina S., Aponte, Raphael A., Zimmermann, Sabine, Weber, Annika, Reinstein, Jochen
Published in Chembiochem : a European journal of chemical biology (04.07.2011)
Published in Chembiochem : a European journal of chemical biology (04.07.2011)
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Inhibition profile of trifludimoxazin towards PPO2 target site mutations
Porri, Aimone, Betz, Michael, Seebruck, Kathryn, Knapp, Michael, Johnen, Philipp, Witschel, Matthias, Aponte, Raphael, Liebl, Rex, Tranel, Patrick J., Lerchl, Jens
Published in Pest management science (01.02.2023)
Published in Pest management science (01.02.2023)
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Discovery, Mode of Action, Resistance Mechanisms, and Plan of Action for Sustainable Use of Group 14 Herbicides
Barker, Abigail L., Pawlak, John, Duke, Stephen O., Beffa, Roland, Tranel, Patrick J., Wuerffel, Joe, Young, Bryan, Porri, Aimone, Liebl, Rex, Aponte, Raphael, Findley, Douglas, Betz, Michael, Lerchl, Jens, Culpepper, Stanley, Bradley, Kevin, Dayan, Franck E.
Published in Weed science (01.05.2023)
Published in Weed science (01.05.2023)
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Acetohydroxyacid synthase (AHAS) amino acid substitution Asp376Glu in Lolium perenne: effect on herbicide efficacy and plant growth
Menegat, Alexander, Bailly, Geraldine C., Aponte, Raphael, Heinrich, Gregor M. T., Sievernich, Bernd, Gerhards, Roland
Published in Journal of plant diseases and protection (2006) (01.08.2016)
Published in Journal of plant diseases and protection (2006) (01.08.2016)
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제초성 우라실피리드
NEWTON TREVOR WILLIAM, APONTE RAPHAEL, LANDES ANDREAS, JOHANNES MANUEL, EVANS RICHARD R, MASSA DARIO, MIETZNER THOMAS, WITSCHEL MATTHIAS, SEITZ THOMAS, SEISER TOBIAS, PARRA RAPADO LILIANA
Year of Publication 25.01.2019
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Year of Publication 25.01.2019
Patent
PLANTS HAVING INCREASED TOLERANCE TO HERBICIDES
LERCHL JENS, PAULIK JILL MARIE, APONTE RAPHAEL, TRESCH STEFAN, BROMMER CHAD, MASSA DARIO, WITSCHEL MATTHIAS, SEISER TOBIAS
Year of Publication 05.03.2015
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Year of Publication 05.03.2015
Patent
PLANTS HAVING INCREASED TOLERANCE TO HERBICIDES
LERCHL JENS, APONTE RAPHAEL, MIETZNER THOMAS, TRESCH STEFAN, HUTZLER JOHANNES, WITSCHEL MATTHIAS, MANKIN S. LUKE, SIMON ANJA
Year of Publication 18.03.2014
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Year of Publication 18.03.2014
Patent
SUBSTITUTED 1,2,5-OXADIAZOLE COMPOUNDS AND THEIR USE AS HERBICIDES
NEWTON TREVOR WILLIAM, LERCHL JENS, APONTE RAPHAEL, EVANS RICHARD R, KRAUS HELMUT, WITSCHEL MATTHIAS, SEITZ THOMAS, KREUZ KLAUS, GROSSMANN KLAUS, PARRA RAPADO LILIANA
Year of Publication 07.08.2014
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Year of Publication 07.08.2014
Patent