AB‐Bind: Antibody binding mutational database for computational affinity predictions
Sirin, Sarah, Apgar, James R., Bennett, Eric M., Keating, Amy E.
Published in Protein science (01.02.2016)
Published in Protein science (01.02.2016)
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Journal Article
Modeling and mitigation of high-concentration antibody viscosity through structure-based computer-aided protein design
Apgar, James R, Tam, Amy S P, Sorm, Rhady, Moesta, Sybille, King, Amy C, Yang, Han, Kelleher, Kerry, Murphy, Denise, D'Antona, Aaron M, Yan, Guoying, Zhong, Xiaotian, Rodriguez, Linette, Ma, Weijun, Ferguson, Darren E, Carven, Gregory J, Bennett, Eric M, Lin, Laura
Published in PloS one (07.05.2020)
Published in PloS one (07.05.2020)
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Journal Article
Ibrexafungerp: An orally active β-1,3-glucan synthesis inhibitor
Apgar, James M., Wilkening, Robert R., Parker, Dann L., Meng, Dongfang, Wildonger, Kenneth J., Sperbeck, Donald, Greenlee, Mark L., Balkovec, James M., Flattery, Amy M., Abruzzo, George K., Galgoci, Andrew M., Giacobbe, Robert A., Gill, Charles J., Hsu, Ming-Jo, Liberator, Paul, Misura, Andrew S., Motyl, Mary, Nielsen Kahn, Jennifer, Powles, Maryann, Racine, Fred, Dragovic, Jasminka, Fan, Weiming, Kirwan, Robin, Lee, Shu, Liu, Hao, Mamai, Ahmed, Nelson, Kingsley, Peel, Michael
Published in Bioorganic & medicinal chemistry letters (15.01.2021)
Published in Bioorganic & medicinal chemistry letters (15.01.2021)
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Journal Article
Establishing in vitro in vivo correlations to screen monoclonal antibodies for physicochemical properties related to favorable human pharmacokinetics
Avery, Lindsay B, Wade, Jason, Wang, Mengmeng, Tam, Amy, King, Amy, Piche-Nicholas, Nicole, Kavosi, Mania S, Penn, Steve, Cirelli, David, Kurz, Jeffrey C, Zhang, Minlei, Cunningham, Orla, Jones, Rhys, Fennell, Brian J, McDonnell, Barry, Sakorafas, Paul, Apgar, James, Finlay, William J, Lin, Laura, Bloom, Laird, O'Hara, Denise M
Published in mAbs (17.02.2018)
Published in mAbs (17.02.2018)
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Journal Article
Structure-function relationships of the soluble form of the antiaging protein Klotho have therapeutic implications for managing kidney disease
Zhong, Xiaotian, Jagarlapudi, Srinath, Weng, Yan, Ly, Mellisa, Rouse, Jason C., McClure, Kim, Ishino, Tetsuya, Zhang, Yan, Sousa, Eric, Cohen, Justin, Tzvetkova, Boriana, Cote, Kaffa, Scarcelli, John J., Johnson, Keith, Palandra, Joe, Apgar, James R., Yaddanapudi, Suma, Gonzalez-Villalobos, Romer A., Opsahl, Alan C., Lam, Khetemenee, Yao, Qing, Duan, Weili, Sievers, Annette, Zhou, Jing, Ferguson, Darren, D'Antona, Aaron, Zollner, Richard, Zhu, Hongli L., Kriz, Ron, Lin, Laura, Clerin, Valerie
Published in The Journal of biological chemistry (06.03.2020)
Published in The Journal of biological chemistry (06.03.2020)
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Journal Article
Combining random mutagenesis, structure-guided design and next-generation sequencing to mitigate polyreactivity of an anti-IL-21R antibody
Campbell, Sharon M, DeBartolo, Joseph, Apgar, James R, Mosyak, Lydia, McManus, Virginie, Beyer, Sonia, Bennett, Eric M, Lambert, Matthew, Cunningham, Orla
Published in mAbs (01.01.2021)
Published in mAbs (01.01.2021)
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Journal Article
Beyond CDR-grafting: Structure-guided humanization of framework and CDR regions of an anti-myostatin antibody
Apgar, James R, Mader, Michelle, Agostinelli, Rita, Benard, Susan, Bialek, Peter, Johnson, Mark, Gao, Yijie, Krebs, Mark, Owens, Jane, Parris, Kevin, St Andre, Michael, Svenson, Kris, Morris, Carl, Tchistiakova, Lioudmila
Published in mAbs (02.10.2016)
Published in mAbs (02.10.2016)
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Journal Article
Modeling Backbone Flexibility to Achieve Sequence Diversity: The Design of Novel α-Helical Ligands for Bcl-xL
Fu, Xiaoran, Apgar, James R., Keating, Amy E.
Published in Journal of molecular biology (24.08.2007)
Published in Journal of molecular biology (24.08.2007)
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Journal Article
Augmented Binary Substitution: Single-pass CDR germ-lining and stabilization of therapeutic antibodies
Townsend, Sue, Fennell, Brian J., Apgar, James R., Lambert, Matthew, McDonnell, Barry, Grant, Joanne, Wade, Jason, Franklin, Edward, Foy, Niall, Shúilleabháin, Deirdre Ní, Fields, Conor, Darmanin-Sheehan, Alfredo, King, Amy, Paulsen, Janet E., Hickling, Timothy P., Tchistiakova, Lioudmila, Cunningham, Orla, Finlay, William J. J.
Published in Proceedings of the National Academy of Sciences - PNAS (15.12.2015)
Published in Proceedings of the National Academy of Sciences - PNAS (15.12.2015)
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Journal Article
MK-5204: An orally active β-1,3-glucan synthesis inhibitor
Apgar, James M., Wilkening, Robert R., Parker, Dann L., Meng, Dongfang, Wildonger, Kenneth J., Sperbeck, Donald, Greenlee, Mark L., Balkovec, James M., Flattery, Amy M., Abruzzo, George K., Galgoci, Andrew M., Giacobbe, Robert A., Gill, Charles J., Hsu, Ming-Jo, Liberator, Paul, Misura, Andrew S., Motyl, Mary, Kahn, Jennifer Nielsen, Powles, Maryann, Racine, Fred, Dragovic, Jasminka, Fan, Weiming, Kirwan, Robin, Lee, Shu, Liu, Hao, Mamai, Ahmed, Nelson, Kingsley, Peel, Michael
Published in Bioorganic & medicinal chemistry letters (01.09.2020)
Published in Bioorganic & medicinal chemistry letters (01.09.2020)
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Journal Article
Novel orally active inhibitors of β-1,3-glucan synthesis derived from enfumafungin
Apgar, James M., Wilkening, Robert R., Greenlee, Mark L., Balkovec, James M., Flattery, Amy M., Abruzzo, George K., Galgoci, Andrew M., Giacobbe, Robert A., Gill, Charles J., Hsu, Ming Jo, Liberator, Paul, Misura, Andrew S., Motyl, Mary, Nielsen Kahn, Jennifer, Powles, Maryann, Racine, Fred, Dragovic, Jasminka, Habulihaz, Bahanu, Fan, Weiming, Kirwan, Robin, Lee, Shu, Liu, Hao, Mamai, Ahmed, Nelson, Kingsley, Peel, Michael
Published in Bioorganic & medicinal chemistry letters (15.12.2015)
Published in Bioorganic & medicinal chemistry letters (15.12.2015)
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Journal Article
Structure–activity-relationship of amide and sulfonamide analogs of omarigliptin
Chen, Ping, Feng, Dennis, Qian, Xiaoxia, Apgar, James, Wilkening, Robert, Kuethe, Jeffrey T., Gao, Ying-Duo, Scapin, Giovanna, Cox, Jason, Doss, George, Eiermann, George, He, Huaibing, Li, Xiaohua, Lyons, Kathryn A., Metzger, Joseph, Petrov, Aleksandr, Wu, Joseph K., Xu, Shiyao, Weber, Ann E., Yan, Youwei, Roy, Ranabir Sinha, Biftu, Tesfaye
Published in Bioorganic & medicinal chemistry letters (15.12.2015)
Published in Bioorganic & medicinal chemistry letters (15.12.2015)
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Journal Article
Predicting helix orientation for coiled-coil dimers
Apgar, James R., Gutwin, Karl N., Keating, Amy E.
Published in Proteins, structure, function, and bioinformatics (15.08.2008)
Published in Proteins, structure, function, and bioinformatics (15.08.2008)
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Journal Article
Cluster expansion models for flexible-backbone protein energetics
Apgar, James R, Hahn, Seungsoo, Grigoryan, Gevorg, Keating, Amy E
Published in Journal of computational chemistry (30.11.2009)
Published in Journal of computational chemistry (30.11.2009)
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Journal Article
A predictive model of intein insertion site for use in the engineering of molecular switches
Apgar, James, Ross, Mary, Zuo, Xiao, Dohle, Sarah, Sturtevant, Derek, Shen, Binzhang, de la Vega, Humberto, Lessard, Philip, Lazar, Gabor, Raab, R Michael
Published in PloS one (23.05.2012)
Published in PloS one (23.05.2012)
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Journal Article
Pharmacological AMPK activation induces transcriptional responses congruent to exercise in skeletal and cardiac muscle, adipose tissues and liver
Muise, Eric S, Guan, Hong-Ping, Liu, Jinqi, Nawrocki, Andrea R, Yang, Xiaodong, Wang, Chuanlin, Rodríguez, Carlos G, Zhou, Dan, Gorski, Judith N, Kurtz, Marc M, Feng, Danqing, Leavitt, Kenneth J, Wei, Lan, Wilkening, Robert R, Apgar, James M, Xu, Shiyao, Lu, Ku, Feng, Wen, Li, Ying, He, Huaibing, Previs, Stephen F, Shen, Xiaolan, van Heek, Margaret, Souza, Sandra C, Rosenbach, Mark J, Biftu, Tesfaye, Erion, Mark D, Kelley, David E, Kemp, Daniel M, Myers, Robert W, Sebhat, Iyassu K
Published in PloS one (27.02.2019)
Published in PloS one (27.02.2019)
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Journal Article
THERAPEUTIC ANTIBODIES AND THEIR USES
NOCULA LUGOWSKA MALGORZATA AGNIESZKA, HOOPER ANDREA THERESE, WU LEI, APGAR JAMES REASONER
Year of Publication 17.07.2023
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Year of Publication 17.07.2023
Patent
Engineering a thermoregulated intein-modified xylanase into maize for consolidated lignocellulosic biomass processing
BINZHANG SHEN, XUEGUANG SUN, LUCERO, Hector, GRAY, Benjamin, EKBORG, Nathan A, DONGCHENG ZHANG, SCHLEY JOHNSON, Jeremy C, LAZAR, Gabor, RAAB, R. Michael, XIAO ZUO, SHILLING, Taran, APGAR, James, ROSS, Mary, BOUGRI, Oleg, SAMOYLOV, Vladimir, PARKER, Matthew, HANCOCK, Elaina
Published in Nature biotechnology (01.11.2012)
Published in Nature biotechnology (01.11.2012)
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Journal Article
치료 항체 및 그의 용도
NOCULA LUGOWSKA MALGORZATA AGNIESZKA, HOOPER ANDREA THERESE, WU LEI, APGAR JAMES REASONER
Year of Publication 14.02.2023
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Year of Publication 14.02.2023
Patent