Pd-Catalyzed Cross-Coupling Reactions Promoted by Biaryl Phosphorinane Ligands
Laffoon, Summer D, Chan, Vincent S, Fickes, Michael G, Kotecki, Brian, Ickes, Andrew R, Henle, Jeremy, Napolitano, José G, Franczyk, Thaddeus S, Dunn, Travis B, Barnes, David M, Haight, Anthony R, Henry, Rodger F, Shekhar, Shashank
Published in ACS catalysis (06.12.2019)
Published in ACS catalysis (06.12.2019)
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Journal Article
A General Method for the Synthesis of Unsymmetrically Substituted Ureas via Palladium-Catalyzed Amidation
Kotecki, Brian J, Fernando, Dilinie P, Haight, Anthony R, Lukin, Kirill A
Published in Organic letters (19.02.2009)
Published in Organic letters (19.02.2009)
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Journal Article
General Method for the Palladium-Catalyzed Allylation of Aliphatic Alcohols
Haight, Anthony R, Stoner, Eric J, Peterson, Matthew J, Grover, Vandana K
Published in Journal of organic chemistry (17.10.2003)
Published in Journal of organic chemistry (17.10.2003)
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Journal Article
Discovery and Development of Metal-Catalyzed Coupling Reactions in the Synthesis of Dasabuvir, an HCV-Polymerase Inhibitor
Barnes, David M, Shekhar, Shashank, Dunn, Travis B, Barkalow, Jufang H, Chan, Vincent S, Franczyk, Thaddeus S, Haight, Anthony R, Hengeveld, John E, Kolaczkowski, Lawrence, Kotecki, Brian J, Liang, Guangxin, Marek, James C, McLaughlin, Maureen A, Montavon, Donna K, Napier, James J
Published in Journal of organic chemistry (19.04.2019)
Published in Journal of organic chemistry (19.04.2019)
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Journal Article
Synthesis of the Quinolone ABT-492: Crystallizations for Optimal Processing
Haight, Anthony R, Ariman, Sema Z, Barnes, David M, Benz, Nancy J, Gueffier, Francoix X, Henry, Rodger F, Hsu, Margaret C, Lee, Elaine C, Morin, Larry, Pearl, Kurt B, Peterson, Matthew J, Plata, Daniel J, Willcox, David R
Published in Organic process research & development (21.07.2006)
Published in Organic process research & development (21.07.2006)
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Journal Article
Internal coordination at tin promotes selective alkyl transfer in the Stille coupling reaction
Vedejs, Edwin, Haight, Anthony R, Moss, William O
Published in Journal of the American Chemical Society (01.07.1992)
Published in Journal of the American Chemical Society (01.07.1992)
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Journal Article
The Discovery and Development of a Safe, Practical Synthesis of ABT-869
Kruger, Albert W, Rozema, Michael J, Chu-Kung, Alexander, Gandarilla, Jorge, Haight, Anthony R, Kotecki, Brian J, Richter, Steven M, Schwartz, Albert M, Wang, Zhe
Published in Organic process research & development (20.11.2009)
Published in Organic process research & development (20.11.2009)
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Journal Article
Process Development for ABT-472, a Benzimidazole PARP Inhibitor
Barkalow, Jufang H, Breting, Jeffrey, Gaede, Bruce J, Haight, Anthony R, Henry, Rodger, Kotecki, Brian, Mei, Jianzhang, Pearl, Kurt B, Tedrow, Jason S, Viswanath, Shekhar K
Published in Organic process research & development (01.07.2007)
Published in Organic process research & development (01.07.2007)
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Journal Article
Impact of Entropic Effects in the Classical Resolution of a 2-Arylpyrrolidine
Barnes, David M, Barkalow, Jufang, Chen, Yong, Gupta, Ashok, Haight, Anthony R, Hengeveld, John E, Kerdesky, Francis A. J, Kotecki, Brian J, Macri, Bryan, Pal, Agnes
Published in Organic process research & development (20.03.2009)
Published in Organic process research & development (20.03.2009)
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Journal Article
A Scaleable Synthesis of Fiduxosin
Haight, Anthony R, Bailey, Anne E, Baker, William S, Cain, Michael H, Copp, Richard R, DeMattei, John A, Ford, Kelley L, Henry, Rodger F, Hsu, Margaret C, Keyes, Robert F, King, Steven A, McLaughlin, Maureen A, Melcher, Laura M, Nadler, William R, Oliver, Patricia A, Parekh, Shyamal I, Patel, Hemant H, Seif, Louis S, Staeger, Mike A, Wayne, Gregory S, Wittenberger, Steven J, Zhang, Weijiang
Published in Organic process research & development (01.11.2004)
Published in Organic process research & development (01.11.2004)
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Journal Article
Chlorination at the 8-Position of a Functionalized Quinolone and the Synthesis of Quinolone Antibiotic ABT-492
Barnes, David M, Christesen, Alan C, Engstrom, Kenneth M, Haight, Anthony R, Hsu, Margaret C, Lee, Elaine C, Peterson, Matthew J, Plata, Daniel J, Raje, Prasad S, Stoner, Eric J, Tedrow, Jason S, Wagaw, Seble
Published in Organic process research & development (21.07.2006)
Published in Organic process research & development (21.07.2006)
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Journal Article
Synthesis of Erythromycin Derivatives via the Olefin Cross-Metathesis Reaction
Hsu, Margaret C, Junia, Adam J, Haight, Anthony R, Zhang, Weijiang
Published in Journal of organic chemistry (28.05.2004)
Published in Journal of organic chemistry (28.05.2004)
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Journal Article
Reduction of an Enaminone: Synthesis of the Diamino Alcohol Core of Ritonavir
Haight, Anthony R, Stuk, Timothy L, Allen, Michael S, Bhagavatula, Lakshmi, Fitzgerald, Michael, Hannick, Steven M, Kerdesky, Francis A. J, Menzia, Jerome A, Parekh, Shyamal I, Robbins, Timothy A, Scarpetti, David, Tien, Jien-Heh J
Published in Organic process research & development (01.03.1999)
Published in Organic process research & development (01.03.1999)
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Journal Article
New conditions for the synthesis of thiophenes via the Knoevenagel/Gewald reaction sequence. Application to the synthesis of a multitargeted kinase inhibitor
Barnes, David M., Haight, Anthony R., Hameury, Thomas, McLaughlin, Maureen A., Mei, Jianzhang, Tedrow, Jason S., Riva Toma, Joan Dalla
Published in Tetrahedron (04.12.2006)
Published in Tetrahedron (04.12.2006)
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Journal Article
Diastereoselectivity in the osmium-catalyzed dihydroxylation of allylic amides and carbamates
Krysan, Damian J., Rockway, Todd W., Haight, Anthony R.
Published in Tetrahedron: asymmetry (01.04.1994)
Published in Tetrahedron: asymmetry (01.04.1994)
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Journal Article
An Efficient Stereocontrolled Strategy for the Synthesis of Hydroxyethylene Dipeptide Isosteres
Stuk, Timothy L, Haight, Anthony R, Scarpetti, David, Allen, Michael S, Menzia, Jerome A, Robbins, Timothy A, Parekh, Shyamal I, Langridge, Denton C, Tien, Jien-Heh J
Published in Journal of organic chemistry (01.07.1994)
Published in Journal of organic chemistry (01.07.1994)
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Journal Article
Characterization and Synthesis of a 6-Substituted Benzo[b]thiophene
Haight, Anthony R, Wayne, Gregory S, Lannoye, Gregory S, Parekh, Shyamal I, Zhang, Weijiang, Copp, Richard R, Hollis, L. Steven
Published in Journal of organic chemistry (21.08.1998)
Published in Journal of organic chemistry (21.08.1998)
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Journal Article
Synthesis of a 5-substituted benzo[b]thiophene
Wayne, GS, Lannoye, GS, Haight, AR, Parekh, SI, Zhang, WJ, Copp, RR
Published in Heterocycles (01.05.2000)
Published in Heterocycles (01.05.2000)
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