1-(2-Aminoethyl)-3-(arylsulfonyl)-1H-pyrrolopyridines are 5-HT6 receptor ligands
Bernotas, Ronald C., Antane, Schuyler A., Lenicek, Steven E., Haydar, Simon N., Robichaud, Albert J., Harrison, Boyd L., Zhang, Guo Ming, Smith, Deborah, Coupet, Joseph, Schechter, Lee E.
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
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Journal Article
Synthesis and potassium channel opening activity of substituted 10H-benzo[4,5]furo[3,2-b]indole- and 5,10-dihydro-indeno[1,2-b]indole-1-carboxylic acids
BUTERA, John A, ANTANE, Schuyler A, HIRTH, Bradford, LENNOX, Joseph R, SHELDON, Jeffrey H, NORTON, N. Wesley, WARGA, Dawn, ARGENTIERI, Thomas M
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
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Journal Article
Comparison of the Potassium Channel Openers, WAY-133537, ZD6169, and Celikalim on Isolated Bladder Tissue and In Vivo Bladder Instability in Rat
Wojdan, A, Freeden, C, Woods, M, Oshiro, G, Spinelli, W, Colatsky, T J, Sheldon, J H, Norton, N W, Warga, D, Antane, M M, Antane, S A, Butera, J A, Argentieri, T M
Published in The Journal of pharmacology and experimental therapeutics (01.06.1999)
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Published in The Journal of pharmacology and experimental therapeutics (01.06.1999)
Journal Article
Design and SAR of Novel Potassium Channel Openers Targeted for Urge Urinary Incontinence. 1. N-Cyanoguanidine Bioisosteres Possessing in Vivo Bladder Selectivity
Butera, John A, Antane, Madelene M, Antane, Schuyler A, Argentieri, Thomas M, Freeden, Chris, Graceffa, Russell F, Hirth, Bradford H, Jenkins, Douglas, Lennox, Joseph R, Matelan, Edward, Norton, N. Wesley, Quagliato, Dominick, Sheldon, Jeffrey H, Spinelli, Walter, Warga, Dawn, Wojdan, Alexandra, Woods, Morgan
Published in Journal of medicinal chemistry (23.03.2000)
Published in Journal of medicinal chemistry (23.03.2000)
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Journal Article
Synthesis and potassium channel opening activity of substituted 10H-Benzofuro[3,2-b]indole- and 5,10-Dihydro-indeno[1,2-b]indole-1-carboxylic acids
Butera, John A., Antane, Schuyler A., Hirth, Bradford, Lennox, Joseph R., Sheldon, Jeffrey H., Norton, N.Wesley, Warga, Dawn, Argentieri, Thomas M.
Published in Bioorganic & medicinal chemistry letters (01.08.2001)
Published in Bioorganic & medicinal chemistry letters (01.08.2001)
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Journal Article
1-(2-Aminoethyl)-3-(arylsulfonyl)-1H-pyrrolopyridines are 5-HT sub(6) receptor ligands
Bernotas, Ronald C, Antane, Schuyler A, Lenicek, Steven E, Haydar, Simon N, Robichaud, Albert J, Harrison, Boyd L, Zhang, Guo Ming, Smith, Deborah, Coupet, Joseph, Schechter, Lee E
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
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Journal Article
1-(2-Aminoethyl)-3-(arylsulfonyl)-1H-pyrrolopyridines are 5-HT(6) receptor ligands
Bernotas, Ronald C, Antane, Schuyler A, Lenicek, Steven E, Haydar, Simon N, Robichaud, Albert J, Harrison, Boyd L, Zhang, Guo Ming, Smith, Deborah, Coupet, Joseph, Schechter, Lee E
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
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Journal Article
Synthesis and potassium channel opening activity of substituted 10 H-Benzo [4,5]furo[3,2- b]indole- and 5,10-Dihydro-indeno[1,2- b]indole-1-carboxylic acids
Butera, John A., Antane, Schuyler A., Hirth, Bradford, Lennox, Joseph R., Sheldon, Jeffrey H., Norton, N.Wesley, Warga, Dawn, Argentieri, Thomas M.
Published in Bioorganic & medicinal chemistry letters (2001)
Published in Bioorganic & medicinal chemistry letters (2001)
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Journal Article
1-(Aminoalkyl)-3-sulfonylazaindoler som 5-hydroxytryptamin-6-ligander
ANTANE, SCHUYLER, A, BERNOTAS, RONALD, CHARLES, LENICEK, STEVEN, EDWARD
Year of Publication 16.04.2007
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Year of Publication 16.04.2007
Patent
1-(AMINOALKYL)-3-SULFONYLAZAINDOLES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS
ANTANE, SCHUYLER, A, BERNOTAS, RONALD, CHARLES, LENICEK, STEVEN, EDWARD
Year of Publication 28.02.2007
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Year of Publication 28.02.2007
Patent
1-(AMINOALKYL)-3-SULFONYLAZAINDOLE ALS 5- HYDROXYTRYPTAMIN-6 LIGANDEN
ANTANE, SCHUYLER, A, BERNOTAS, RONALD, CHARLES, LENICEK, STEVEN, EDWARD
Year of Publication 15.03.2006
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Year of Publication 15.03.2006
Patent