Design of Novel Exendin-Based Dual Glucagon-like Peptide 1 (GLP-1)/Glucagon Receptor Agonists
Evers, Andreas, Haack, Torsten, Lorenz, Martin, Bossart, Martin, Elvert, Ralf, Henkel, Bernd, Stengelin, Siegfried, Kurz, Michael, Glien, Maike, Dudda, Angela, Lorenz, Katrin, Kadereit, Dieter, Wagner, Michael
Published in Journal of medicinal chemistry (25.05.2017)
Published in Journal of medicinal chemistry (25.05.2017)
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Running on mixed fuel‐dual agonistic approach of GLP‐1 and GCG receptors leads to beneficial impact on body weight and blood glucose control: A comparative study between mice and non‐human primates
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Published in Diabetes, obesity & metabolism (01.08.2018)
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Team Players or Opponents: Coadministration of Selective Glucagon and GLP-1 Receptor Agonists in Obese Diabetic Monkeys
Elvert, Ralf, Bossart, Martin, Herling, Andreas W, Weiss, Tilo, Zhang, Baohong, Kannt, Aimo, Wagner, Michael, Haack, Torsten, Evers, Andreas, Dudda, Angela, Keil, Stefanie, Lorenz, Martin, Lorenz, Katrin, Riz, Michela, Hennerici, Wolfgang, Larsen, Philip J
Published in Endocrinology (Philadelphia) (01.08.2018)
Published in Endocrinology (Philadelphia) (01.08.2018)
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Lipid oxidation products in ischemic porcine heart tissue
Dudda, Angela, Spiteller, Gerhard, Kobelt, Frank
Published in Chemistry and physics of lipids (30.07.1996)
Published in Chemistry and physics of lipids (30.07.1996)
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Weight Loss Outcomes with Species-Specific Dual GLP-1R/GCGR Agonists in Animal Models
ELVERT, RALF, BOSSART, MARTIN, ZHANG, BOB, KANNT, AIMO, WAGNER, MICHAEL, HAACK, TORSTEN, EVERS, ANDREAS, DUDDA, ANGELA, LORENZ, MARTIN, KEIL, STEFANIE, LARSEN, PHILIP J.
Published in Diabetes (New York, N.Y.) (01.07.2018)
Published in Diabetes (New York, N.Y.) (01.07.2018)
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Mechanistic investigations of the liver toxicity of the free fatty acid receptor 1 agonist fasiglifam (TAK875) and its primary metabolites
Ackerson, Timothy, Amberg, Alexander, Atzrodt, Jens, Arabeyre, Catherine, Defossa, Elisabeth, Dorau, Martina, Dudda, Angela, Dwyer, Jacquelyn, Holla, Wolfgang, Kissner, Thomas, Kohlmann, Markus, Kürzel, Ulrich, Pánczél, József, Rajanna, Shibani, Riedel, Jens, Schmidt, Friedemann, Wäse, Kerstin, Weitz, Dietmar, Derdau, Volker
Published in Journal of biochemical and molecular toxicology (01.08.2019)
Published in Journal of biochemical and molecular toxicology (01.08.2019)
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Correction to Design of Novel Exendin-Based Dual Glucagon-like Peptide 1 (GLP-1)/Glucagon Receptor Agonist
Evers, Andreas, Haack, Torsten, Lorenz, Martin, Bossart, Martin, Elvert, Ralf, Henkel, Bernd, Stengelin, Siegfried, Kurz, Michael, Glien, Maike, Dudda, Angela, Lorenz, Katrin, Kadereit, Dieter, Wagner, Michael
Published in Journal of medicinal chemistry (13.07.2017)
Published in Journal of medicinal chemistry (13.07.2017)
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Modulation of Hexadecyl-LPA-Mediated Activation of Mast Cells and Microglia by a Chemical Probe for LPA5
Kozian, Detlef H., von Haeften, Elisabeth, Joho, Sabrina, Czechtizky, Werngard, Anumala, Upendra R., Roux, Pascale, Dudda, Angela, Evers, Andreas, Nazare, Marc
Published in Chembiochem : a European journal of chemical biology (03.05.2016)
Published in Chembiochem : a European journal of chemical biology (03.05.2016)
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Selective inhibition of 12-lipoxygenase protects islets and beta cells from inflammatory cytokine-mediated beta cell dysfunction
Taylor-Fishwick, David A., Weaver, Jessica, Glenn, Lindsey, Kuhn, Norine, Rai, Ganesha, Jadhav, Ajit, Simeonov, Anton, Dudda, Angela, Schmoll, Dieter, Holman, Theodore R., Maloney, David J., Nadler, Jerry L.
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Published in Diabetologia (01.03.2015)
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Cover Image, Volume 20, Issue 8
Elvert, Ralf, Herling, Andreas W., Bossart, Martin, Weiss, Tilo, Zhang, Baohong, Wenski, Pierre, Wandschneider, Jörn, Kleutsch, Sabrina, Butty, Uwe, Kannt, Aimo, Wagner, Michael, Haack, Torsten, Evers, Andreas, Dudda, Angela, Lorenz, Martin, Keil, Stefanie, Larsen, Philip J.
Published in Diabetes, obesity & metabolism (01.08.2018)
Published in Diabetes, obesity & metabolism (01.08.2018)
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Factor Xa inhibitors based on a 2-carboxyindole scaffold: SAR of neutral P1 substituents
Nazaré, Marc, Essrich, Melanie, Will, David W, Matter, Hans, Ritter, Kurt, Urmann, Matthias, Bauer, Armin, Schreuder, Herman, Dudda, Angela, Czech, Jörg, Lorenz, Martin, Laux, Volker, Wehner, Volkmar
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
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Novel factor Xa inhibitors based on a benzoic acid scaffold and incorporating a neutral P1 ligand
Nazaré, Marc, Matter, Hans, Klingler, Otmar, Al-Obeidi, Fahad, Schreuder, Herman, Zoller, Gerhard, Czech, Jörg, Lorenz, Martin, Dudda, Angela, Peyman, Anusch, Nestler, Hans Peter, Urmann, Matthias, Bauer, Armin, Laux, Volker, Wehner, Volkmar, Will, David W.
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
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SUBSTITUTED 6-(4-HYDROXY-PHENYL)-1H-PYRAZOLO[3,4-B]PYRIDINE DERIVATIVES AS KINASE INHIBITORS
KANNT, AIMO, LOEHN, MATTHIAS, PFEIFFER-MAREK, STEFANIA, HACHTEL, STEPHANIE, SCHOENAU, CHRISTIAN, PLETTENBURG, OLIVER, DEDIO, JUERGEN, GAUL, HOLGER, SCHIFFER, ALEXANDER, DUDDA, ANGELA
Year of Publication 15.06.2016
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Year of Publication 15.06.2016
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Naphthyl Sulfonamide Pyrrolidine Derivatives as KEAP-1 Modulators for the Treatment of Diabetes, Obesity, Dyslipidemia and Related Disorders
CHRISTOPHER KALLUS, STEFAN GUESSREGEN, BETTINA ELSHORST, HAUKE SZILL, AIRNO KANNT, KARLRISTIAN ENGEL, PETER MONECKE, HEINER GLOMBIK, DIETER SCHMOLL, ANGELA DUDDA, SVEN RUF
Year of Publication 23.03.2016
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Year of Publication 23.03.2016
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Naphthyl sulfonamide derivatives as KEAP-1 modulators for the treatment of diabetes, obesity, dyslipidemia and related disorders
CHRISTOPHER KALLUS, BETTINA ELSHORST, AIMO KANNT, KARLRISTIAN ENGEL, PETER MONECKE, HEINER GLOMBIK, HAUKE SZILLAT, ANGELA DUDDA, SVEN RUF, STEFAN GUOSSREGEN, DIETER SCHMOL
Year of Publication 23.03.2016
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Year of Publication 23.03.2016
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Substituted 6-(4-hydroxy-phenyl)-1H-pyrazolo[3,4-b]pyridine derivatives as kinase inhibitors
PFEIFFER-MAREK STEFANIA, KANNT AIMO, GAUL HOLGER, DEDIO JUERGEN, HACHTEL STEPHANIE, LOEHN MATTHIAS, PLETTENBURG OLIVER, DUDDA ANGELA, SCHOENAU CHRISTIAN, SCHIFFER ALEXANDER
Year of Publication 15.09.2015
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Year of Publication 15.09.2015
Patent