Synthesis of the Azaphilones (+)-Sclerotiorin and (+)-8-O-Methylsclerotiorinamine Utilizing (+)-Sparteine Surrogates in Copper-Mediated Oxidative Dearomatization
Germain, Andrew R, Bruggemeyer, Daniel M, Zhu, Jianglong, Genet, Cedric, O’Brien, Peter, Porco, John A
Published in Journal of organic chemistry (15.04.2011)
Published in Journal of organic chemistry (15.04.2011)
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Inhibitors of Glycogen Synthase Kinase 3 with Exquisite Kinome-Wide Selectivity and Their Functional Effects
Wagner, Florence F, Bishop, Joshua A, Gale, Jennifer P, Shi, Xi, Walk, Michelle, Ketterman, Joshua, Patnaik, Debasis, Barker, Doug, Walpita, Deepika, Campbell, Arthur J, Nguyen, Shannon, Lewis, Michael, Ross, Linda, Weïwer, Michel, An, W. Frank, Germain, Andrew R, Nag, Partha P, Metkar, Shailesh, Kaya, Taner, Dandapani, Sivaraman, Olson, David E, Barbe, Anne-Laure, Lazzaro, Fanny, Sacher, Joshua R, Cheah, Jaime H, Fei, David, Perez, Jose, Munoz, Benito, Palmer, Michelle, Stegmaier, Kimberly, Schreiber, Stuart L, Scolnick, Edward, Zhang, Yan-Ling, Haggarty, Stephen J, Holson, Edward B, Pan, Jen Q
Published in ACS chemical biology (15.07.2016)
Published in ACS chemical biology (15.07.2016)
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Identification of a selective small molecule inhibitor of breast cancer stem cells
Germain, Andrew R., Carmody, Leigh C., Morgan, Barbara, Fernandez, Cristina, Forbeck, Erin, Lewis, Timothy A., Nag, Partha P., Ting, Amal, VerPlank, Lynn, Feng, Yuxiong, Perez, Jose R., Dandapani, Sivaraman, Palmer, Michelle, Lander, Eric S., Gupta, Piyush B., Schreiber, Stuart L., Munoz, Benito
Published in Bioorganic & medicinal chemistry letters (15.05.2012)
Published in Bioorganic & medicinal chemistry letters (15.05.2012)
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Journal Article
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells
Germain, Andrew R., Carmody, Leigh C., Nag, Partha P., Morgan, Barbara, VerPlank, Lynn, Fernandez, Cristina, Donckele, Etienne, Feng, Yuxiong, Perez, Jose R., Dandapani, Sivaraman, Palmer, Michelle, Lander, Eric S., Gupta, Piyush B., Schreiber, Stuart L., Munoz, Benito
Published in Bioorganic & medicinal chemistry letters (15.03.2013)
Published in Bioorganic & medicinal chemistry letters (15.03.2013)
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Phenotypic high-throughput screening elucidates target pathway in breast cancer stem cell-like cells
Carmody, Leigh C, Germain, Andrew R, VerPlank, Lynn, Nag, Partha P, Muñoz, Benito, Perez, Jose R, Palmer, Michelle A J
Published in Journal of biomolecular screening (01.10.2012)
Published in Journal of biomolecular screening (01.10.2012)
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Identification of small-molecule inhibitors of Trypansoma cruzi replication
Germain, Andrew R., Carmody, Leigh C., Dockendorff, Chris, Galan-Rodriguez, Cristina, Rodriguez, Ana, Johnston, Stephen, Bittker, Joshua A., MacPherson, Lawrence, Dandapani, Sivaraman, Palmer, Michelle, Schreiber, Stuart L., Munoz, Benito
Published in Bioorganic & medicinal chemistry letters (01.12.2011)
Published in Bioorganic & medicinal chemistry letters (01.12.2011)
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Journal Article
Macrocyclic Hedgehog Pathway Inhibitors: Optimization of Cellular Activity and Mode of Action Studies
Dockendorff, Chris, Nagiec, Marek M, Weïwer, Michel, Buhrlage, Sara, Ting, Amal, Nag, Partha P, Germain, Andrew, Kim, Han-Je, Youngsaye, Willmen, Scherer, Christina, Bennion, Melissa, Xue, Linlong, Stanton, Benjamin Z, Lewis, Timothy A, MacPherson, Lawrence, Palmer, Michelle, Foley, Michael A, Perez, José R, Schreiber, Stuart L
Published in ACS medicinal chemistry letters (11.10.2012)
Published in ACS medicinal chemistry letters (11.10.2012)
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Diversity-Oriented Synthesis Yields a New Drug Lead for Treatment of Chagas Disease
Dandapani, Sivaraman, Germain, Andrew R, Jewett, Ivan, le Quement, Sebastian, Marie, Jean-Charles, Muncipinto, Giovanni, Duvall, Jeremy R, Carmody, Leigh C, Perez, Jose R, Engel, Juan C, Gut, Jiri, Kellar, Danielle, Siqueira-Neto, Jair Lage, McKerrow, James H, Kaiser, Marcel, Rodriguez, Ana, Palmer, Michelle A, Foley, Michael, Schreiber, Stuart L, Munoz, Benito
Published in ACS medicinal chemistry letters (13.02.2014)
Published in ACS medicinal chemistry letters (13.02.2014)
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Discovery of bisamide-heterocycles as inhibitors of scavenger receptor BI (SR-BI)-mediated lipid uptake
Dockendorff, Chris, Faloon, Patrick W., Germain, Andrew, Yu, Miao, Youngsaye, Willmen, Nag, Partha P., Bennion, Melissa, Penman, Marsha, Nieland, Thomas J.F., Dandapani, Sivaraman, Perez, José R., Munoz, Benito, Palmer, Michelle A., Schreiber, Stuart L., Krieger, Monty
Published in Bioorganic & medicinal chemistry letters (15.06.2015)
Published in Bioorganic & medicinal chemistry letters (15.06.2015)
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Year of Publication 27.09.2018
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Year of Publication 27.09.2018
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LARGER SCALE PREPARATION OF OPTICALLY-ACTIVE ALLYLIC ALCOHOLS
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Published in Journal of the Chemical Society, Perkin Transactions 1 (1993)
Published in Journal of the Chemical Society, Perkin Transactions 1 (1993)
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Year of Publication 26.05.2022
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Year of Publication 26.05.2022
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Kinase inhibitors and methods of use thereof
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Year of Publication 06.07.2021
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Year of Publication 06.07.2021
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GSK3 INHIBITORS AND METHODS OF USE THEREOF
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Year of Publication 15.12.2020
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Year of Publication 15.12.2020
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GSK3 INHIBITORS AND METHODS OF USE THEREOF
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Year of Publication 30.09.2019
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Year of Publication 30.09.2019
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