Total synthesis of bryostatin 3
Trost, Barry M, Wang, Youliang, Buckl, Andreas K, Huang, Zhongxing, Nguyen, Minh H, Kuzmina, Olesya
Published in Science (American Association for the Advancement of Science) (29.05.2020)
Published in Science (American Association for the Advancement of Science) (29.05.2020)
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Journal Article
Spirocyclic Oxetanes: Synthesis and Properties
Wuitschik, Georg, Rogers-Evans, Mark, Buckl, Andreas, Bernasconi, Maurizio, Märki, Moritz, Godel, Thierry, Fischer, Holger, Wagner, Björn, Parrilla, Isabelle, Schuler, Franz, Schneider, Josef, Alker, André, Schweizer, W. Bernd, Müller, Klaus, Carreira, Erick M.
Published in Angewandte Chemie (International ed.) (02.06.2008)
Published in Angewandte Chemie (International ed.) (02.06.2008)
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Journal Article
Abstract 1273: Discovery of a potent, selective, and orally bioavailable SOS1 inhibitor, RMC-023, an in vivo tool compound that blocks RAS activation via disruption of the RAS-SOS1 interaction
Buckl, Andreas, Quintana, Elsa, Lee, Grace J., Shifrin, Nataliya, Zhong, Mengqi, Garrenton, Lindsay S., Montgomery, David C., Stahlhut, Carlos, Zhao, Frances, Whalen, Dan M., Thompson, Severin K., Tambo-ong, Arlyn, Gliedt, Micah, Knox, John E., Cregg, James J., Aay, Naing, Choi, Jong, Nguyen, Bao, Tripathi, Atti, Zhao, Ruiping, Saldajeno-Concar, Mae, Marquez, Abby, Hsieh, Daphne, McDowell, Laura L., Koltun, Elena S., Bermingham, Alun, Wildes, David, Singh, Mallika, Wang, Zhengping, Hansen, Richard, Smith, Jan A., Gill, Adrian L.
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Journal Article
Abstract 4877: Allosteric inhibition of SHP2 variants containing cancer-associated activating mutations
Wildes, David, Aay, Naing, Buckl, Andreas, Hsieh, Daphne, Jogalekar, Ashutosh S., Kiss, Gert, Koltun, Elena S., Marquez, Abby, Mellem, Kevin T., Romero, Jason, Saldajeno-Concar, Mae, Schulze, Christopher J., Semko, Chris M., Won, Walter, Nichols, Robert J., Stahlhut, Carlos, Tzitzilonis, Christos, Gill, Adrian L., Smith, Jacqueline A.
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Abstract 4878: RMC-4550, an allosteric inhibitor of SHP2: Synthesis, structure, and anti-tumor activity
Koltun, Elena S., Aay, Naing, Buckl, Andreas, Jogalekar, Ashutosh S., Kiss, Gert, Marquez, Abby, Mellem, Kevin T., Mordec, Kasia, Saldajeno-Concar, Mae, Semko, Chris M., Tibrewal, Nidhi, Tzitzilonis, Christos, Won, Walter, Smith, Jacqueline A., Wilson, Susan E., Nichols, Robert J., Wang, Zhengping, Wilds, David, Singh, Mallika, Gill, Adrian L.
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Abstract 1598: RM-046, a first-in-class, mutant-selective, and oral KRASQ61H(ON) inhibitor that drives tumor regression in preclinical models and validates KRASQ61H as a therapeutic target
Yang, Yu C., Thompson, Severin, Montgomery, David, Quiñones, Antonio J., Wei, Xing, Madej, Benjamin, Tomlinson, Aidan, Shifrin, Nataliya T., McNamara, Alexander, Ahler, Ethan, McDowell, Laura L., Flagella, Michael, Setser, John, Chang, Stephanie, Wang, Zhican, Wang, Zhengping, Huang, Jun, Ballmer, Steve, li, Shaong, Buckl, Andreas, Koltun, Elena, Gill, Adrian, Jiang, Jingjing, Singh, Mallika, Smith, Jacqueline A.
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Published in Cancer research (Chicago, Ill.) (04.04.2023)
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Journal Article
The Search for Tricyanomethane (Cyanoform)
Šišak, Dubravka, McCusker, Lynne B., Buckl, Andreas, Wuitschik, Georg, Wu, Yi-Lin, Schweizer, W. Bernd, Dunitz, Jack D.
Published in Chemistry : a European journal (25.06.2010)
Published in Chemistry : a European journal (25.06.2010)
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Journal Article
Inside Cover: Spirocyclic Oxetanes: Synthesis and Properties (Angew. Chem. Int. Ed. 24/2008)
Wuitschik, Georg, Rogers-Evans, Mark, Buckl, Andreas, Bernasconi, Maurizio, Märki, Moritz, Godel, Thierry, Fischer, Holger, Wagner, Björn, Parrilla, Isabelle, Schuler, Franz, Schneider, Josef, Alker, André, Schweizer, W. Bernd, Müller, Klaus, Carreira, Erick M.
Published in Angewandte Chemie (International ed.) (02.06.2008)
Published in Angewandte Chemie (International ed.) (02.06.2008)
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Journal Article
SOS1 INHIBITORS AND USES THEREOF
THOMPSON, Severin, DUNCTON, Matthew Alexander James, BUCKL, Andreas, GILL, Adrian L, KNOX, John E
Year of Publication 04.04.2024
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Year of Publication 04.04.2024
Patent
PYRIDINE COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS
KISS, Gert, GILL, Adrian, AAY, Naing, MELLEM, Kevin, SEMKO, Christopher, BUCKL, Andreas, KOLTUN, Elena S
Year of Publication 21.03.2024
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Year of Publication 21.03.2024
Patent
SOS1 INHIBITORS AND USES THEREOF
THOMPSON, Severin, DUNCTON, Matthew Alexander James, BUCKL, Andreas, GILL, Adrian L, KNOX, John E
Year of Publication 09.11.2023
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Year of Publication 09.11.2023
Patent
PYRIDINE COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS
KISS, Gert, GILL, Adrian, AAY, Naing, MELLEM, Kevin, SEMKO, Christopher, BUCKL, Andreas, KOLTUN, Elena S
Year of Publication 11.10.2023
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Year of Publication 11.10.2023
Patent
PYRIDINE COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS
KISS, Gert, GILL, Adrian, AAY, Naing, MELLEM, Kevin, SEMKO, Christopher, BUCKL, Andreas, KOLTUN, Elena S
Year of Publication 23.08.2023
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Year of Publication 23.08.2023
Patent
COMPOUNDS, COMPLEXES, AND METHODS FOR THEIR PREPARATION AND OF THEIR USE
BURNETT, G, KNOX, John, GILL, Adrian, KOLTUN, Elena, PITZEN, Jennifer, SEMKO, Christopher, EDWARDS, Anne, AGGEN, James, BUCKL, Andreas, GLIEDT, Micah
Year of Publication 20.06.2024
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Year of Publication 20.06.2024
Patent