Enhanced pulmonary absorption of poorly soluble itraconazole by micronized cocrystal dry powder formulations
Karashima, Masatoshi, Sano, Noriyasu, Yamamoto, Syunsuke, Arai, Yuta, Yamamoto, Katsuhiko, Amano, Nobuyuki, Ikeda, Yukihiro
Published in European journal of pharmaceutics and biopharmaceutics (01.06.2017)
Published in European journal of pharmaceutics and biopharmaceutics (01.06.2017)
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Journal Article
Characterization of plasma protein binding in two mouse models of humanized liver, PXB mouse and humanized TK-NOG mouse
Miyamoto, Maki, Kosugi, Yohei, Iwasaki, Shinji, Chisaki, Ikumi, Nakagawa, Sayaka, Amano, Nobuyuki, Hirabayashi, Hideki
Published in Xenobiotica (02.01.2021)
Published in Xenobiotica (02.01.2021)
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Journal Article
Relationship of MATE1 Inhibition and Cytotoxicity in Nephrotoxicity: Application for Safety Evaluation in Early Drug Discovery
Tohyama, Kimio, Chisaki, Ikumi, Takai, Yuichi, Handa, Yasuhiro, Miyamoto, Makoto, Amano, Nobuyuki
Published in Toxicological sciences (01.07.2019)
Published in Toxicological sciences (01.07.2019)
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Journal Article
Direct Drug Delivery of Low-Permeable Compounds to the Central Nervous System Via Intranasal Administration in Rats and Monkeys
Iwasaki, Shinji, Yamamoto, Syunsuke, Sano, Noriyasu, Tohyama, Kimio, Kosugi, Yohei, Furuta, Atsutoshi, Hamada, Teruki, Igari, Tomoko, Fujioka, Yasushi, Hirabayashi, Hideki, Amano, Nobuyuki
Published in Pharmaceutical research (01.05.2019)
Published in Pharmaceutical research (01.05.2019)
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Journal Article
Appropriate risk criteria for OATP inhibition at the drug discovery stage based on the clinical relevancy between OATP inhibitors and drug-induced adverse effect
Nakakariya, Masanori, Goto, Akihiko, Amano, Nobuyuki
Published in Drug metabolism and pharmacokinetics (01.10.2016)
Published in Drug metabolism and pharmacokinetics (01.10.2016)
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Journal Article
Novel Application of Cultured Epithelial Autografts (CEA) with Expanded Mesh Skin Grafting Over an Artificial Dermis or Dermal Wound Bed Preparation
Akita, Sadanori, Hayashida, Kenji, Yoshimoto, Hiroshi, Fujioka, Masaki, Senju, Chikako, Morooka, Shin, Nishimura, Gozo, Mukae, Nobuhiko, Kobayashi, Kazuo, Anraku, Kuniaki, Murakami, Ryuichi, Hirano, Akiyoshi, Oishi, Masao, Ikenoya, Shintaro, Amano, Nobuyuki, Nakagawa, Hiroshi
Published in International journal of molecular sciences (01.01.2018)
Published in International journal of molecular sciences (01.01.2018)
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Journal Article
Discovery of a Novel Series of N‑Phenylindoline-5-sulfonamide Derivatives as Potent, Selective, and Orally Bioavailable Acyl CoA:Monoacylglycerol Acyltransferase‑2 Inhibitors
Sato, Kenjiro, Takahagi, Hiroki, Yoshikawa, Takeshi, Morimoto, Shinji, Takai, Takafumi, Hidaka, Kousuke, Kamaura, Masahiro, Kubo, Osamu, Adachi, Ryutaro, Ishii, Tsuyoshi, Maki, Toshiyuki, Mochida, Taisuke, Takekawa, Shiro, Nakakariya, Masanori, Amano, Nobuyuki, Kitazaki, Tomoyuki
Published in Journal of medicinal chemistry (14.05.2015)
Published in Journal of medicinal chemistry (14.05.2015)
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Journal Article
Pharmacological Inhibition of Monoacylglycerol O-Acyltransferase 2 Improves Hyperlipidemia, Obesity, and Diabetes by Change in Intestinal Fat Utilization
Take, Kazumi, Mochida, Taisuke, Maki, Toshiyuki, Satomi, Yoshinori, Hirayama, Megumi, Nakakariya, Masanori, Amano, Nobuyuki, Adachi, Ryutaro, Sato, Kenjiro, Kitazaki, Tomoyuki, Takekawa, Shiro
Published in PloS one (03.03.2016)
Published in PloS one (03.03.2016)
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Journal Article
Quantitative Investigation of the Impact of P-Glycoprotein Inhibition on Drug Transport across Blood-Brain Barrier in Rats
SUGIMOTO, Hiroshi, HIRABAYASHI, Hideki, KIMURA, Yoshiaki, FURUTA, Atsutoshi, AMANO, Nobuyuki, MORIWAKI, Toshiya
Published in Drug metabolism and disposition (01.01.2011)
Published in Drug metabolism and disposition (01.01.2011)
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Journal Article
Utility of Göttingen minipigs for Prediction of Human Pharmacokinetic Profiles After Dermal Drug Application
Yamamoto, Syunsuke, Karashima, Masatoshi, Sano, Noriyasu, Fukushi, Chiharu, Tohyama, Kimio, Arai, Yuta, Hirabayashi, Hideki, Amano, Nobuyuki
Published in Pharmaceutical research (01.11.2017)
Published in Pharmaceutical research (01.11.2017)
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Journal Article
Evaluation of Acid Tolerance of Drugs Using Rats and Dogs Controlled for Gastric Acid Secretion
Kosugi, Yohei, Yamamoto, Syunsuke, Sano, Noriyasu, Furuta, Atsutoshi, Igari, Tomoko, Fujioka, Yasushi, Amano, Nobuyuki
Published in Journal of pharmaceutical sciences (01.09.2015)
Published in Journal of pharmaceutical sciences (01.09.2015)
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Journal Article
Establishment of In Vitro P-Glycoprotein Inhibition Assay and Its Exclusion Criteria to Assess the Risk Of Drug–Drug Interaction at the Drug Discovery Stage
Sugimoto, Hiroshi, Matsumoto, Shin-Ichi, Tachibana, Miho, Niwa, Shin-Ichi, Hirabayashi, Hideki, Amano, Nobuyuki, Moriwaki, Toshiya
Published in Journal of pharmaceutical sciences (01.09.2011)
Published in Journal of pharmaceutical sciences (01.09.2011)
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Journal Article
Discovery of TAK-960: An orally available small molecule inhibitor of polo-like kinase 1 (PLK1)
Nie, Zhe, Feher, Victoria, Natala, Srinivasa, McBride, Christopher, Kiryanov, Andre, Jones, Benjamin, Lam, Betty, Liu, Yan, Kaldor, Stephen, Stafford, Jeffrey, Hikami, Kouki, Uchiyama, Noriko, Kawamoto, Tomohiro, Hikichi, Yuichi, Matsumoto, Shin-ichi, Amano, Nobuyuki, Zhang, Lilly, Hosfield, David, Skene, Robert, Zou, Hua, Cao, Xiaodong, Ichikawa, Takashi
Published in Bioorganic & medicinal chemistry letters (15.06.2013)
Published in Bioorganic & medicinal chemistry letters (15.06.2013)
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Journal Article
Optimization of a novel series of N-phenylindoline-5-sulfonamide-based acyl CoA:monoacylglycerol acyltransferase-2 inhibitors: Mitigation of CYP3A4 time-dependent inhibition and phototoxic liabilities
Sato, Kenjiro, Takahagi, Hiroki, Kubo, Osamu, Hidaka, Kousuke, Yoshikawa, Takeshi, Kamaura, Masahiro, Nakakariya, Masanori, Amano, Nobuyuki, Adachi, Ryutaro, Maki, Toshiyuki, Take, Kazumi, Takekawa, Shiro, Kitazaki, Tomoyuki, Maekawa, Tsuyoshi
Published in Bioorganic & medicinal chemistry (01.08.2015)
Published in Bioorganic & medicinal chemistry (01.08.2015)
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Journal Article
A Short-Length Peptide YY Analogue with Anorectic Effect in Mice
Nishizawa, Naoki, Niida, Ayumu, Masuda, Yasushi, Kumano, Satoshi, Yokoyama, Kotaro, Hirabayashi, Hideki, Amano, Nobuyuki, Ohtaki, Tetsuya, Asami, Taiji
Published in ACS omega (31.05.2017)
Published in ACS omega (31.05.2017)
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Journal Article
Asymmetric Intestinal First-Pass Metabolism Causes Minimal Oral Bioavailability of Midazolam in Cynomolgus Monkey
NISHIMURA, Tomohiro, AMANO, Nobuyuki, KUBO, Yoshiyuki, ONO, Midori, KATO, Yukio, FUJITA, Hisashi, KIMURA, Yoshiaki, TSUJI, Akira
Published in Drug metabolism and disposition (01.08.2007)
Published in Drug metabolism and disposition (01.08.2007)
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Journal Article
Construction and Functional Evaluation of a Three-Dimensional Blood–Brain Barrier Model Equipped With Human Induced Pluripotent Stem Cell-Derived Brain Microvascular Endothelial Cells
Kurosawa, Toshiki, Sako, Daiki, Tega, Yuma, Debori, Yasuyuki, Tomihara, Yumi, Aoyama, Kazunobu, Kubo, Yoshiyuki, Amano, Nobuyuki, Deguchi, Yoshiharu
Published in Pharmaceutical research (01.07.2022)
Published in Pharmaceutical research (01.07.2022)
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