Assessing the Use of the sGC Stimulator BAY-747, as a Potential Treatment for Duchenne Muscular Dystrophy
Krishnan, Shalini Murali, Nordlohne, Johannes, Dietz, Lisa, Vakalopoulos, Alexandros, Haning, Petra, Hartmann, Elke, Seifert, Roland, Hüser, Jörg, Mathar, Ilka, Sandner, Peter
Published in International journal of molecular sciences (01.08.2021)
Published in International journal of molecular sciences (01.08.2021)
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Journal Article
Investigations Into Chemically Stabilized Four-Letter DNA for DNA-Encoded Chemistry
Potowski, Marco, Kunig, Verena B. K., Eberlein, Lukas, Škopić, Mateja Klika, Vakalopoulos, Alexandros, Kast, Stefan M., Brunschweiger, Andreas
Published in Frontiers in chemistry (09.06.2022)
Published in Frontiers in chemistry (09.06.2022)
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Identification and characterization of the new generation soluble guanylate cyclase stimulator BAY‐747 designed for the treatment of resistant hypertension
Wunder, Frank, Stasch, Johannes‐Peter, Knorr, Andreas, Mondritzki, Thomas, Brockschnieder, Damian, Becker‐Pelster, Eva‐Maria, Sandner, Peter, Tinel, Hanna, Redlich, Gorden, Hartung, Ingo V., Vakalopoulos, Alexandros, Follmann, Markus
Published in British journal of pharmacology (01.10.2023)
Published in British journal of pharmacology (01.10.2023)
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Neladenoson Bialanate Hydrochloride: A Prodrug of a Partial Adenosine A1 Receptor Agonist for the Chronic Treatment of Heart Diseases
Meibom, Daniel, Albrecht‐Küpper, Barbara, Diedrichs, Nicole, Hübsch, Walter, Kast, Raimund, Krämer, Thomas, Krenz, Ursula, Lerchen, Hans‐Georg, Mittendorf, Joachim, Nell, Peter G., Süssmeier, Frank, Vakalopoulos, Alexandros, Zimmermann, Katja
Published in ChemMedChem (22.05.2017)
Published in ChemMedChem (22.05.2017)
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Journal Article
New Generation of sGC Stimulators: Discovery of Imidazo[1,2‑a]pyridine Carboxamide BAY 1165747 (BAY-747), a Long-Acting Soluble Guanylate Cyclase Stimulator for the Treatment of Resistant Hypertension
Vakalopoulos, Alexandros, Wunder, Frank, Hartung, Ingo V., Redlich, Gorden, Jautelat, Rolf, Buchgraber, Philipp, Hassfeld, Jorma, Gromov, Alexey V., Lindner, Niels, Bierer, Donald, Gries, Jörg, Kroh, Walter, Paulsen, Holger, Mittendorf, Joachim, Lang, Dieter, Becker-Pelster, Eva, Brockschnieder, Damian, Geiss, Volker, Li, Volkhart, Straub, Alexander, Knorr, Andreas, Mondritzki, Thomas, Trübel, Hubert, Raschke, Marian, Schaefer, Martina, Thomas, Dirk, Sandner, Peter, Stasch, Johannes-Peter, Follmann, Markus
Published in Journal of medicinal chemistry (08.06.2023)
Published in Journal of medicinal chemistry (08.06.2023)
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Journal Article
Neladenoson Bialanate Hydrochloride: A Prodrug of a Partial Adenosine A(1) Receptor Agonist for the Chronic Treatment of Heart Diseases
Meibom, Daniel, Albrecht-Kuepper, Barbara, Diedrichs, Nicole, Huebsch, Walter, Kast, Raimund, Kraemer, Thomas, Krenz, Ursula, Lerchen, Hans-Georg, Mittendorf, Joachim, Nell, Peter G., Suessmeier, Frank, Vakalopoulos, Alexandros, Zimmermann, Katja
Published in ChemMedChem (22.05.2017)
Published in ChemMedChem (22.05.2017)
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Journal Article
Novel tetrahydrochinoline derived CETP inhibitors
Schmeck, Carsten, Gielen-Haertwig, Heike, Vakalopoulos, Alexandros, Bischoff, Hilmar, Li, Volkhart, Wirtz, Gabriele, Weber, Olaf
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
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Journal Article
Quinazolinone Derivatives as Orally Available Ghrelin Receptor Antagonists for the Treatment of Diabetes and Obesity
Rudolph, Joachim, Esler, William P, O'Connor, Stephen, Coish, Philip D. G, Wickens, Philip L, Brands, Michael, Bierer, Donald E, Bloomquist, Brian T, Bondar, Georgiy, Chen, Libing, Chuang, Chih-Yuan, Claus, Thomas H, Fathi, Zahra, Fu, Wenlang, Khire, Uday R, Kristie, James A, Liu, Xiao-Gao, Lowe, Derek B, McClure, Andrea C, Michels, Martin, Ortiz, Astrid A, Ramsden, Philip D, Schoenleber, Robert W, Shelekhin, Tatiana E, Vakalopoulos, Alexandros, Tang, Weifeng, Wang, Lei, Yi, Lin, Gardell, Stephen J, Livingston, James N, Sweet, Laurel J, Bullock, William H
Published in Journal of medicinal chemistry (18.10.2007)
Published in Journal of medicinal chemistry (18.10.2007)
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Journal Article
Neladenoson Bialanate Hydrochloride: A Prodrug of a Partial Adenosine A 1 Receptor Agonist for the Chronic Treatment of Heart Diseases
Meibom, Daniel, Albrecht-Küpper, Barbara, Diedrichs, Nicole, Hübsch, Walter, Kast, Raimund, Krämer, Thomas, Krenz, Ursula, Lerchen, Hans-Georg, Mittendorf, Joachim, Nell, Peter G, Süssmeier, Frank, Vakalopoulos, Alexandros, Zimmermann, Katja
Published in ChemMedChem (22.05.2017)
Published in ChemMedChem (22.05.2017)
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Journal Article
Chromanol derivatives—A novel class of CETP inhibitors
Vakalopoulos, Alexandros, Schmeck, Carsten, Thutewohl, Michael, Li, Volkhart, Bischoff, Hilmar, Lustig, Klemens, Weber, Olaf, Paulsen, Holger, Elias, Harry
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
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Journal Article
Neladenoson Bialanate Hydrochloride: A Prodrug of a Partial AdenosineA1 Receptor Agonist for the Chronic Treatment of Heart Diseases
Meibom, Daniel, Albrecht-Kupper, Barbara, Diedrichs, Nicole, Hubsch, Walter, Kast, Raimund, Kramer, Thomas, Krenz, Ursula, Lerchen, Hans-Georg, Mittendorf, Joachim, Nell, Peter G, Sussmeier, Frank, Vakalopoulos, Alexandros, Zimmermann, Katja
Published in ChemMedChem (01.05.2017)
Published in ChemMedChem (01.05.2017)
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Journal Article
New copper-mediated O-arylations of phenols with arylstannanes
Vakalopoulos, Alexandros, Kavazoudi, Xanthoula, Schoof, Joachim
Published in Tetrahedron letters (27.11.2006)
Published in Tetrahedron letters (27.11.2006)
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Prediction of a potentially effective dose in humans for BAY 60–5521, a potent inhibitor of cholesteryl ester transfer protein (CETP) by allometric species scaling and combined pharmacodynamic and physiologically‐based pharmacokinetic modelling
Weber, Olaf, Willmann, Stefan, Bischoff, Hilmar, Li, Volkhart, Vakalopoulos, Alexandros, Lustig, Klemens, Hafner, Frank‐Thorsten, Heinig, Roland, Schmeck, Carsten, Buehner, Klaus
Published in British journal of clinical pharmacology (01.02.2012)
Published in British journal of clinical pharmacology (01.02.2012)
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Journal Article
Chemisch stabilisierte DNA‐Codes für DNA‐kodierte Chemie
Potowski, Marco, Kunig, Verena B. K., Eberlein, Lukas, Vakalopoulos, Alexandros, Kast, Stefan M., Brunschweiger, Andreas
Published in Angewandte Chemie (01.09.2021)
Published in Angewandte Chemie (01.09.2021)
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Journal Article
Dibenzodioxocinones—A new class of CETP inhibitors
Brückner, David, Hafner, Frank-Thorsten, Li, Volkhart, Schmeck, Carsten, Telser, Joachim, Vakalopoulos, Alexandros, Wirtz, Gabriele
Published in Bioorganic & medicinal chemistry letters (01.08.2005)
Published in Bioorganic & medicinal chemistry letters (01.08.2005)
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