A Formal [3 + 3] Cycloaddition Reaction. 5. An Enantioselective Intramolecular Formal Aza-[3 + 3] Cycloaddition Reaction Promoted by Chiral Amine Salts
Gerasyuto, Aleksey I, Hsung, Richard P, Sydorenko, Nadiya, Slafer, Brian
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Published in Journal of organic chemistry (27.05.2005)
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AutoDesigner - Core Design, a De Novo Design Algorithm for Chemical Scaffolds: Application to the Design and Synthesis of Novel Selective Wee1 Inhibitors
Bos, Pieter H., Ranalli, Fabio, Flood, Emelie, Watts, Shawn, Inoyama, Daigo, Knight, Jennifer L., Clark, Anthony J., Placzeck, Andrew, Wang, Jiashi, Gerasyuto, Aleksey I., Silvergleid, Sarah, Yin, Wu, Sun, Shaoxian, Abel, Robert, Bhat, Sathesh
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The Discovery of MORF-627, a Highly Selective Conformationally-Biased Zwitterionic Integrin αvβ6 Inhibitor for Fibrosis
Harrison, Bryce A, Dowling, James E, Bursavich, Matthew G, Troast, Dawn M, Chong, Katherine M, Hahn, Kristopher N, Zhong, Cheng, Mulvihill, Kristen M, Nguyen, Hanh, Monroy, Meghan F, Qiao, Qi, Sosa, Brian, Mostafavi, Siavash, Smukste, Inese, Lee, Dooyoung, Cappellucci, Laura, Konopka, Elizabeth H, Nowakowski, Patrycja, Stawski, Lukasz, Senices, Mayra, Nguyen, Minh Hai, Kapoor, Parmita S, Luus, Lia, Sullivan, Andrew, Bortolato, Andrea, Svensson, Mats, Hickey, Eugene R, Konze, Kyle D, Day, Tyler, Kim, Byungchan, Negri, Ana, Gerasyuto, Aleksey I, Moy, Terence I, Lu, Min, Ray, Adrian S, Wang, Liangsu, Cui, Dan, Lin, Fu-Yang, Lippa, Blaise, Rogers, Bruce N
Published in Journal of medicinal chemistry (24.10.2024)
Published in Journal of medicinal chemistry (24.10.2024)
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Discovery and Optimization of Indolyl-Containing 4‑Hydroxy-2-Pyridone Type II DNA Topoisomerase Inhibitors Active against Multidrug Resistant Gram-negative Bacteria
Gerasyuto, Aleksey I, Arnold, Michael A, Wang, Jiashi, Chen, Guangming, Zhang, Xiaoyan, Smith, Sean, Woll, Matthew G, Baird, John, Zhang, Nanjing, Almstead, Neil G, Narasimhan, Jana, Peddi, Srinivasa, Dumble, Melissa, Sheedy, Josephine, Weetall, Marla, Branstrom, Arthur A, Prasad, J. V. N, Karp, Gary M
Published in Journal of medicinal chemistry (24.05.2018)
Published in Journal of medicinal chemistry (24.05.2018)
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4-Hydroxy-2-pyridones: Discovery and evaluation of a novel class of antibacterial agents targeting DNA synthesis
Arnold, Michael A., Gerasyuto, Aleksey I., Wang, Jiashi, Du, Wu, Gorske, Yi Jin Kim, Arasu, Tamil, Baird, John, Almstead, Neil G., Narasimhan, Jana, Peddi, Srinivasa, Ginzburg, Olya, Lue, Stanley W., Hedrick, Jean, Sheedy, Josephine, Lagaud, Guy, Branstrom, Arthur A., Weetall, Marla, Prasad, J.V.N. Vara, Karp, Gary M.
Published in Bioorganic & medicinal chemistry letters (15.11.2017)
Published in Bioorganic & medicinal chemistry letters (15.11.2017)
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Correction to Discovery and Optimization of Indolyl-Containing 4‑Hydroxy-2-pyridone Type II DNA Topoisomerase Inhibitors Active against Multidrug Resistant Gram-Negative Bacteria
Gerasyuto, Aleksey I, Arnold, Michael A, Wang, Jiashi, Chen, Guangming, Zhang, Xiaoyan, Smith, Sean, Woll, Matthew G, Baird, John, Zhang, Nanjing, Almstead, Neil G, Narasimhan, Jana, Peddi, Srinivasa, Dumble, Melissa, Sheedy, Josephine, Weetall, Marla, Branstrom, Arthur A, Prasad, J. V. N, Karp, Gary M
Published in Journal of medicinal chemistry (25.10.2018)
Published in Journal of medicinal chemistry (25.10.2018)
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Stereoselective Formal [3 + 3] Cycloaddition Approach to cis-1-Azadecalins and Synthesis of (−)-4a,8a-diepi-Pumiliotoxin C. Evidence for the First Highly Stereoselective 6π-Electron Electrocyclic Ring Closures of 1-Azatrienes
Sklenicka, Heather M, Hsung, Richard P, McLaughlin, Michael J, Wei, Lin-li, Gerasyuto, Aleksey I, Brennessel, William B
Published in Journal of the American Chemical Society (04.09.2002)
Published in Journal of the American Chemical Society (04.09.2002)
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A Novel and Highly Stereoselective Intramolecular Formal [3+3] Cycloaddition Reaction of Vinylogous Amides Tethered with α,β-Unsaturated Aldehydes: A Formal Total Synthesis of (+)-Gephyrotoxin
Wei, Lin-Li, Hsung, Richard P., Sklenicka, Heather M., Gerasyuto, Aleksey I.
Published in Angewandte Chemie International Edition (17.04.2001)
Published in Angewandte Chemie International Edition (17.04.2001)
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Total syntheses of enantiomerically enriched R-(+)- and S-(-)-deplancheine
Sydorenko, N, Zificsak, CA, Gerasyuto, AI, Hsung, RP
Published in Organic & biomolecular chemistry (07.06.2005)
Published in Organic & biomolecular chemistry (07.06.2005)
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A Formal [3 + 3] Cycloaddition Reaction. Improved Reactivity Using α,β-Unsaturated Iminium Salts and Evidence for Reversibility of 6π-Electron Electrocyclic Ring Closure of 1-Oxatrienes
Shen, Hong C, Wang, Jiashi, Cole, Kevin P, McLaughlin, Michael J, Morgan, Christopher D, Douglas, Christopher J, Hsung, Richard P, Coverdale, Heather A, Gerasyuto, Aleksey I, Hahn, Juliet M, Liu, Jia, Sklenicka, Heather M, Wei, Lin-Li, Zehnder, Luke R, Zificsak, Craig A
Published in Journal of organic chemistry (07.03.2003)
Published in Journal of organic chemistry (07.03.2003)
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A CYCLIC ACETAL TETHERED INTRAMOLECULAR DIELS-ALDER CYCLOADDITION. STUDIES DIRECTED TOWARD A TOTAL SYNTHESIS OF (+/-)-FUSIDILACTONE C
Ghosh, Sunil K., Wei, Yonggang, Gerasyuto, Aleksey I., Feltenberger, John B., Wang, Jiashi, Hsung, Richard P.
Published in Heterocycles (01.03.2011)
Published in Heterocycles (01.03.2011)
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INHIBITING HUMAN INTEGRIN α4β7
BLAISE S LIPPA, CUI DAN, BRYCE A HARRISON, KIM BYUNGCHAN, EUGENE HICKEY, ROBERT ZAHLER, TYLER DAY, EVELYNE HOUANG, ALEKSEY I GERASYUTO, MATTHEW G BURSAVICH, KYLE D KONZE, BRUCE N ROGERS, JAMES E DOWLING, SALMA RAFI, KRISTOPHER N HAHN, LIN FU-YANG, DAWN M TROAST, ZHONG CHENG
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Year of Publication 16.04.2024
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BLAISE S LIPPA, BRYCE A HARRISON, KIM BYUNGCHAN, TYLER DAY, ALEKSEY I GERASYUTO, MATTHEW G BURSAVICH, KYLE D KONZE, BRUCE N ROGERS, ALEXEY A LUGOVSKOY, KRISTOPHER N HAHN, LIN FU-YANG, BRIAN SOSA, DAWN M TROAST, MATS A SVENSSON, ZHONG CHENG
Year of Publication 09.01.2024
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Year of Publication 09.01.2024
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