Acyclovir Diphosphate Dimyristoylglycerol: A Phospholipid Prodrug with Activity Against Acyclovir-Resistant Herpes Simplex Virus
Hostetler, Karl Y., Parker, Suezanne, Sridhar, C. N., Martin, Michael J., Li, Jui-Lien, Stuhmiller, Louise M., Gijsbert M. T. van Wijk, van den Bosch, Henk, Gardner, Michael F., Aldern, Kathy A., Richman, Douglas D.
Published in Proceedings of the National Academy of Sciences - PNAS (15.12.1993)
Published in Proceedings of the National Academy of Sciences - PNAS (15.12.1993)
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Antiviral effect in human cytomegalovirus-infected cells, pharmacokinetics, and intravitreal toxicology in rabbits of acyclovir diphosphate dimyristoylglycerol
SHAKIBA, S, FREEMAN, W. R, GARDNER, M. F, HOSTETLER, K. Y, FLORES-AGUILAR, M, MUNGUIA, D, TATEBAYASHI, M, BESEN, G, AMANI, R, WILEY, C. A, CHOU VUONG, ALDERN, K. A
Published in Antimicrobial Agents and Chemotherapy (01.06.1995)
Published in Antimicrobial Agents and Chemotherapy (01.06.1995)
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In vitro and in vivo activity of 1-O-hexadecylpropanediol-3-phospho-ganciclovir and 1-O-hexadecylpropanediol-3-phospho-penciclovir in cytomegalovirus and herpes simplex virus infections
Hostetler, K Y, Rybak, R J, Beadle, J R, Gardner, M F, Aldern, K A, Wright, K N, Kern, E R
Published in Antiviral chemistry & chemotherapy (01.01.2001)
Published in Antiviral chemistry & chemotherapy (01.01.2001)
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Alkylthioglycerol Prodrugs of Foscarnet: Synthesis, Oral Bioavailability and Structure–Activity Studies in Human Cytomegalovirus-, Herpes Simplex Virus Type 1- and Human Immunodeficiency Virus Type 1-Infected Cells
Beadle, JR, Kini, GD, Aldern, KA, Gardner, MF, Wright, KN, Richman, DD, Hostetler, KY
Published in Antiviral chemistry & chemotherapy (01.01.1998)
Published in Antiviral chemistry & chemotherapy (01.01.1998)
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Comparative evaluation of amiodarone-induced phospholipidosis and drug accumulation in Fischer-344 and Sprague-Dawley rats
Reasor, Mark J., McCloud, Christy M., Beard, Terry L., Ebert, Debora C., Kacew, sam, Gardner, Michael F., Aldern, Kathy A., Hostetler, Karl Y.
Published in Toxicology (Amsterdam) (08.01.1996)
Published in Toxicology (Amsterdam) (08.01.1996)
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Alkoxy propane prodrugs of foscarnet: effect of alkyl chain length on in vitro antiviral activity in cells infected with HIV-1, HSV-1 and HCMV
Kini, Ganesh D, Beadle, James R, Xie, Hong, Aldern, Kathy A, Richman, Douglas D, Y. Hostetler, Karl
Published in Antiviral research (01.09.1997)
Published in Antiviral research (01.09.1997)
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In vitro Anti-HIV-1 Activity of sn-2-Substituted 1-O-Octadecyl-sn-Glycero-3-Phosphonoformate Analogues and Synergy with Zidovudine
Hostetler, Karl Y, Hammond, Jennifer L, Kini, Ganesh D, Hostetler, Saskia E, Beadle, James R, Aldern, Kathy A, Chou, Ting-Chao, Richman, Douglas D, Mellors, John W
Published in Antiviral chemistry & chemotherapy (01.05.2000)
Published in Antiviral chemistry & chemotherapy (01.05.2000)
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Steroidogenic enzyme activities in cultured human definitive zone adrenocortical cells: comparison with bovine adrenocortical cells and resultant differences in adrenal androgen synthesis
Hornsby, P J, Aldern, K A
Published in The journal of clinical endocrinology and metabolism (01.01.1984)
Published in The journal of clinical endocrinology and metabolism (01.01.1984)
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Alkylglycerol Prodrugs of Phosphonoformate Are Potent In Vitro Inhibitors of Nucleoside-Resistant Human Immunodeficiency Virus Type 1 and Select for Resistance Mutations That Suppress Zidovudine Resistance
HAMMOND, Jennifer L, KOONTZ, Dianna L, BAZMI, Holly Z, BEADLE, James R, HOSTETLER, Saskia E, KINI, Ganesh D, ALDERN, Kathy A, RICHMAN, Douglas D, HOSTETLER, Karl Y, MELLORS, John W
Published in Antimicrobial Agents and Chemotherapy (01.06.2001)
Published in Antimicrobial Agents and Chemotherapy (01.06.2001)
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Selenium deficiency in cultured adrenocortical cells: restoration of glutathione peroxidase and resistance to hydroperoxides on addition of selenium
Hornsby, P J, Pearson, D W, Autor, A P, Aldern, K A, Harris, S E
Published in Journal of cellular physiology (01.04.1985)
Published in Journal of cellular physiology (01.04.1985)
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Evaluation of a novel lipid prodrug for intraocular drug delivery: effect of acyclovir diphosphate dimyristoylglycerol in a rabbit model with herpes simplex virus-1 retinitis
Taskintuna, I, Banker, A S, Flores-Aguilar, M, Bergeron-Lynn, G, Aldern, K A, Hostetler, K Y, Freeman, W R
Published in Retina (Philadelphia, Pa.) (1997)
Published in Retina (Philadelphia, Pa.) (1997)
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Lipid prodrugs of phosphonoacids: greatly enhanced antiviral activity of 1- O-octadecyl- sn-glycero-3-phosphonoformate in HIV-1, HSV-1 and HCMV-infected cells, in vitro
Hostetler, Karl Y., Kini, Ganesh D., Beadle, James R., Aldern, Kathy A., Gardner, Michael F., Border, Richard, Kumar, Raj, Barshak, Lena, Sridhar, C.N., Wheeler, Carl J., Richman, Douglas D.
Published in Antiviral research (01.06.1996)
Published in Antiviral research (01.06.1996)
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Synthesis and Antiviral Evaluation of 1-O-Hexadecylpropanediol-3-P-acyclovir: Efficacy Against HSV-1 Infection in Mice
Beadle, James R., Kini, Ganesh D., Aldern, Kathy A., Gardner, Michael F., Wright, Kristine N., Rybak, Rachel J., Kern, Earl R., Hostetler, Karl Y.
Published in Nucleosides, nucleotides & nucleic acids (01.01.2000)
Published in Nucleosides, nucleotides & nucleic acids (01.01.2000)
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