Preclinical evaluation of FAP-2286 for fibroblast activation protein targeted radionuclide imaging and therapy
Zboralski, Dirk, Hoehne, Aileen, Bredenbeck, Anne, Schumann, Anne, Nguyen, Minh, Schneider, Eberhard, Ungewiss, Jan, Paschke, Matthias, Haase, Christian, von Hacht, Jan L., Kwan, Tanya, Lin, Kevin K., Lenore, Jan, Harding, Thomas C., Xiao, Jim, Simmons, Andrew D., Mohan, Ajay-Mohan, Beindorff, Nicola, Reineke, Ulrich, Smerling, Christiane, Osterkamp, Frank
Published in European journal of nuclear medicine and molecular imaging (01.09.2022)
Published in European journal of nuclear medicine and molecular imaging (01.09.2022)
Get full text
Journal Article
A PET Imaging Strategy to Visualize Activated T Cells in Acute Graft-versus-Host Disease Elicited by Allogenic Hematopoietic Cell Transplant
Ronald, John A, Kim, Byung-Su, Gowrishankar, Gayatri, Namavari, Mohammad, Alam, Israt S, D'Souza, Aloma, Nishikii, Hidekazu, Chuang, Hui-Yen, Ilovich, Ohad, Lin, Chih-Feng, Reeves, Robert, Shuhendler, Adam, Hoehne, Aileen, Chan, Carmel T, Baker, Jeanette, Yaghoubi, Shahriar S, VanBrocklin, Henry F, Hawkins, Randall, Franc, Benjamin L, Jivan, Salma, Slater, James B, Verdin, Emily F, Gao, Kenneth T, Benjamin, Jonathan, Negrin, Robert, Gambhir, Sanjiv Sam
Published in Cancer research (Chicago, Ill.) (01.06.2017)
Published in Cancer research (Chicago, Ill.) (01.06.2017)
Get full text
Journal Article
Modelling ligand depletion for simultaneous affinity and binding site quantification on cells and tissue
Weber, Judith, Djurberg, Klara, Lundsten Salomonsson, Sara, Kamprath, Maria, Hoehne, Aileen, Westin, Hadis, Vergara, Fernanda, Bondza, Sina
Published in Scientific reports (20.06.2023)
Published in Scientific reports (20.06.2023)
Get full text
Journal Article
Antiviral drug ganciclovir is a potent inhibitor of microglial proliferation and neuroinflammation
Ding, Zhaoqing, Mathur, Vidhu, Ho, Peggy P, James, Michelle L, Lucin, Kurt M, Hoehne, Aileen, Alabsi, Haitham, Gambhir, Sanjiv S, Steinman, Lawrence, Luo, Jian, Wyss-Coray, Tony
Published in The Journal of experimental medicine (10.02.2014)
Published in The Journal of experimental medicine (10.02.2014)
Get full text
Journal Article
Feasibility, Biodistribution, and Preliminary Dosimetry in Peptide-Targeted Radionuclide Therapy of Diverse Adenocarcinomas Using 177Lu-FAP-2286: First-in-Humans Results
Baum, Richard P, Schuchardt, Christiane, Singh, Aviral, Chantadisai, Maythinee, Robiller, Franz C, Zhang, Jingjing, Mueller, Dirk, Eismant, Alexander, Almaguel, Frankis, Zboralski, Dirk, Osterkamp, Frank, Hoehne, Aileen, Reineke, Ulrich, Smerling, Christiane, Kulkarni, Harshad R
Published in The Journal of nuclear medicine (1978) (01.03.2022)
Published in The Journal of nuclear medicine (1978) (01.03.2022)
Get full text
Journal Article
3BP-3940, a highly potent FAP-targeting peptide for theranostics - production, validation and first in human experience with Ga-68 and Lu-177
Greifenstein, Lukas, Gunkel, Annika, Hoehne, Aileen, Osterkamp, Frank, Smerling, Christiane, Landvogt, Christian, Mueller, Corinna, Baum, Richard P.
Published in iScience (15.12.2023)
Published in iScience (15.12.2023)
Get full text
Journal Article
Pilot Preclinical and Clinical Evaluation of (4S)-4-(3-[18F]Fluoropropyl)-L-Glutamate (18F-FSPG) for PET/CT Imaging of Intracranial Malignancies
Mittra, Erik S, Koglin, Norman, Mosci, Camila, Kumar, Meena, Hoehne, Aileen, Keu, Khun Visith, Iagaru, Andrei H, Mueller, Andre, Berndt, Mathias, Bullich, Santiago, Friebe, Matthias, Schmitt-Willich, Heribert, Gekeler, Volker, Fels, Lüder M, Bacher-Stier, Claudia, Moon, Dae Hyuk, Chin, Frederick T, Stephens, Andrew W, Dinkelborg, Ludger M, Gambhir, Sanjiv S
Published in PloS one (18.02.2016)
Published in PloS one (18.02.2016)
Get full text
Journal Article
[ 18 F]FSPG-PET reveals increased cystine/glutamate antiporter (xc-) activity in a mouse model of multiple sclerosis
Hoehne, Aileen, James, Michelle L, Alam, Israt S, Ronald, John A, Schneider, Bernadette, D'Souza, Aloma, Witney, Timothy H, Andrews, Lauren E, Cropper, Haley C, Behera, Deepak, Gowrishankar, Gayatri, Ding, Zhaoqing, Wyss-Coray, Tony, Chin, Frederick T, Biswal, Sandip, Gambhir, Sanjiv S
Published in Journal of neuroinflammation (22.02.2018)
Published in Journal of neuroinflammation (22.02.2018)
Get full text
Journal Article
Discovery and validation of small-molecule heat-shock protein 90 inhibitors through multimodality molecular imaging in living subjects
Chan, Carmel T, Reeves, Robert E, Geller, Ron, Yaghoubi, Shahriar S, Hoehne, Aileen, Solow-Cordero, David E, Chiosis, Gabriela, Massoud, Tarik F, Paulmurugan, Ramasamy, Gambhir, Sanjiv S
Published in Proceedings of the National Academy of Sciences - PNAS (11.09.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (11.09.2012)
Get full text
Journal Article
Preclinical Characterization of DPI-4452: A 68 Ga/ 177 Lu Theranostic Ligand for Carbonic Anhydrase IX
Massière, Frédéric, Wiedemann, Norbert, Borrego, Inês, Hoehne, Aileen, Osterkamp, Frank, Paschke, Matthias, Zboralski, Dirk, Schumann, Anne, Bredenbeck, Anne, Brichory, Franck, Attinger, Antoine
Published in Journal of Nuclear Medicine (01.05.2024)
Published in Journal of Nuclear Medicine (01.05.2024)
Get full text
Journal Article
Fibroblast activation protein targeted radiotherapy induces an immunogenic tumor microenvironment and enhances the efficacy of PD-1 immune checkpoint inhibition
Zboralski, Dirk, Osterkamp, Frank, Christensen, Esben, Bredenbeck, Anne, Schumann, Anne, Hoehne, Aileen, Schneider, Eberhard, Paschke, Matthias, Ungewiss, Jan, Haase, Christian, Robillard, Liliane, Simmons, Andrew D., Harding, Thomas C., Nguyen, Minh
Published in European journal of nuclear medicine and molecular imaging (01.07.2023)
Published in European journal of nuclear medicine and molecular imaging (01.07.2023)
Get full text
Journal Article
Assessment of Tumor Redox Status through ( S )-4-(3-[ 18 F]fluoropropyl)-L-Glutamic Acid PET Imaging of System x c - Activity
McCormick, Patrick N, Greenwood, Hannah E, Glaser, Matthias, Maddocks, Oliver D K, Gendron, Thibault, Sander, Kerstin, Gowrishankar, Gayatri, Hoehne, Aileen, Zhang, Tong, Shuhendler, Adam J, Lewis, David Y, Berndt, Mathias, Koglin, Norman, Lythgoe, Mark F, Gambhir, Sanjiv S, Årstad, Erik, Witney, Timothy H
Published in Cancer research (Chicago, Ill.) (15.02.2019)
Published in Cancer research (Chicago, Ill.) (15.02.2019)
Get full text
Journal Article
Abstract LBA032: Pan-cancer analysis of fibroblast activation protein alpha (FAP) expression to guide tumor selection for the peptide-targeted radionuclide therapy FAP-2286
Kwan, Tanya T., Nguyen, Minh, Zboralski, Dirk, Schumann, Anne, Bredenbeck, Anne, Paschke, Matthias, Haase, Christian, Hoehne, Aileen, Reineke, Ulrich, Smerling, Christiane, Osterkamp, Frank, Xiao, Jim, Simmons, Andrew D., Harding, Thomas C., Lin, Kevin L.
Published in Molecular cancer therapeutics (01.12.2021)
Published in Molecular cancer therapeutics (01.12.2021)
Get full text
Journal Article
PET imaging of tumor glycolysis downstream of hexokinase through noninvasive measurement of pyruvate kinase M2
Witney, Timothy H, James, Michelle L, Shen, Bin, Chang, Edwin, Pohling, Christoph, Arksey, Natasha, Hoehne, Aileen, Shuhendler, Adam, Park, Jun-Hyung, Bodapati, Deepika, Weber, Judith, Gowrishankar, Gayatri, Rao, Jianghong, Chin, Frederick T, Gambhir, Sanjiv Sam
Published in Science translational medicine (21.10.2015)
Published in Science translational medicine (21.10.2015)
Get more information
Journal Article
Feasibility, Biodistribution, and Preliminary Dosimetry in Peptide-Targeted Radionuclide Therapy of Diverse Adenocarcinomas Using 177 Lu-FAP-2286: First-in-Humans Results
Baum, Richard P, Schuchardt, Christiane, Singh, Aviral, Chantadisai, Maythinee, Robiller, Franz C, Zhang, Jingjing, Mueller, Dirk, Eismant, Alexander, Almaguel, Frankis, Zboralski, Dirk, Osterkamp, Frank, Hoehne, Aileen, Reineke, Ulrich, Smerling, Christiane, Kulkarni, Harshad R
Published in Journal of Nuclear Medicine (01.03.2022)
Published in Journal of Nuclear Medicine (01.03.2022)
Get full text
Journal Article
[ 18 F]GE-180 PET Detects Reduced Microglia Activation After LM11A-31 Therapy in a Mouse Model of Alzheimer's Disease
James, Michelle L, Belichenko, Nadia P, Shuhendler, Adam J, Hoehne, Aileen, Andrews, Lauren E, Condon, Christina, Nguyen, Thuy-Vi V, Reiser, Vladimer, Jones, Paul, Trigg, William, Rao, Jianghong, Gambhir, Sanjiv S, Longo, Frank M
Published in Theranostics (01.01.2017)
Published in Theranostics (01.01.2017)
Get full text
Journal Article
Silicon-based building blocks for one-step (18)F-radiolabeling of peptides for PET imaging
Mu, Linjing, Hoehne, Aileen, Schubiger, R. August, Ametamey, Simon M., Graham, Keith, Cyr, John E., Dinkelborg, Ludger, Stellfeld, Tmo, Srinivasan, Ananth, Voigtmann, Ulrike, Klar, Ulrich
Published in Angewandte Chemie International Edition (01.01.2008)
Published in Angewandte Chemie International Edition (01.01.2008)
Get full text
Journal Article
A F-18-Labeled Saxitoxin Derivative for in Vivo PET-MR Imaging of Voltage-Gated Sodium Channel Expression Following Nerve Injury
Hoehne, Aileen, Behera, Deepak, Parsons, William H., James, Michelle L., Shen, Bin, Borgohain, Preeti, Bodapati, Deepika, Prabhakar, Archana, Gambhir, Sanjiv S., Yeomans, David C., Biswal, Sandip, Chin, Frederick T., Du Bois, J.
Published in Journal of the American Chemical Society (04.12.2013)
Published in Journal of the American Chemical Society (04.12.2013)
Get full text
Journal Article