The first synthesis of ent-agelasine F
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Published in Tetrahedron (01.01.2009)
Published in Tetrahedron (01.01.2009)
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Journal Article
Synthesis, Antimicrobial and Antineoplastic Activities for Agelasine and Agelasimine Analogs with a β-Cyclocitral Derived Substituent
Proszenyák, Ágnes, Charnock, Colin, Hedner, Erik, Larsson, Rolf, Bohlin, Lars, Gundersen, Lise-Lotte
Published in Archiv der Pharmazie (Weinheim) (01.12.2007)
Published in Archiv der Pharmazie (Weinheim) (01.12.2007)
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Oxamides as novel NR2B selective NMDA receptor antagonists
Barta-Szalai, Gizella, Borza, István, Bozó, Éva, Kiss, Csilla, Ágai, Béla, Proszenyák, Ágnes, Keserű, György M, Gere, Anikó, Kolok, Sándor, Galgóczy, Kornél, Horváth, Csilla, Farkas, Sándor, Domány, György
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
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Journal Article
Hydrogenation of a 4-benzylpyridine derivative over supported precious metal catalysts
Proszenyák, Ágnes, Ágai, Béla, Hegedűs, László, Faigl, Ferenc
Published in Applied catalysis. A, General (18.08.2004)
Published in Applied catalysis. A, General (18.08.2004)
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Discovery of S64315, a Potent and Selective Mcl‑1 Inhibitor
Szlavik, Zoltan, Csekei, Marton, Paczal, Attila, Szabo, Zoltan B, Sipos, Szabolcs, Radics, Gabor, Proszenyak, Agnes, Balint, Balazs, Murray, James, Davidson, James, Chen, Ijen, Dokurno, Pawel, Surgenor, Allan E, Daniels, Zoe Marie, Hubbard, Roderick E, Le Toumelin-Braizat, Gaëtane, Claperon, Audrey, Lysiak-Auvity, Gaëlle, Girard, Anne-Marie, Bruno, Alain, Chanrion, Maia, Colland, Frédéric, Maragno, Ana-Leticia, Demarles, Didier, Geneste, Olivier, Kotschy, Andras
Published in Journal of medicinal chemistry (25.11.2020)
Published in Journal of medicinal chemistry (25.11.2020)
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Abstract 4482: S64315 (MIK665) is a potent and selective Mcl1 inhibitor with strong antitumor activity across a diverse range of hematologic tumor models
Maragno, Ana Leticia, Mistry, Prakash, Kotschy, András, Szlavik, Zoltán, Murray, James, Davidson, James, Toumelin-Braizat, Gaëtane Le, Chanrion, Maïa, Bruno, Alain, Claperon, Audrey, Maacke, Heiko, Morris, Erick, Wang, Youzhen, Derreal, Alix, Csekei, Márton, Paczal, Attila, Szabo, Zoltán, Sipos, Szabolcs, Proszenyak, Agnes, Balint, Balázs, Surgenor, Allan, Dokurno, Pawel, Matassova, Natalia, Chen, Ijen, Lysiak-Auvity, Gaëlle, Girard, Anne-Marie, Grave, Fabienne, Colland, Frédéric, Halilovic, Ensar, Geneste, Olivier
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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Journal Article
The first synthesis of enr-agelasine F
PROSZENYAK, Agnes, BRAANDVANG, Morten, CHARNOCK, Colin, GUNDERSEN, Lise-Lotte
Published in Tetrahedron (2009)
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Published in Tetrahedron (2009)
Journal Article
Screening of agelasine D and analogs for inhibitory activity against pathogenic protozoa; identification of hits for visceral leishmaniasis and Chagas disease
Vik, Anders, Proszenyák, Agnes, Vermeersch, Marieke, Cos, Paul, Maes, Louis, Gundersen, Lise-Lotte
Published in Molecules (Basel, Switzerland) (08.01.2009)
Published in Molecules (Basel, Switzerland) (08.01.2009)
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Journal Article
The Effect of Core Replacement on S64315, a Selective MCL‑1 Inhibitor, and Its Analogues
Sipos, Szabolcs, Bálint, Balázs, Szabó, Zoltán B, Ondi, Levente, Csékei, Márton, Szlávik, Zoltán, Proszenyák, Ágnes, Murray, James B, Davidson, James, Chen, Ijen, Dokurno, Pawel, Surgenor, Allan E, Pedder, Christopher, Hubbard, Roderick E, Maragno, Ana-Leticia, Chanrion, Maia, Colland, Frederic, Geneste, Olivier, Kotschy, András
Published in ACS omega (31.08.2021)
Published in ACS omega (31.08.2021)
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NEW THIENOPYRIMIDINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
JAMES BROOKE MURRAY, MAERTON CSEKEI, SZABOLCS SIPOS, ZOLTAN SZABO, OLIVIER GENESTE, ZOLTAN SZLAVIK, JAMES EDWARD PAUL DAVIDSON, GABOR RADICS, ATTILA PACZAL, CHEN YI-JEN, FRANCOISE PERRON-SIERRA, ANDRAS KOTSCHY, BALAZS BALINT, ALAIN BRUNO, AGNES PROSZENYAK
Year of Publication 16.07.2015
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Year of Publication 16.07.2015
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NEW HYDROXYACID DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Year of Publication 28.08.2023
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Year of Publication 28.08.2023
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NEW HYDROXYACID DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Year of Publication 31.07.2023
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Year of Publication 31.07.2023
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HYDROXYACID DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Year of Publication 07.04.2022
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Year of Publication 07.04.2022
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HYDROXYACID DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Year of Publication 25.05.2021
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Year of Publication 25.05.2021
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Year of Publication 16.02.2022
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Year of Publication 16.02.2022
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NEW THIENOPYRIMIDINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Year of Publication 28.07.2021
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Year of Publication 28.07.2021
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NEW THIENOPYRIMIDINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
Balazs BALINT, James Edward Paul DAVIDSON, Marton CSEKEI, Gabor RADICS, CHEN I-Jen, Szabolcs SIPOS, Attila PACZAL, Andras KOTSCHY, Zoltan SZLAVIK, Alain BRUNO, Olivier GENESTE, Zoltan SZABO, Agnes PROSZENYAK, James Brooke MURRAY, Francoise PERRON-SIERRA
Year of Publication 30.04.2021
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Year of Publication 30.04.2021
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