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Cariprazine (RGH-188), a potent D3/D2 dopamine receptor partial agonist, binds to dopamine D3 receptors in vivo and shows antipsychotic-like and procognitive effects in rodents

Cariprazine (RGH-188), a potent D3/D2 dopamine receptor partial agonist, binds to dopamine D3 receptors in vivo and shows antipsychotic-like and procognitive effects in rodents

by GYERTYAN, Istvan, KISS, Béla, AGAI CSONGOR, Eva, DOMANY, György, TIHANYI, Károly, SZOMBATHELYI, Zsolt, SAGHY, Katalin, LASZY, Judit, SZABO, Györgyi, SZABADOS, Tamás, GEMESI, Larisza I, PASZTOR, Gabriella, ZAJER-BALAZS, Mária, KAPAS, Margit
Published in Neurochemistry international (01.11.2011)

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Journal Article

Cariprazine (RGH-188), a potent D 3/D 2 dopamine receptor partial agonist, binds to dopamine D 3 receptors in vivo and shows antipsychotic-like and procognitive effects in rodents

Cariprazine (RGH-188), a potent D 3/D 2 dopamine receptor partial agonist, binds to dopamine D 3 receptors in vivo and shows antipsychotic-like and procognitive effects in rodents

by Gyertyán, István, Kiss, Béla, Sághy, Katalin, Laszy, Judit, Szabó, Györgyi, Szabados, Tamás, Gémesi, Larisza I., Pásztor, Gabriella, Zájer-Balázs, Mária, Kapás, Margit, Csongor, Éva Ágai, Domány, György, Tihanyi, Károly, Szombathelyi, Zsolt
Published in Neurochemistry international (01.11.2011)

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Journal Article

Subnanomolar dopamine D3 receptor antagonism coupled to moderate D2 affinity results in favourable antipsychotic-like activity in rodent models: II. behavioural characterisation of RG-15

Subnanomolar dopamine D3 receptor antagonism coupled to moderate D2 affinity results in favourable antipsychotic-like activity in rodent models: II. behavioural characterisation of RG-15

by Gyertyán, István, Sághy, Katalin, Laszy, Judit, Elekes, Ottilia, Kedves, Rita, Gémesi, Larisza I., Pásztor, Gabriella, Zájer-Balázs, Mária, Kapás, Margit, Ágai Csongor, Éva, Domány, György, Kiss, Béla, Szombathelyi, Zsolt
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.11.2008)

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Journal Article

Effects of RGH-237 [ N -{4-[4-(3-Aminocarbonyl-phenyl)-piperazin-1-yl]-butyl}-4-bromo-benzamide], an Orally Active, Selective Dopamine D 3 Receptor Partial Agonist in Animal Models of Cocaine Abuse

Effects of RGH-237 [ N -{4-[4-(3-Aminocarbonyl-phenyl)-piperazin-1-yl]-butyl}-4-bromo-benzamide], an Orally Active, Selective Dopamine D 3 Receptor Partial Agonist in Animal Models of Cocaine Abuse

by Gyertyán, István, Kiss, Béla, Gál, Krisztina, Laszlovszky, István, Horváth, Attila, Gémesi, Larisza I., Sághy, Katalin, Pásztor, Gabriella, Zájer, Mária, Kapás, Margit, Csongor, Éva Ágai, Domány, György, Tihanyi, Károly, Szombathelyi, Zsolt
Published in The Journal of pharmacology and experimental therapeutics (01.03.2007)

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Journal Article

Indole-2-carboxamides as novel NR2B selective NMDA receptor antagonists

Indole-2-carboxamides as novel NR2B selective NMDA receptor antagonists

by BORZA, Istvan, KOLOK, Sandor, BIELIK, Attila, NAGY, Jozsef, FARKAS, Sandor, DOMANY, György, GERE, Aniko, AGAI-CSONGOR, Eva, AGAI, Béla, TARKANYI, Gabor, HORVATH, Csilla, BARTA-SZALAI, Gizella, BOZO, Eva, KISS, Csilla
Published in Bioorganic & medicinal chemistry letters (03.11.2003)

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Journal Article

ChemInform Abstract: Discovery of Cariprazine (RGH-188): A Novel Antipsychotic Acting on Dopamine D3/D2 Receptors

ChemInform Abstract: Discovery of Cariprazine (RGH-188): A Novel Antipsychotic Acting on Dopamine D3/D2 Receptors

by Agai‐Csongor, Eva, et al, et al
Published in ChemInform (25.09.2012)

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Journal Article

Cariprazine (RGH-188), a Dopamine D 3 Receptor-Preferring, D 3 /D 2 Dopamine Receptor Antagonist–Partial Agonist Antipsychotic Candidate: In Vitro and Neurochemical Profile

by Kiss, Béla, Horváth, Attila, Némethy, Zsolt, Schmidt, Éva, Laszlovszky, István, Bugovics, Gyula, Fazekas, Károly, Hornok, Katalin, Orosz, Szabolcs, Gyertyán, István, Ágai-Csongor, Éva, Domány, György, Tihanyi, Károly, Adham, Nika, Szombathelyi, Zsolt
Published in The Journal of pharmacology and experimental therapeutics (01.04.2010)

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Journal Article

Multiple Fragment Docking and Linking in Primary and Secondary Pockets of Dopamine Receptors

Multiple Fragment Docking and Linking in Primary and Secondary Pockets of Dopamine Receptors

by Vass, Márton, Ágai-Csongor, Éva, Horti, Ferenc, Keserű, György M
Published in ACS medicinal chemistry letters (11.09.2014)

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Journal Article

Design of novel multiple-acting ligands towards SERT and 5-HT sub(2C) receptors

Design of novel multiple-acting ligands towards SERT and 5-HT sub(2C) receptors

by Elias, Oliver, Agai-Csongor, Eva, Domany, Gyorgy, Keserue, Gyorgy Miklos, Gere, Aniko, Kiss, Bela, Hellinger, Eva, Vastag, Monika, Gyertyan, Istvan
Published in Bioorganic & medicinal chemistry letters (01.05.2014)

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Journal Article

Design of novel multiple-acting ligands towards SERT and 5-HT2C receptors

Design of novel multiple-acting ligands towards SERT and 5-HT2C receptors

by Éliás, Olivér, Ágai-Csongor, Éva, Domány, György, Keserű, György Miklós, Gere, Anikó, Kiss, Béla, Hellinger, Éva, Vastag, Mónika, Gyertyán, István
Published in Bioorganic & medicinal chemistry letters (01.05.2014)

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Journal Article

Sensitive LC–MS/MS methods for the quantification of RGH-188 and its active metabolites, desmethyl- and didesmethyl-RGH-188 in human plasma and urine

Sensitive LC–MS/MS methods for the quantification of RGH-188 and its active metabolites, desmethyl- and didesmethyl-RGH-188 in human plasma and urine

by PASZTOR MEZAROS, Gabriella, AGAI-CSONGOR, Eva, KAPAS, Margit
Published in Journal of pharmaceutical and biomedical analysis (29.09.2008)

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Journal Article Conference Proceeding

Subnanomolar dopamine D3 receptor antagonism coupled to moderate D2 affinity results in favourable antipsychotic-like activity in rodent models: I. neurochemical characterisation of RG-15

Subnanomolar dopamine D3 receptor antagonism coupled to moderate D2 affinity results in favourable antipsychotic-like activity in rodent models: I. neurochemical characterisation of RG-15

by Kiss, Béla, Laszlovszky, István, Horváth, Attila, Némethy, Zsolt, Schmidt, Éva, Bugovics, Gyula, Fazekas, Károly, Gyertyán, István, Ágai-Csongor, Éva, Domány, György, Szombathelyi, Zsolt
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.11.2008)

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Journal Article

ChemInform Abstract: Discovery of Cariprazine (RGH‐188): A Novel Antipsychotic Acting on Dopamine D 3 /D 2 Receptors

ChemInform Abstract: Discovery of Cariprazine (RGH‐188): A Novel Antipsychotic Acting on Dopamine D 3 /D 2 Receptors

by Agai‐Csongor, Eva
Published in ChemInform (25.09.2012)

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Journal Article

Discovery of cariprazine (RGH-188): A novel antipsychotic acting on dopamine D3/D2 receptors

Discovery of cariprazine (RGH-188): A novel antipsychotic acting on dopamine D3/D2 receptors

by Ágai-Csongor, Éva, Domány, György, Nógrádi, Katalin, Galambos, János, Vágó, István, Keserű, György Miklós, Greiner, István, Laszlovszky, István, Gere, Anikó, Schmidt, Éva, Kiss, Béla, Vastag, Mónika, Tihanyi, Károly, Sághy, Katalin, Laszy, Judit, Gyertyán, István, Zájer-Balázs, Mária, Gémesi, Larisza, Kapás, Margit, Szombathelyi, Zsolt
Published in Bioorganic & medicinal chemistry letters (15.05.2012)

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Journal Article

Cariprazine (RGH-188), a dopamine D(3) receptor-preferring, D(3)/D(2) dopamine receptor antagonist-partial agonist antipsychotic candidate: in vitro and neurochemical profile

by Kiss, Béla, Horváth, Attila, Némethy, Zsolt, Schmidt, Eva, Laszlovszky, István, Bugovics, Gyula, Fazekas, Károly, Hornok, Katalin, Orosz, Szabolcs, Gyertyán, István, Agai-Csongor, Eva, Domány, György, Tihanyi, Károly, Adham, Nika, Szombathelyi, Zsolt
Published in The Journal of pharmacology and experimental therapeutics (01.04.2010)

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Journal Article

Novel sulfonamides having dual dopamine D2 and D3 receptor affinity show in vivo antipsychotic efficacy with beneficial cognitive and EPS profile

by Ágai-Csongor, Éva, Nógrádi, Katalin, Galambos, János, Vágó, István, Bielik, Attila, Magdó, Ildikó, Ignácz-Szendrei, Györgyi, Keserű, György Miklós, Greiner, István, Laszlovszky, István, Béla Kiss, Éva Schmidt, Judit Laszy, Katalin Sághy, Gyertyán, István, Zájer-Balázs, Mária, Gémesi, Larisza, Domány, György
Published in Bioorganic & medicinal chemistry letters (01.10.2007)

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Journal Article

PROCEDIMENTO PER LA PREPARAZIONE DI N-METIL-3-FENIL-3(4-TRIFLUORORO METIL)FENOSSI) PROPILAMMINA E DI SUOI SALI ACIDI DI ADDIZIONE

PROCEDIMENTO PER LA PREPARAZIONE DI N-METIL-3-FENIL-3(4-TRIFLUORORO METIL)FENOSSI) PROPILAMMINA E DI SUOI SALI ACIDI DI ADDIZIONE

by UJVARI BEATRIX, CSONGOR AGAI EVA, GAL VARGA GIZELLA, HARSANYI KALMAN, TRISCHLER ARACS ZSUSANNA, DREXLER FERENC
Year of Publication 27.12.1993

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Patent

Effects of RGH-237 [N-{4-[4-(3-Aminocarbonyl-phenyl)-piperazin-1-yl]-butyl}-4-bromo-benzamide], an Orally Active, Selective Dopamine D3 Receptor Partial Agonist in Animal Models of Cocaine Abuse

Effects of RGH-237 [N-{4-[4-(3-Aminocarbonyl-phenyl)-piperazin-1-yl]-butyl}-4-bromo-benzamide], an Orally Active, Selective Dopamine D3 Receptor Partial Agonist in Animal Models of Cocaine Abuse

by IstvÃ¡n GyertyÃ¡n, BÃ©la Kiss, Krisztina GÃ¡l, IstvÃ¡n Laszlovszky, Attila HorvÃ¡th, Larisza I. GÃ©mesi, Katalin SÃ¡ghy, Gabriella PÃ¡sztor, MÃ¡ria ZÃ¡jer, Margit KapÃ¡s, Ãva Ãgai Csongor, GyÃ¶rgy DomÃ¡ny, KÃ¡roly Tihanyi, Zsolt Szombathelyi
Published in The Journal of pharmacology and experimental therapeutics (01.03.2007)

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Journal Article

Process for the preparation of N-methyl-3-phenyl-3-[4-(trifluoromethyl)phenoxy]propylamine and acid addition salts thereof

Process for the preparation of N-methyl-3-phenyl-3-[4-(trifluoromethyl)phenoxy]propylamine and acid addition salts thereof

by UJVARI BEATRIX, KALMAN HARSANYI DR, GIZELLA VARGA - GAL, AGAI CSONGOR EVA, TRISCHLER ARACS ZSUZSANNA, DREXLER FERENC
Year of Publication 28.02.1994

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Patent

Process for the preparation of piperazine derivatives

Process for the preparation of piperazine derivatives

by CSEHI, ATTILA, GIZUR, TIBOR, HARSANYI, KALMAN, DEMETER-SZABO, ANIKU, VAJDA, EVA, TRISCHLER, FERENC, AGAI-CSONGOR, EVA, SZABO-KOMLOSI, GYOERGYI
Year of Publication 06.05.1992

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Patent