Discovery of Dabrafenib: A Selective Inhibitor of Raf Kinases with Antitumor Activity against B‑Raf-Driven Tumors
Rheault, Tara R., Stellwagen, John C., Adjabeng, George M., Hornberger, Keith R., Petrov, Kimberly G., Waterson, Alex G., Dickerson, Scott H., Mook, Robert A., Laquerre, Sylvie G., King, Alastair J., Rossanese, Olivia W., Arnone, Marc R., Smitheman, Kimberly N., Kane-Carson, Laurie S., Han, Chao, Moorthy, Ganesh S., Moss, Katherine G., Uehling, David E.
Published in ACS medicinal chemistry letters (14.03.2013)
Published in ACS medicinal chemistry letters (14.03.2013)
Get full text
Journal Article
Room-Temperature Pd-Catalyzed Amidation of Aryl Bromides Using tert-Butyl Carbamate
Bhagwanth, Swapna, Waterson, Alex G, Adjabeng, George M, Hornberger, Keith R
Published in Journal of organic chemistry (19.06.2009)
Published in Journal of organic chemistry (19.06.2009)
Get full text
Journal Article
Phosphaadamantanes as Ligands for Palladium Catalyzed Cross-Coupling Chemistry: Library Synthesis, Characterization, and Screening in the Suzuki Coupling of Alkyl Halides and Tosylates Containing β-Hydrogens with Boronic Acids and Alkylboranes
Brenstrum, Tim, Gerristma, David A, Adjabeng, George M, Frampton, Christopher S, Britten, James, Robertson, Alan J, McNulty, James, Capretta, Alfredo
Published in Journal of organic chemistry (29.10.2004)
Published in Journal of organic chemistry (29.10.2004)
Get full text
Journal Article
Novel Class of Tertiary Phosphine Ligands Based on a Phospha-adamantane Framework and Use in the Suzuki Cross-Coupling Reactions of Aryl Halides under Mild Conditions
Adjabeng, George, Brenstrum, Tim, Wilson, Jeffrey, Frampton, Christopher, Robertson, Al, Hillhouse, John, McNulty, James, Capretta, Alfredo
Published in Organic letters (20.03.2003)
Published in Organic letters (20.03.2003)
Get full text
Journal Article
Development of potent B-RafV600E inhibitors containing an arylsulfonamide headgroup
STELLWAGEN, John C, ADJABENG, George M, ROMINGER, Cynthia M, ROSSANESE, Olivia W, SMITHEMAN, Kimberly N, WATERSON, Alex G, UEHLING, David E, ARNONE, Marc R, DICKERSON, Scott H, CHAO HAN, HORNBERGER, Keith R, KING, Alastair J, MOOK, Robert A, PETROV, Kimberly G, RHEAULT, Tara R
Published in Bioorganic & medicinal chemistry letters (01.08.2011)
Published in Bioorganic & medicinal chemistry letters (01.08.2011)
Get full text
Journal Article
Abstract B88: A selective Raf kinase inhibitor induces cell death and tumor regression of human cancer cell lines encoding B-RafV600E mutation
Laquerre, Sylvie, Arnone, Marc, Moss, Katherine, Yang, Jingsong, Fisher, Kelly, Kane-Carson, Laurie S., Smitheman, Kimberly, Ward, Jessica, Heidrich, Bradley, Rheault, Tara, Adjabeng, George, Hornberger, Keith, Stellwagen, John, Waterson, Alex, Han, Chao, Mook, Robert A., Uehling, David, King, Alastair J.
Published in Molecular cancer therapeutics (10.12.2009)
Published in Molecular cancer therapeutics (10.12.2009)
Get full text
Journal Article
Rhodium Phosphinates as Catalysts for Metal-Stabilized Carbene Chemistry: Synthesis, Characterization, and Application of Rh2(O2PMe2)4
Adjabeng, George M, Gerritsma, David A, Bhanabhai, Hitesh, Frampton, Christopher S, Capretta, Alfredo
Published in Organometallics (02.01.2006)
Published in Organometallics (02.01.2006)
Get full text
Journal Article
GSK2818713, a Novel Biphenylene Scaffold-Based Hepatitis C NS5A Replication Complex Inhibitor with Broad Genotype Coverage
Kazmierski, Wieslaw M, Baskaran, Sam, Walker, Jill T, Miriyala, Nagaraju, Meesala, Ramu, Beesu, Mallesh, Adjabeng, George, Grimes, Richard M, Hamatake, Robert, Leivers, Martin R, Crosby, Renae, Xia, Bing, Remlinger, Katja
Published in Journal of medicinal chemistry (23.04.2020)
Published in Journal of medicinal chemistry (23.04.2020)
Get full text
Journal Article
Palladium Complexes of 1,3,5,7-Tetramethyl-2,4,8-trioxa-6-phenyl-6-phosphaadamantane: Synthesis, Crystal Structure and Use in the Suzuki and Sonogashira Reactions and the α-Arylation of Ketones
Adjabeng, George, Brenstrum, Tim, Frampton, Christopher S, Robertson, Al J, Hillhouse, John, McNulty, James, Capretta, Alfredo
Published in Journal of organic chemistry (23.07.2004)
Published in Journal of organic chemistry (23.07.2004)
Get full text
Journal Article
A mild, one-pot synthesis of disubstituted benzimidazoles from 2-nitroanilines
Hornberger, Keith R., Adjabeng, George M., Dickson, Hamilton D., Davis-Ward, Ronda G.
Published in Tetrahedron letters (24.07.2006)
Published in Tetrahedron letters (24.07.2006)
Get full text
Journal Article