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Novel Indolylindazolylmaleimides as Inhibitors of Protein Kinase C-β: Synthesis, Biological Activity, and Cardiovascular Safety
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Design, Synthesis, and Biological Characterization of a Peptide-Mimetic Antagonist for a Tethered-Ligand Receptor
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Published in Proceedings of the National Academy of Sciences - PNAS (26.10.1999)
Published in Proceedings of the National Academy of Sciences - PNAS (26.10.1999)
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Administration of a Potent Antagonist of Protease-Activated Receptor-1 (PAR-1) Attenuates Vascular Restenosis Following Balloon Angioplasty in Rats
Andrade-Gordon, P, Derian, C K, Maryanoff, B E, Zhang, H C, Addo, M F, Cheung Wm, Damiano, B P, D'Andrea, M R, Darrow, A L, de Garavilla, L, Eckardt, A J, Giardino, E C, Haertlein, B J, McComsey, D F
Published in The Journal of pharmacology and experimental therapeutics (01.07.2001)
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Published in The Journal of pharmacology and experimental therapeutics (01.07.2001)
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Macrocyclic bisindolylmaleimides as inhibitors of protein kinase C and glycogen synthase kinase-3
Zhang, Han-Cheng, White, Kimberly B., Ye, Hong, McComsey, David F., Derian, Claudia K., Addo, Michael F., Andrade-Gordon, Patricia, Eckardt, Annette J., Conway, Bruce R., Westover, Lori, Xu, Jun Z., Look, Richard, Demarest, Keith T., Emanuel, Stuart, Maryanoff, Bruce E.
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
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Discovery and Optimization of a Novel Series of Thrombin Receptor (PAR-1) Antagonists: Potent, Selective Peptide Mimetics Based on Indole and Indazole Templates
Zhang, Han-Cheng, Derian, Claudia K, Andrade-Gordon, Patricia, Hoekstra, William J, McComsey, David F, White, Kimberly B, Poulter, Brenda L, Addo, Michael F, Cheung, Wai-Man, Damiano, Bruce P, Oksenberg, Donna, Reynolds, Elwood E, Pandey, Anjali, Scarborough, Robert M, Maryanoff, Bruce E
Published in Journal of medicinal chemistry (29.03.2001)
Published in Journal of medicinal chemistry (29.03.2001)
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1,2,4-Triazolo[3,4- a]pyridine as a novel, constrained template for fibrinogen receptor (GPIIb/IIIa) antagonists
Lawson, Edward C, Hoekstra, William J, Addo, Michael F, Andrade-Gordon, Patricia, Damiano, Bruce P, Kauffman, Jack A, Mitchell, John A, Maryanoff, Bruce E
Published in Bioorganic & medicinal chemistry letters (08.10.2001)
Published in Bioorganic & medicinal chemistry letters (08.10.2001)
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Zhang, Han-Cheng, White, Kimberly B., McComsey, David F., Addo, Michael F., Andrade-Gordon, Patricia, Derian, Claudia K., Oksenberg, Donna, Maryanoff, Bruce E.
Published in Bioorganic & medicinal chemistry letters (07.07.2003)
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Thrombin receptor (PAR-1) antagonists. Solid-Phase synthesis of indole-Based peptide mimetics by anchoring to a secondary amide
Zhang, Han-Cheng, McComsey, David F, White, Kimberly B, Addo, Michael F, Andrade-Gordon, Patricia, Derian, Claudia K, Oksenberg, Donna, Maryanoff, Bruce E
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
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Thrombin receptor-activating peptides (TRAPs): Investigation of bioactive conformations via structure–activity, spectroscopic, and computational studies
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Published in Bioorganic & medicinal chemistry (01.11.1999)
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Novel indolylindazolylmaleimides as inhibitors of protein kinase C- : Synthesis, biological activity, and cardiovascular safety
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Published in Journal of medicinal chemistry (2005)
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Heterocycle-peptide hybrid compounds. Aminotriazole-containing agonists of the thrombin receptor (PAR-1)
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Published in Bioorganic & medicinal chemistry letters (17.05.1999)
Published in Bioorganic & medicinal chemistry letters (17.05.1999)
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Macrocyclic bisindolylmaleimides as inhibitors of protein kinase C and glycogen synthase kinase-3: Recent advances in the design of kinase inhibitors as novel therapeutic agents
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Published in Bioorganic & medicinal chemistry letters (2003)
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Published in Bioorganic & medicinal chemistry letters (2003)
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Thrombin receptor (PAR-1) antagonists. Heterocycle-based peptidomimetics of the SFLLR agonist motif
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Novel thieno[2,3- b]- and [3,4- b]pyrans as potassium channel openers. Thiophene systems—XVII
Press, Jeffery B., McNally, James J., Sanfilippo, Pauline J., Addo, Michael F., Loughney, Deborah, Giardino, Edward, Katz, Laurence B., Falotico, Robert, Haertlein, Barbara J.
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Published in Bioorganic & medicinal chemistry (01.12.1993)
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Guinea pig proteinase-activated receptor 4 and its activating peptide
ADDO MICHAEL F, DERIAN CLAUDIA K, DARROW ANDREW L, ANDRADE-GORDON PATRICIA
Year of Publication 09.10.2008
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Year of Publication 09.10.2008
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Guinea pig proteinase-activated receptor 4 and its activating peptide
ADDO MICHAEL F, DERIAN CLAUDIA K, DARROW ANDREW L, ANDRADE-GORDON PATRICIA
Year of Publication 20.02.2007
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Year of Publication 20.02.2007
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Guinea pig proteinase-activated receptor 4 and its activating peptide
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Year of Publication 20.02.2007
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Year of Publication 20.02.2007
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