An improved high yield total synthesis and cytotoxicity study of the marine alkaloid neoamphimedine: an ATP-competitive inhibitor of topoisomerase IIα and potent anticancer agent
Li, Linfeng, Abraham, Adedoyin D, Zhou, Qiong, Ali, Hadi, O'Brien, Jeremy V, Hamill, Brayden D, Arcaroli, John J, Messersmith, Wells A, LaBarbera, Daniel V
Published in Marine drugs (19.09.2014)
Published in Marine drugs (19.09.2014)
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Journal Article
Neoamphimedine circumvents metnase-enhanced DNA topoisomerase IIα activity through ATP-competitive inhibition
Ponder, Jessica, Yoo, Byong Hoon, Abraham, Adedoyin D, Li, Qun, Ashley, Amanda K, Amerin, Courtney L, Zhou, Qiong, Reid, Brian G, Reigan, Philip, Hromas, Robert, Nickoloff, Jac A, LaBarbera, Daniel V
Published in Marine drugs (2011)
Published in Marine drugs (2011)
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Journal Article
Isolating and targeting the real-time plasticity and malignant properties of epithelial-mesenchymal transition in cancer
Esquer, Hector, Zhou, Qiong, Nemkov, Travis, Abraham, Adedoyin D, Rinaldetti, Sébastien, Chen, Yu-Chi, Zhang, Xiaohu, Orman, Michael V, D'Alessandro, Angelo, Ferrer, Marc, Messersmith, Wells A, LaBarbera, Daniel V
Published in Oncogene (22.04.2021)
Published in Oncogene (22.04.2021)
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Journal Article
Design, Synthesis, and Biological Evaluation of the First Inhibitors of Oncogenic CHD1L
Prigaro, Brett J, Esquer, Hector, Zhou, Qiong, Pike, Laura A, Awolade, Paul, Lai, Xin-He, Abraham, Adedoyin D, Abbott, Joshua M, Matter, Brock, Kompella, Uday B, Messersmith, Wells A, Gustafson, Daniel L, LaBarbera, Daniel V
Published in Journal of medicinal chemistry (10.03.2022)
Published in Journal of medicinal chemistry (10.03.2022)
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Journal Article
First-in-Class Inhibitors of Oncogenic CHD1L with Preclinical Activity against Colorectal Cancer
Abbott, Joshua M, Zhou, Qiong, Esquer, Hector, Pike, Laura, Broneske, Travis P, Rinaldetti, Sébastien, Abraham, Adedoyin D, Ramirez, Dominique A, Lunghofer, Paul J, Pitts, Todd M, Regan, Daniel P, Tan, Aik Choon, Gustafson, Daniel L, Messersmith, Wells A, LaBarbera, Daniel V
Published in Molecular cancer therapeutics (01.08.2020)
Published in Molecular cancer therapeutics (01.08.2020)
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Journal Article
Advanced High-Content-Screening Applications of Clonogenicity in Cancer
Esquer, Hector, Zhou, Qiong, Abraham, Adedoyin D., LaBarbera, Daniel V.
Published in SLAS discovery (01.08.2020)
Published in SLAS discovery (01.08.2020)
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Journal Article
Design of an Amide N‑Glycoside Derivative of β‑Glucogallin: A Stable, Potent, and Specific Inhibitor of Aldose Reductase
Li, Linfeng, Chang, Kun-Che, Zhou, Yaming, Shieh, Biehuoy, Ponder, Jessica, Abraham, Adedoyin D, Ali, Hadi, Snow, Anson, Petrash, J. Mark, LaBarbera, Daniel V
Published in Journal of medicinal chemistry (09.01.2014)
Published in Journal of medicinal chemistry (09.01.2014)
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Journal Article
Drug Design Targeting T‑Cell Factor-Driven Epithelial–Mesenchymal Transition as a Therapeutic Strategy for Colorectal Cancer
Abraham, Adedoyin D, Esquer, Hector, Zhou, Qiong, Tomlinson, Nicholas, Hamill, Brayden D, Abbott, Joshua M, Li, Linfeng, Pike, Laura A, Rinaldetti, Sébastien, Ramirez, Dominique A, Lunghofer, Paul J, Gomez, Jose D, Schaack, Jerome, Nemkov, Travis, D’Alessandro, Angelo, Hansen, Kirk C, Gustafson, Daniel L, Messersmith, Wells A, LaBarbera, Daniel V
Published in Journal of medicinal chemistry (27.11.2019)
Published in Journal of medicinal chemistry (27.11.2019)
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Journal Article
Tumor organoids for drug discovery and personalized medicine
Zhou, Qiong, Li, Linfeng, Abraham, Adedoyin D, LaBarbera, Daniel V
Published in The Journal of nuclear medicine (1978) (01.02.2018)
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Published in The Journal of nuclear medicine (1978) (01.02.2018)
Journal Article
An Improved High Yield Total Synthesis and Cytotoxicity Study of the Marine Alkaloid Neoamphimedine: An ATP-Competitive Inhibitor of Topoisomerase II[alpha] and Potent Anticancer Agent
Li, Linfeng, Abraham, Adedoyin D, Zhou, Qiong, Ali, Hadi, O'Brien, Jeremy V, Hamill, Brayden D, Arcaroli, John J, Messersmith, Wells A, LaBarbera, Daniel V
Published in Marine drugs (01.09.2014)
Published in Marine drugs (01.09.2014)
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Journal Article
Neoamphimedine Circumvents Metnase-Enhanced DNA Topoisomerase II[alpha] Activity Through ATP-Competitive Inhibition
Ponder, Jessica, Yoo, Byong Hoon, Abraham, Adedoyin D, Li, Qun, Ashley, Amanda K, Amerin, Courtney L, Zhou, Qiong, Reid, Brian G, Reigan, Philip, Hromas, Robert, Nickoloff, Jac A, LaBarbera, Daniel V
Published in Marine drugs (01.11.2011)
Published in Marine drugs (01.11.2011)
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Journal Article
Neoamphimedine Circumvents Metnase-Enhanced DNA Topoisomerase IIα Activity Through ATP-Competitive Inhibition
Jessica Ponder, Byong Hoon Yoo, Adedoyin D. Abraham, Qun Li, Amanda K. Ashley, Courtney L. Amerin, Qiong Zhou, Brian G. Reid, Philip Reigan, Robert Hromas, Jac A. Nickoloff, Daniel V. LaBarbera
Year of Publication 2011
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Year of Publication 2011
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