Structure-Activity Studies on the Corticotropin Releasing Factor Antagonist Astressin, leading to a Minimal Sequence necessary for Antagonistic Activity
Rijkers, Dirk T.S, Kruijtzer, John A.W, van Oostenbrugge, Marja, Ronken, Eric, den Hartog, Jack A.J, Liskamp, Rob M.J
Published in Chembiochem : a European journal of chemical biology (05.03.2004)
Published in Chembiochem : a European journal of chemical biology (05.03.2004)
Get full text
Journal Article
Design and Synthesis of an orally active GPIIb/IIIa antagonist based on a phenylpiperazine scaffold
van Maarseveen, Jan H, den Hartog, Jack A.J, Tipker, Koos, Reinders, Jan-Hendrik, Brakkee, Joost, Schön, Uwe, Kehrbach, Wolfgang, Kruse, Chris G
Published in Bioorganic & medicinal chemistry letters (16.06.1998)
Published in Bioorganic & medicinal chemistry letters (16.06.1998)
Get full text
Journal Article
A straightforward synthesis of 1,3-dichloro-5,8-dihydroisoquinoline by consecutive Stille cross-coupling and metathesis reactions
van den Hoogenband, Adri, den Hartog, Jack A.J., Faber-Hilhorst, Nancy, Lange, Jos H.M., Terpstra, Jan Willem
Published in Tetrahedron letters (02.09.2009)
Published in Tetrahedron letters (02.09.2009)
Get full text
Journal Article
Synthesis and biological activity of N-terminal lipidated and/or fluorescently labeled conjugates of astressin as corticotropin releasing factor antagonists
Rijkers, Dirk T.S., den Hartog, Jack A.J., Liskamp, Rob M.J.
Published in Bioorganic & medicinal chemistry (01.10.2004)
Published in Bioorganic & medicinal chemistry (01.10.2004)
Get full text
Journal Article
An optimized solid phase synthesis strategy- including on-resin lactamization-of astressin, its retro-, inverso-, and retro-inverso isomers as corticotropin releasing factor antagonists
Rijkers, Dirk T. S., den Hartog, Jack A. J., Liskamp, Rob M. J.
Published in Biopolymers (01.02.2002)
Published in Biopolymers (01.02.2002)
Get full text
Journal Article
derivados heterocíclicos fundidos como moduladores s1p
HEIN K.A.C. COOLEN, JACOBUS A.J. DEN HARTOG, WOUTER I. IWEMA BAKKER, MARIA J.P. VAN DONGEN, PIETER SMID, LEONARDUS A.J.M. SLIEDREGT
Year of Publication 24.05.2016
Get full text
Year of Publication 24.05.2016
Patent
FUSED HETEROCYCLIC DERIVATIVES AS S1P MODULATORS
IWEMA BAKKER, WOUTER I, HOBSON, ADRIAN D, COOLEN, HEIN K.A.C, VAN DONGEN, MARIA J.P, DEN HARTOG, JACOBUS A.J, SLIEDREGT, LEONARDUS A.J.M, SMID, PIETER
Year of Publication 11.06.2019
Get full text
Year of Publication 11.06.2019
Patent
Two novel syntheses of the histamine H3 antagonist thioperamide
Lange, Jos H.M., Wals, Henri C., den Hoogenband, Adri van, de Kuilen, Aalt van, den Hartog, Jack A.J.
Published in Tetrahedron (01.11.1995)
Published in Tetrahedron (01.11.1995)
Get full text
Journal Article
DERIVADOS HETEROCICLICOS FUSIONADOS COMO MODULADORES S1P
HEIN COOLEN, LEONARDUS, A.J.M. SLIEDREGT, WOUTER, 1 IWEMA BAKKER, MARIA J.P. VAN DONGEN, PIETER SMID, JACOBUS, A.J. DEN HARTOG
Year of Publication 15.10.2013
Get full text
Year of Publication 15.10.2013
Patent
FUSED HETEROCYCLIC DERIVATIVES AS S1P MODULATORS
IWEMA BAKKER, Wouter, I, COOLEN, Hein, K.A.C, DEN HARTOG, Jacobus, A.J, HOBSON, Adrian D, VAN DONGEN, Maria, J.P, SMID, Pieter, SLIEDREGT, Leonardus, A.J.M
Year of Publication 20.09.2017
Get full text
Year of Publication 20.09.2017
Patent
1,3,5-TRIAZINE DERIVATIVES AS LIGANDS FOR HUMAN ADENOSINE-A3 RECEPTORS
JACOBUS A.J. DEN HARTOG, GUUSTAAF J.M. VAN SCHARRENBURG, GARY R GUSTAFSON, MARIA L PRAS-RAVES, JAN H REINDERS
Year of Publication 30.06.2005
Get full text
Year of Publication 30.06.2005
Patent
FUSED HETEROCYCLIC DERIVATIVES AS S1P MODULATORS
VAN DONGEN, MARIA, J.P, DEN HARTOG, JACOBUS, A.J, IWEMA BAKKER, WOUTER, I, COOLEN, HEIN, K.A.C, SLIEDREGT, LEONARDUS, A.J.M, ADRIAN D HOBSON, SMID, PIETER
Year of Publication 14.04.2017
Get full text
Year of Publication 14.04.2017
Patent
Two novel syntheses of the histamine H 3 antagonist thioperamide
Lange, Jos H.M., Wals, Henri C., den Hoogenband, Adri van, de Kuilen, Aalt van, den Hartog, Jack A.J.
Published in Tetrahedron (1995)
Published in Tetrahedron (1995)
Get full text
Journal Article