Discovery of Novel Human Constitutive Androstane Receptor Agonists with the Imidazo[1,2‑a]pyridine Structure
Mejdrová, Ivana, Dušek, Jan, Škach, Kryštof, Stefela, Alžbeta, Skoda, Josef, Chalupský, Karel, Dohnalová, Klára, Pavkova, Ivona, Kronenberger, Thales, Rashidian, Azam, Smutná, Lucie, Duchoslav, Vojtěch, Smutny, Tomas, Pávek, Petr, Nencka, Radim
Published in Journal of medicinal chemistry (23.02.2023)
Published in Journal of medicinal chemistry (23.02.2023)
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Inhibition of FLT3-ITD Kinase in Acute Myeloid Leukemia by New Imidazo[1,2‑b]pyridazine Derivatives Identified by Scaffold Hopping
Břehová, Petra, Řezníčková, Eva, Škach, Kryštof, Jorda, Radek, Dejmek, Milan, Vojáčková, Veronika, Šála, Michal, Kovalová, Markéta, Dračínský, Martin, Dolníková, Alexandra, Strmeň, Timotej, Kinnertová, Monika, Chalupský, Karel, Dvořáková, Alexandra, Gucký, Tomáš, Mertlíková Kaiserová, Helena, Klener, Pavel, Nencka, Radim, Kryštof, Vladimír
Published in Journal of medicinal chemistry (24.08.2023)
Published in Journal of medicinal chemistry (24.08.2023)
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PF74 and Its Novel Derivatives Stabilize Hexameric Lattice of HIV-1 Mature-Like Particles
Dostálková, Alžběta, Škach, Kryštof, Kaufman, Filip, Křížová, Ivana, Hadravová, Romana, Flegel, Martin, Ruml, Tomáš, Hrabal, Richard, Rumlová, Michaela
Published in Molecules (Basel, Switzerland) (20.04.2020)
Published in Molecules (Basel, Switzerland) (20.04.2020)
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Exploring positions 6 and 7 of a quinazoline-based scaffold leads to changes in selectivity and potency towards RIPK2/3 kinases
Misehe, Mbilo, Matoušová, Marika, Dvořáková, Alexandra, Hercík, Kamil, Škach, Kryštof, Chalupská, Dominika, Dejmek, Milan, Šála, Michal, Hájek, Miroslav, Boura, Evzen, Mertlíková-Kaiserová, Helena, Nencka, Radim
Published in European journal of medicinal chemistry (15.11.2023)
Published in European journal of medicinal chemistry (15.11.2023)
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A simple, high-throughput stabilization assay to test HIV-1 uncoating inhibitors
Dostálková, Alžběta, Hadravová, Romana, Kaufman, Filip, Křížová, Ivana, Škach, Kryštof, Flegel, Martin, Hrabal, Richard, Ruml, Tomáš, Rumlová, Michaela
Published in Scientific reports (19.11.2019)
Published in Scientific reports (19.11.2019)
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Structure–activity relationship study of small-molecule inhibitor of Atg12-Atg3 protein–protein interaction
Skach, Krystof, Boserle, Jiri, Nuta, Gal Chaim, Břehová, Petra, Bialik, Shani, Carvalho, Silvia, Kozer, Noga, Barr, Haim, Chaloupecká, Ema, Kimchi, Adi, Nencka, Radim
Published in Bioorganic & medicinal chemistry letters (01.11.2024)
Published in Bioorganic & medicinal chemistry letters (01.11.2024)
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INHIBITORS OF AUTOPHAGY-RELATED PROTEIN-PROTEIN INTERACTIONS
NUTA, Chaim Gal, NENCKA, Radim, BREHOVA, Petra, GILAD, Yuval, SKACH, Krystof, KIMCHI, Adi, BOSERLE, Jiri
Year of Publication 06.07.2023
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Year of Publication 06.07.2023
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