Discovery of a chemical probe for PRDM9
Allali-Hassani, Abdellah, Szewczyk, Magdalena M., Ivanochko, Danton, Organ, Shawna L., Bok, Jabez, Ho, Jessica Sook Yuin, Gay, Florence P. H., Li, Fengling, Blazer, Levi, Eram, Mohammad S., Halabelian, Levon, Dilworth, David, Luciani, Genna M., Lima-Fernandes, Evelyne, Wu, Qin, Loppnau, Peter, Palmer, Nathan, Talib, S. Zakiah A., Brown, Peter J., Schapira, Matthieu, Kaldis, Philipp, O’Hagan, Ronan C., Guccione, Ernesto, Barsyte-Lovejoy, Dalia, Arrowsmith, Cheryl H., Sanders, John M., Kattar, Solomon D., Bennett, D. Jonathan, Nicholson, Benjamin, Vedadi, Masoud
Published in Nature communications (17.12.2019)
Published in Nature communications (17.12.2019)
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Journal Article
Angiogenesis in Skeletal Muscle Precede Improvements in Peak Oxygen Uptake in Peripheral Artery Disease Patients
Duscha, Brian D, Robbins, Jennifer L, Jones, William S, Kraus, William E, Lye, R John, Sanders, John M, Allen, Jason D, Regensteiner, Judith G, Hiatt, William R, Annex, Brian H
Published in Arteriosclerosis, thrombosis, and vascular biology (01.11.2011)
Published in Arteriosclerosis, thrombosis, and vascular biology (01.11.2011)
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Journal Article
Molecular Imaging of Endothelial Vascular Cell Adhesion Molecule-1 Expression and Inflammatory Cell Recruitment During Vasculogenesis and Ischemia-Mediated Arteriogenesis
BEHM, Carolyn Z, KAUFMANN, Beat A, CARR, Chad, LANKFORD, Miles, SANDERS, John M, ROSE, C. Edward, KAUL, Sanjiv, LINDNER, Jonathan R
Published in Circulation (New York, N.Y.) (03.06.2008)
Published in Circulation (New York, N.Y.) (03.06.2008)
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Journal Article
Maximizing Diversity from a Kinase Screen: Identification of Novel and Selective pan-Trk Inhibitors for Chronic Pain
Stachel, Shawn J, Sanders, John M, Henze, Darrell A, Rudd, Mike T, Su, Hua-Poo, Li, Yiwei, Nanda, Kausik K, Egbertson, Melissa S, Manley, Peter J, Jones, Kristen L. G, Brnardic, Edward J, Green, Ahren, Grobler, Jay A, Hanney, Barbara, Leitl, Michael, Lai, Ming-Tain, Munshi, Vandna, Murphy, Dennis, Rickert, Keith, Riley, Daniel, Krasowska-Zoladek, Alicja, Daley, Christopher, Zuck, Paul, Kane, Stephanie A, Bilodeau, Mark T
Published in Journal of medicinal chemistry (10.07.2014)
Published in Journal of medicinal chemistry (10.07.2014)
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Journal Article
NF-E2-related factor 2 regulates the stress response to UVA-1-oxidized phospholipids in skin cells
Gruber, Florian, Mayer, Herbert, Lengauer, Barbara, Mlitz, Veronika, Sanders, John M, Kadl, Alexandra, Bilban, Martin, de Martin, Rainer, Wagner, Oswald, Kensler, Thomas W, Yamamoto, Masayuki, Leitinger, Norbert, Tschachler, Erwin
Published in The FASEB journal (01.01.2010)
Published in The FASEB journal (01.01.2010)
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Journal Article
Endothelial Cell PECAM-1 Promotes Atherosclerotic Lesions in Areas of Disturbed Flow in ApoE-Deficient Mice
Harry, Brian L, Sanders, John M, Feaver, Ryan E, Lansey, Melissa, Deem, Tracy L, Zarbock, Alexander, Bruce, Anthony C, Pryor, Andrew W, Gelfand, Bradley D, Blackman, Brett R, Schwartz, Martin A, Ley, Klaus
Published in Arteriosclerosis, thrombosis, and vascular biology (01.11.2008)
Published in Arteriosclerosis, thrombosis, and vascular biology (01.11.2008)
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Journal Article
Matrix-specific p21-activated kinase activation regulates vascular permeability in atherogenesis
Orr, A. Wayne, Stockton, Rebecca, Simmers, Michael B, Sanders, John M, Sarembock, Ian J, Blackman, Brett R, Schwartz, Martin Alexander
Published in The Journal of cell biology (26.02.2007)
Published in The Journal of cell biology (26.02.2007)
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Journal Article
Discovery and optimization of 2-pyridinone aminal integrase strand transfer inhibitors for the treatment of HIV
Schreier, John D., Embrey, Mark W., Raheem, Izzat T., Barbe, Guillaume, Campeau, Louis-Charles, Dubost, David, McCabe Dunn, Jamie, Grobler, Jay, Hartingh, Timothy J., Hazuda, Daria J., Klein, Daniel, Miller, Michael D., Moore, Keith P., Nguyen, Natalie, Pajkovic, Natasa, Powell, David A., Rada, Vanessa, Sanders, John M., Sisko, John, Steele, Thomas G., Wai, John, Walji, Abbas, Xu, Min, Coleman, Paul J.
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
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Journal Article
Improved Survival and Reduced Vascular Permeability by Eliminating or Blocking 12/15-Lipoxygenase in Mouse Models of Acute Lung Injury (ALI)
Zarbock, Alexander, DiStasi, Matthew R, Smith, Emily, Sanders, John M, Kronke, Gerhard, Harry, Brian L, von Vietinghoff, Sibylle, Buscher, Konrad, Nadler, Jerry L, Ley, Klaus
Published in The Journal of immunology (1950) (01.10.2009)
Published in The Journal of immunology (1950) (01.10.2009)
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Journal Article
Synthesis and Evaluation of Heterocyclic Catechol Mimics as Inhibitors of Catechol-O-methyltransferase (COMT)
Harrison, Scott T, Poslusney, Michael S, Mulhearn, James J, Zhao, Zhijian, Kett, Nathan R, Schubert, Jeffrey W, Melamed, Jeffrey Y, Allison, Timothy J, Patel, Sangita B, Sanders, John M, Sharma, Sujata, Smith, Robert F, Hall, Dawn L, Robinson, Ronald G, Sachs, Nancy A, Hutson, Pete H, Wolkenberg, Scott E, Barrow, James C
Published in ACS medicinal chemistry letters (12.03.2015)
Published in ACS medicinal chemistry letters (12.03.2015)
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Journal Article
Adeno-associated virus serotype 9-mediated overexpression of extracellular superoxide dismutase improves recovery from surgical hind-limb ischemia in BALB/c mice
Saqib, Amina, MBBS, Prasad, Konkal-Matt R., PhD, Katwal, Arabindra B., MBBS, Sanders, John M., BS, Lye, R. John, PhD, French, Brent A., PhD, Annex, Brian H
Published in Journal of vascular surgery (01.09.2011)
Published in Journal of vascular surgery (01.09.2011)
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Journal Article
3-Aryl-5-phenoxymethyl-1,3-oxazolidin-2-ones as positive allosteric modulators of mGluR2 for the treatment of schizophrenia: Hit-to-lead efforts
Brnardic, Edward J., Fraley, Mark E., Garbaccio, Robert M., Layton, Mark E., Sanders, John M., Culberson, Chris, Jacobson, Marlene A., Magliaro, Brian C., Hutson, Pete H., O’Brien, Julie A., Huszar, Sarah L., Uslaner, Jason M., Fillgrove, Kerry L., Tang, Cuyue, Kuo, Yuhsin, Sur, Sylvie M., Hartman, George D.
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
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Journal Article
Single injection of P-selectin or P-selectin glycoprotein ligand-1 monoclonal antibody blocks neointima formation after arterial injury in apolipoprotein E-deficient mice
PHILLIPS, J. William, BARRINGHAUS, Kurt G, SANDERS, John M, HESSELBACHER, Sean E, CZARNIK, Ann C, MANKA, David, VESTWEBER, Dietmar, LEY, Klaus, SAREMBOCK, Ian J
Published in Circulation (New York, N.Y.) (06.05.2003)
Published in Circulation (New York, N.Y.) (06.05.2003)
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Journal Article
Crystallographic Structures of Two Bisphosphonate:1-Deoxyxylulose-5-Phosphate Reductoisomerase Complexes
Yajima, Shunsuke, Hara, Kodai, Sanders, John M, Yin, Fenglin, Ohsawa, Kanju, Wiesner, Jochen, Jomaa, Hassan, Oldfield, Eric
Published in Journal of the American Chemical Society (08.09.2004)
Published in Journal of the American Chemical Society (08.09.2004)
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Journal Article
Integrin Agonists as Adjuvants in Chemotherapy for Melanoma
SCHWARTZ, Martin A, MCROBERTS, Kevin, COYNER, Matthew, ANDARAWEWA, Kumari L, FRIERSON, Henry F, SANDERS, John M, SWENSON, Stephen, MARKLAND, Frank, CONAWAY, Mark R, THEODORESCU, Dan
Published in Clinical cancer research (01.10.2008)
Published in Clinical cancer research (01.10.2008)
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Journal Article
Arterial Macrophages and Regenerating Endothelial Cells Express P-Selectin in Atherosclerosis-Prone Apolipoprotein E-Deficient Mice
Li, Guohong, Sanders, John M., Phan, Elizabeth T., Ley, Klaus, Sarembock, Ian J.
Published in The American journal of pathology (01.12.2005)
Published in The American journal of pathology (01.12.2005)
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Journal Article
Molecular imaging of inflammation in atherosclerosis with targeted ultrasound detection of vascular cell adhesion molecule-1
KAUFMANN, Beat A, SANDERS, John M, DAVIS, Christopher, XIE, Aris, ALDRED, Patrick, SAREMBOCK, Ian J, LINDNER, Jonathan R
Published in Circulation (New York, N.Y.) (17.07.2007)
Published in Circulation (New York, N.Y.) (17.07.2007)
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Journal Article
Rosiglitazone reduces the accelerated neointima formation after arterial injury in a mouse injury model of type 2 diabetes
PHILLIPS, J. William, BARRINGHAUS, Kurt G, SANDERS, John M, ZANDONG YANG, MENG CHEN, HESSELBACHER, Sean, CZARNIK, Ann C, LEY, Klaus, NADLER, Jerry, SAREMBOCK, Ian J
Published in Circulation (New York, N.Y.) (21.10.2003)
Published in Circulation (New York, N.Y.) (21.10.2003)
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Journal Article
Discovery of a 3‑(4-Pyrimidinyl) Indazole (MLi-2), an Orally Available and Selective Leucine-Rich Repeat Kinase 2 (LRRK2) Inhibitor that Reduces Brain Kinase Activity
Scott, Jack D, DeMong, Duane E, Greshock, Thomas J, Basu, Kallol, Dai, Xing, Harris, Joel, Hruza, Alan, Li, Sarah W, Lin, Sue-Ing, Liu, Hong, Macala, Megan K, Hu, Zhiyong, Mei, Hong, Zhang, Honglu, Walsh, Paul, Poirier, Marc, Shi, Zhi-Cai, Xiao, Li, Agnihotri, Gautam, Baptista, Marco A. S, Columbus, John, Fell, Matthew J, Hyde, Lynn A, Kuvelkar, Reshma, Lin, Yinghui, Mirescu, Christian, Morrow, John A, Yin, Zhizhang, Zhang, Xiaoping, Zhou, Xiaoping, Chang, Ronald K, Embrey, Mark W, Sanders, John M, Tiscia, Heather E, Drolet, Robert E, Kern, Jonathan T, Sur, Sylvie M, Renger, John J, Bilodeau, Mark T, Kennedy, Matthew E, Parker, Eric M, Stamford, Andrew W, Nargund, Ravi, McCauley, John A, Miller, Michael W
Published in Journal of medicinal chemistry (13.04.2017)
Published in Journal of medicinal chemistry (13.04.2017)
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Journal Article