Microwave assisted synthesis: a new technology in drug discovery
Santagada, V, Frecentese, F, Perissutti, E, Fiorino, F, Severino, B, Caliendo, G
Published in Mini reviews in medicinal chemistry (01.03.2009)
Published in Mini reviews in medicinal chemistry (01.03.2009)
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Journal Article
Derivatives as 5HT1A Receptor Ligands-Past and Present
CALIENDO, G, SANTAGADA, V, PERISSUTTI, E, FIORINO, F
Published in Current medicinal chemistry (2005)
Published in Current medicinal chemistry (2005)
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Journal Article
Synthesis of phenylpyrimidinones as guanylyl cyclase C inhibitors
Magli, E., Fiorino, F., Severino, B., Corvino, A., Perissutti, E., Frecentese, F., Giordano, F., Saccone, Luciano, P., Zaminelli, T., Santagada, Caliendo, G., de Nucci, G.
Published in Pharmazie (01.01.2019)
Published in Pharmazie (01.01.2019)
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Journal Article
Racemic synthesis and solid phase peptide synthesis application of the chimeric valine/leucine derivative 2-amino-3,3,4-trimethyl-pentanoic acid
Pelà, Zoppo, L. Del, Allegri, Marzola, Trapella, Ruzza, Calo, Perissutti, Frecentese, Salvadori, Guerrini
Published in Pharmazie (01.07.2014)
Published in Pharmazie (01.07.2014)
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Journal Article
Recent advances in synthesis of PAR ligands as therapeutic strategy for inflammatory diseases
Severino, B, Santagada, V, Perissutti, E, Fiorino, F, Frecentese, F, De Angelis, F, Esposito, A, Caliendo, G
Published in Mini reviews in medicinal chemistry (01.06.2009)
Published in Mini reviews in medicinal chemistry (01.06.2009)
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Journal Article
Synthesis and in vitro pharmacological evaluation of a new series of 5-HT1A 5-HT2A and 5-HT2C receptor ligands containing a norbornene nucleus
Fiorino, F., Severino, B., De Angelis, F., Perissutti, E., Magli, E., Frecentese, F., Esposito, A., Massarelli, P., Nencini, C., Viti, B., Santagada, V., Caliendo, G.
Published in Pharmazie (01.09.2009)
Published in Pharmazie (01.09.2009)
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Journal Article
In vitro mutagenicity of anti-inflammatory parsalmide analogues PA7, PA10, and PA31 triggered by biotransformation into hydroxy derivatives
Cardoso, H.S., Bicalho, B., Genari, P., Santagada, V., Caliendo, G., Perissutti, E., Donato, J.L., De Nucci, G.
Published in European journal of medicinal chemistry (01.03.2006)
Published in European journal of medicinal chemistry (01.03.2006)
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Journal Article
Comparative bioavailability of two losartan formulations in healthy human volunteers after a single dose administration
Oliveira, C H, Medeiros Silva, R, Santagada, V, Caliendo, G, Perissutti, E, Prado Galuppo, M, Marcondes Rezende, V, Barrientos-Astigarraga, R E, Mendes, G Duarte, De Nucci, G
Published in International journal of clinical pharmacology and therapeutics (01.03.2006)
Published in International journal of clinical pharmacology and therapeutics (01.03.2006)
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Journal Article
Human Tissue Kallikrein S1 Subsite Recognition of Non-Natural Basic Amino Acids
Melo, Robson L, Barbosa Pozzo, Roseli C, Pimenta, Daniel C, Perissutti, Elisa, Caliendo, Giuseppe, Santagada, Vincenzo, Juliano, Luiz, Juliano, Maria A
Published in Biochemistry (Easton) (01.05.2001)
Published in Biochemistry (Easton) (01.05.2001)
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Journal Article
Structure—affinity relationship studies on benzotriazole derivatives binding to 5-HT receptor subtypes
Caliendo, G, Greco, G, Grieco, P, Novellino, E, Perissutti, E, Santagada, V, Barbarulo, D, Esposito, E, De Blasi, A
Published in European journal of medicinal chemistry (1996)
Published in European journal of medicinal chemistry (1996)
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Journal Article
499 Effect of norbornene derivative in corpus cavernosum relaxation, as 5-HT1A agonist and 5-HT2A antagonist
Justo, A.F.O., Campos, R., Kiguti, L.R., Corvino, A., Fiorino, F., Frecentese, F., Magli, E., Perissutti, E., Saccone, I., De Nucci, G.
Published in Journal of sexual medicine (01.07.2018)
Published in Journal of sexual medicine (01.07.2018)
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Journal Article
Synthesis, local anesthetic activity and QSAR studies for a set of N-[2-(alkylamino)ethyl]benzotriazol- x-yl acetamides
Caliendo, G, Di Carlo, R, Greco, G, Grieco, P, Meli, R, Novellino, E, Perissutti, E, Santagada, V
Published in European journal of medicinal chemistry (1995)
Published in European journal of medicinal chemistry (1995)
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Journal Article
Synthesis and pharmacological evaluation of a set of N-[2-(alkylamino)ethyl]benzotriazol- X-yl isobutyramides acting as local anesthetics
Caliendo, G, Greco, G, Grieco, P, Raso, G Mattace, Meli, R, Novellino, E, Perissutti, E, Santagada, V
Published in European journal of medicinal chemistry (1996)
Published in European journal of medicinal chemistry (1996)
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Journal Article
Synthesis and structure-activity relationships of antiinflammatory 1-methyl-2-(4- X-benzoyl)imidazole-5-acetic acids
Caliendo, G, Cirino, G, Greco, G, Novellino, E, Perissutti, E, Pinto, A, Santagada, V, Silipo, C, Sorrentino, L
Published in European journal of medicinal chemistry (1994)
Published in European journal of medicinal chemistry (1994)
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Journal Article