Iterative Design and Optimization of Initially Inactive Proteolysis Targeting Chimeras (PROTACs) Identify VZ185 as a Potent, Fast, and Selective von Hippel–Lindau (VHL) Based Dual Degrader Probe of BRD9 and BRD7
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Published in Journal of medicinal chemistry (24.01.2019)
Published in Journal of medicinal chemistry (24.01.2019)
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Journal Article
Translating PROTAC chemical series optimization into functional outcomes underlying BRD7 and BRD9 protein degradation
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Published in Current research in chemical biology (2021)
Published in Current research in chemical biology (2021)
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벤젠술폰아미드 유도체 및 그의 용도
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Year of Publication 29.04.2022
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Year of Publication 29.04.2022
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Year of Publication 27.12.2023
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BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF
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Year of Publication 26.07.2023
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Benzenesulfonamide derivatives and uses thereof
Vittoria Zoppi, Siawash Ahmar, Gary K.C. Tin, David Armstrong, Sana Rasheed, Jeffrey Alan Omeara, Ayah Abdeldayem, Ji Sung Park, David Alexander Rosa, Patrick T. Gunning, Graham Simpson, Geordon A. Frere, Aaron D Cabral, Erica J. Quilates, Olga Gozhina
Year of Publication 23.11.2022
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Year of Publication 23.11.2022
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BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF
SIMPSON, Graham, ARMSTRONG, David, PARK, Ji Sung, AHMAR, Siawash, FRERE, Geordon A, QUILATES, Erica J, RASHEED, Sana, ROSA, David Alexander, ZOPPI, Vittoria, GUNNING, Patrick T, TIN, Gary K.C, OMEARA, Jeffrey Alan, GOZHINA, Olga, CABRAL, Aaron D, ABDELDAYEM, Ayah
Year of Publication 08.09.2022
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Year of Publication 08.09.2022
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BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF
TIN, Gary, K.C, FRERE, Geordon, A, SIMPSON, Graham, GUNNING, Patrick, T, ARMSTRONG, David, PARK, Ji Sung, CABRAL, Aaron, D, AHMAR, Siawash, RASHEED, Sana, ROSA, David Alexander, ZOPPI, Vittoria, OMEARA, Jeffrey Alan, GOZHINA, Olga, ABDELDAYEM, Ayah, QUILATES, Erica, J
Year of Publication 29.06.2022
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Year of Publication 29.06.2022
Patent
Benzenesulfonamide derivatives and uses thereof
SIMPSON, Graham, ARMSTRONG, David, PARK, Ji Sung, AHMAR, Siawash, FRERE, Geordon A, QUILATES, Erica J, RASHEED, Sana, ROSA, David Alexander, ZOPPI, Vittoria, GUNNING, Patrick T, TIN, Gary K.C, OMEARA, Jeffrey Alan, GOZHINA, Olga, CABRAL, Aaron D, ABDELDAYEM, Ayah
Year of Publication 24.02.2022
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Year of Publication 24.02.2022
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BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF
OMEARA, JEFFREY ALAN, CABRAL, AARON, AHMAR, SIAWASH, ZOPPI, VITTORIA, FRERE, GEORDON A, QUILATES, ERICA J, GOZHINA, OLGA, SIMPSON, GRAHAM, PARK, JI SUNG, ROSA, DAVID ALEXANDER, ABDELDAYEM, AYAH, TIN, GARY K.C, GUNNING, PATRICK T, ARMSTRONG, DAVID, RASHEED, SANA
Year of Publication 21.01.2021
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Year of Publication 21.01.2021
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Benzenesulfonamide derivative and application thereof
O 'MEARA, JEFFREY, AARON, GUNNING PATRICK T, ROSA DAVID ALEXANDER, ZOPPI, VITTORIA, SIMPSON, GRAHAM, CABRAL AARON D, TING, GARY, K.C, RASHID SANA, GOCHAINA OLGA, QUERATS ERICA J, ARMSTRONG DAVID, FREIRE, JORDAN, A, PARK JI-SUNG, ABDELDAYEM, AYA, AHMAR, SHIAVASH
Year of Publication 13.05.2022
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Year of Publication 13.05.2022
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BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF
SIMPSON Graham, CABRAL Aaron D, FRERE Geordon A, QUILATES Erica J, ARMSTRONG David, TIN Gary K. C, AHMAR Siawash, ABDELDAYEM Ayah, ROSA David Alexander, PARK Ji Sung, GOZHINA Olga, OMEARA Jeffrey Alan, GUNNING Patrick T, RASHEED Sana, ZOPPI Vittoria
Year of Publication 27.04.2022
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Year of Publication 27.04.2022
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