Trivalent PROTACs enhance protein degradation via combined avidity and cooperativity
Imaide, Satomi, Riching, Kristin M., Makukhin, Nikolai, Vetma, Vesna, Whitworth, Claire, Hughes, Scott J., Trainor, Nicole, Mahan, Sarah D., Murphy, Nancy, Cowan, Angus D., Chan, Kwok-Ho, Craigon, Conner, Testa, Andrea, Maniaci, Chiara, Urh, Marjeta, Daniels, Danette L., Ciulli, Alessio
Published in Nature chemical biology (01.11.2021)
Published in Nature chemical biology (01.11.2021)
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Journal Article
Selective targeting of BD1 and BD2 of the BET proteins in cancer and immunoinflammation
Gilan, Omer, Rioja, Inmaculada, Knezevic, Kathy, Bell, Matthew J, Yeung, Miriam M, Harker, Nicola R, Lam, Enid Y N, Chung, Chun-Wa, Bamborough, Paul, Petretich, Massimo, Urh, Marjeta, Atkinson, Stephen J, Bassil, Anna K, Roberts, Emma J, Vassiliadis, Dane, Burr, Marian L, Preston, Alex G S, Wellaway, Christopher, Werner, Thilo, Gray, James R, Michon, Anne-Marie, Gobbetti, Thomas, Kumar, Vinod, Soden, Peter E, Haynes, Andrea, Vappiani, Johanna, Tough, David F, Taylor, Simon, Dawson, Sarah-Jane, Bantscheff, Marcus, Lindon, Matthew, Drewes, Gerard, Demont, Emmanuel H, Daniels, Danette L, Grandi, Paola, Prinjha, Rab K, Dawson, Mark A
Published in Science (American Association for the Advancement of Science) (24.04.2020)
Published in Science (American Association for the Advancement of Science) (24.04.2020)
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Journal Article
Development of NanoLuc bridging immunoassay for detection of anti-drug antibodies
Nath, Nidhi, Flemming, Rod, Godat, Becky, Urh, Marjeta
Published in Journal of immunological methods (01.11.2017)
Published in Journal of immunological methods (01.11.2017)
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Journal Article
TET2 and TET3 regulate GlcNAcylation and H3K4 methylation through OGT and SET1/COMPASS
Deplus, Rachel, Delatte, Benjamin, Schwinn, Marie K, Defrance, Matthieu, Méndez, Jacqui, Murphy, Nancy, Dawson, Mark A, Volkmar, Michael, Putmans, Pascale, Calonne, Emilie, Shih, Alan H, Levine, Ross L, Bernard, Olivier, Mercher, Thomas, Solary, Eric, Urh, Marjeta, Daniels, Danette L, Fuks, François
Published in The EMBO journal (06.03.2013)
Published in The EMBO journal (06.03.2013)
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Journal Article
Generation of a Selective Small Molecule Inhibitor of the CBP/p300 Bromodomain for Leukemia Therapy
Picaud, Sarah, Fedorov, Oleg, Thanasopoulou, Angeliki, Leonards, Katharina, Jones, Katherine, Meier, Julia, Olzscha, Heidi, Monteiro, Octovia, Martin, Sarah, Philpott, Martin, Tumber, Anthony, Filippakopoulos, Panagis, Yapp, Clarence, Wells, Christopher, Che, Ka Hing, Bannister, Andrew, Robson, Samuel, Kumar, Umesh, Parr, Nigel, Lee, Kevin, Lugo, Dave, Jeffrey, Philip, Taylor, Simon, Vecellio, Matteo L, Bountra, Chas, Brennan, Paul E, O'Mahony, Alison, Velichko, Sharlene, Müller, Susanne, Hay, Duncan, Daniels, Danette L, Urh, Marjeta, La Thangue, Nicholas B, Kouzarides, Tony, Prinjha, Rab, Schwaller, Jürg, Knapp, Stefan
Published in Cancer research (Chicago, Ill.) (01.12.2015)
Published in Cancer research (Chicago, Ill.) (01.12.2015)
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Journal Article
The TIP60 Complex Is a Conserved Coactivator of HIF1A
Perez-Perri, Joel I., Dengler, Veronica L., Audetat, K. Audrey, Pandey, Ahwan, Bonner, Elizabeth A., Urh, Marjeta, Mendez, Jacqui, Daniels, Danette L., Wappner, Pablo, Galbraith, Matthew D., Espinosa, Joaquín M.
Published in Cell reports (Cambridge) (28.06.2016)
Published in Cell reports (Cambridge) (28.06.2016)
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Journal Article
Selective CK1α degraders exert antiproliferative activity against a broad range of human cancer cell lines
Nishiguchi, Gisele, Mascibroda, Lauren G., Young, Sarah M., Caine, Elizabeth A., Abdelhamed, Sherif, Kooijman, Jeffrey J., Miller, Darcie J., Das, Sourav, McGowan, Kevin, Mayasundari, Anand, Shi, Zhe, Barajas, Juan M., Hiltenbrand, Ryan, Aggarwal, Anup, Chang, Yunchao, Mishra, Vibhor, Narina, Shilpa, Thomas, Melvin, Loughran, Allister J., Kalathur, Ravi, Yu, Kaiwen, Zhou, Suiping, Wang, Xusheng, High, Anthony A., Peng, Junmin, Pruett-Miller, Shondra M., Daniels, Danette L., Urh, Marjeta, Shelat, Anang A., Mullighan, Charles G., Riching, Kristin M., Zaman, Guido J. R., Fischer, Marcus, Klco, Jeffery M., Rankovic, Zoran
Published in Nature communications (16.01.2024)
Published in Nature communications (16.01.2024)
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Journal Article
Highly Efficient Protein and Complex Purification from Mammalian Cells Using the HaloTag® Technology
Méndez, Jacqui L, Ohana, Rachel Friedman, Hurst, Robin, Murphy, Nancy, Benink, Hélène, Slater, Michael R, Brueck, Chad, Daniels, Danette L, Urh, Marjeta
Published in BioTechniques (01.10.2011)
Published in BioTechniques (01.10.2011)
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Journal Article
Quantitative Live-Cell Kinetic Degradation and Mechanistic Profiling of PROTAC Mode of Action
Riching, Kristin M, Mahan, Sarah, Corona, Cesear R, McDougall, Mark, Vasta, James D, Robers, Matthew B, Urh, Marjeta, Daniels, Danette L
Published in ACS chemical biology (21.09.2018)
Published in ACS chemical biology (21.09.2018)
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Journal Article
Characterization and quantification of succinimide using peptide mapping under low-pH conditions and hydrophobic interaction chromatography
Cao, Mingyan, Mulagapati, Sri Hari Raju, Vemulapalli, Bhargavi, Wang, Jihong, Saveliev, Sergei V., Urh, Marjeta, Hunter, Alan, Liu, Dengfeng
Published in Analytical biochemistry (01.02.2019)
Published in Analytical biochemistry (01.02.2019)
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Journal Article
Addressing common challenges of biotherapeutic protein peptide mapping using recombinant trypsin
Menneteau, Thomas, Saveliev, Sergei, Butré, Claire I., Rivera, Alba Katiria González, Urh, Marjeta, Delobel, Arnaud
Published in Journal of pharmaceutical and biomedical analysis (15.06.2024)
Published in Journal of pharmaceutical and biomedical analysis (15.06.2024)
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Journal Article
Modeling the CRL4A ligase complex to predict target protein ubiquitination induced by cereblon-recruiting PROTACs
Bai, Nan, Riching, Kristin M., Makaju, Aman, Wu, Hao, Acker, Timothy M., Ou, Shu-Ching, Zhang, Yaru, Shen, Xiaomeng, Bulloch, Daryl N., Rui, Huan, Gibson, Bradford W., Daniels, Danette L., Urh, Marjeta, Rock, Brooke M., Humphreys, Sara C.
Published in The Journal of biological chemistry (01.04.2022)
Published in The Journal of biological chemistry (01.04.2022)
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Journal Article
On-bead antibody-small molecule conjugation using high-capacity magnetic beads
Nath, Nidhi, Godat, Becky, Benink, Hélène, Urh, Marjeta
Published in Journal of immunological methods (01.11.2015)
Published in Journal of immunological methods (01.11.2015)
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Journal Article
An Automated and Qualified Platform Method for Site-Specific Succinimide and Deamidation Quantitation Using Low-pH Peptide Mapping
Cao, Mingyan, Xu, Weichen, Niu, Ben, Kabundi, Ivy, Luo, Haibin, Prophet, Meagan, Chen, Weimin, Liu, Dengfeng, Saveliev, Sergei V., Urh, Marjeta, Wang, Jihong
Published in Journal of pharmaceutical sciences (01.11.2019)
Published in Journal of pharmaceutical sciences (01.11.2019)
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Journal Article