1,2,3-Triazolyl-tetrahydropyrimidine Conjugates as Potential Sterol Carrier Protein-2 Inhibitors: Larvicidal Activity against the Malaria Vector Anopheles arabiensis and In Silico Molecular Docking Study
Venugopala, Katharigatta N, Shinu, Pottathil, Tratrat, Christophe, Deb, Pran Kishore, Gleiser, Raquel M, Chandrashekharappa, Sandeep, Chopra, Deepak, Attimarad, Mahesh, Nair, Anroop B, Sreeharsha, Nagaraja, Mahomoodally, Fawzi M, Haroun, Michelyne, Kandeel, Mahmoud, Asdaq, Syed Mohammed Basheeruddin, Mohanlall, Viresh, Al-Shar'i, Nizar A, Morsy, Mohamed A
Published in Molecules (Basel, Switzerland) (21.04.2022)
Published in Molecules (Basel, Switzerland) (21.04.2022)
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Journal Article
Larvicidal Activities of 2-Aryl-2,3-Dihydroquinazolin -4-ones against Malaria Vector Anopheles arabiensis , In Silico ADMET Prediction and Molecular Target Investigation
Venugopala, Katharigatta N, Ramachandra, Pushpalatha, Tratrat, Christophe, Gleiser, Raquel M, Bhandary, Subhrajyoti, Chopra, Deepak, Morsy, Mohamed A, Aldhubiab, Bandar E, Attimarad, Mahesh, Nair, Anroop B, Sreeharsha, Nagaraja, Venugopala, Rashmi, Deb, Pran Kishore, Chandrashekharappa, Sandeep, Khalil, Hany Ezzat, Alwassil, Osama I, Abed, Sara Nidal, Bataineh, Yazan A, Palenge, Ramachandra, Haroun, Michelyne, Pottathil, Shinu, Girish, Meravanige B, Akrawi, Sabah H, Mohanlall, Viresh
Published in Molecules (Basel, Switzerland) (13.03.2020)
Published in Molecules (Basel, Switzerland) (13.03.2020)
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Journal Article
Redescription of immatures of Dasyhelea flavifrons Guérin-Méneville (Culicomorpha: Ceratopogonidae) and new contribution to the knowledge of its larval habitats
Díaz, Florentina, Mangudo, Carolina, Gleiser, Raquel M, Ronderos, María M
Published in Anais da Academia Brasileira de Ciências (2019)
Published in Anais da Academia Brasileira de Ciências (2019)
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Journal Article
Culicidae community composition and temporal dynamics in Guapiaçu Ecological Reserve, Cachoeiras de Macacu, Rio de Janeiro, Brazil
Alencar, Jeronimo, de Mello, Cecilia Ferreira, Guimarães, Anthony Érico, Gil-Santana, Hélcio R, Silva, Júlia Dos Santos, Santos-Mallet, Jacenir R, Gleiser, Raquel M
Published in PloS one (27.03.2015)
Published in PloS one (27.03.2015)
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Journal Article
Geometric morphometrics of endophytic oviposition traces of Odonata (Eocene, Argentina)
Romero-Lebrón, Eugenia, Gleiser, Raquel M, Petrulevičius, Julián F
Published in Royal Society open science (01.12.2020)
Published in Royal Society open science (01.12.2020)
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Journal Article
Biodiversity and Temporal Distribution of Immature Culicidae in the Atlantic Forest, Rio de Janeiro State, Brazil
Alencar, Jeronimo, de Mello, Cecília Ferreira, Serra-Freire, Nicolau Maués, Guimarães, Anthony Érico, Gil-Santana, Hélcio R, Gleiser, Raquel M
Published in PloS one (12.07.2016)
Published in PloS one (12.07.2016)
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Journal Article
Greener synthesis of indolizine analogues using water as a base and solvent: study for larvicidal activity against Anopheles arabiensis
Sandeep, Chandrashekharappa, Venugopala, Katharigatta N., Gleiser, Raquel M., Chetram, Abeen, Padmashali, Basavaraj, Kulkarni, Rashmi S., Venugopala, Rashmi, Odhav, Bharti
Published in Chemical biology & drug design (01.12.2016)
Published in Chemical biology & drug design (01.12.2016)
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Journal Article
One-pot microwave assisted synthesis and structural elucidation of novel ethyl 3-substituted-7-methylindolizine-1-carboxylates with larvicidal activity against Anopheles arabiensis
Chandrashekharappa, Sandeep, Venugopala, Katharigatta N., Nayak, Susanta K., M. Gleiser, Raquel, García, Daniel A., Kumalo, Hezekiel M., Kulkarni, Rashmi S., Mahomoodally, Fawzi M., Venugopala, Rashmi, Mohan, Mahendra K., Odhav, Bharti
Published in Journal of molecular structure (15.03.2018)
Published in Journal of molecular structure (15.03.2018)
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Journal Article
Effects of the essential oils of Lippia turbinata and Lippia polystachya (Verbenaceae) on the temporal pattern of locomotion of the mosquito Culex quinquefasciatus (Diptera: Culicidae) larvae
Kembro, Jackelyn M, Marin, Raúl H, Zygadlo, Julio A, Gleiser, Raquel M
Published in Parasitology research (1987) (01.04.2009)
Published in Parasitology research (1987) (01.04.2009)
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Journal Article
Synthesis and antimosquito properties of 2,6-substituted benzo[d]thiazole and 2,4-substituted benzo[d]thiazole analogues against Anopheles arabiensis
Venugopala, Katharigatta Narayanaswamy, Krishnappa, Manjula, Nayak, Susanta K., Subrahmanya, Bhat K., Vaderapura, Jayashankaragowda P., Chalannavar, Raju K., Gleiser, Raquel M., Odhav, Bharti
Published in European journal of medicinal chemistry (01.07.2013)
Published in European journal of medicinal chemistry (01.07.2013)
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Journal Article
Use of Aedes aegypti Oviposition Surveillance and a Geographic Information System for Planning Anti-Vectorial Measures
Abán Moreyra, Daira N., Castillo, Paola M., Escalada, Andrés, Mangudo, Carolina, Copa, Griselda N., Gleiser, Raquel M., Nasser, Julio R., Gil, José F.
Published in The American journal of tropical medicine and hygiene (12.10.2022)
Published in The American journal of tropical medicine and hygiene (12.10.2022)
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Journal Article
Larvicidal study of tetrahydropyrimidine scaffolds against Anopheles arabiensis and structural insight by single crystal X‐ray studies
Bairagi, Keshab M., Venugopala, Katharigatta N., Mondal, Pradip Kumar, Gleiser, Raquel M., Chopra, Deepak, García, Daniel, Odhav, Bharti, Nayak, Susanta K.
Published in Chemical biology & drug design (01.12.2018)
Published in Chemical biology & drug design (01.12.2018)
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Journal Article
Synthesis and characterization of a novel series of 1,4‐dihydropyridine analogues for larvicidal activity against Anopheles arabiensis
Dharma Rao, Bhaskara D., Bhandary, Subhrajyoti, Chopra, Deepak, Venugopala, Katharigatta N., Gleiser, Raquel M., Kasumbwe, Kabange, Odhav, Bharti
Published in Chemical biology & drug design (01.09.2017)
Published in Chemical biology & drug design (01.09.2017)
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Journal Article
Membrane effects of dihydropyrimidine analogues with larvicidal activity
Sánchez-Borzone, Mariela E., Mariani, Maria E., Miguel, Virginia, Gleiser, Raquel M., Odhav, Bharti, Venugopala, Katharigatta N., García, Daniel A.
Published in Colloids and surfaces, B, Biointerfaces (01.02.2017)
Published in Colloids and surfaces, B, Biointerfaces (01.02.2017)
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Journal Article
Snail shells as larval habitat of Limatus durhamii (Diptera: Culicidae) in the Yungas of Argentina
Mangudo, Carolina, Campos, Raúl E., Rossi, Gustavo C., Gleiser, Raquel M.
Published in Acta tropica (01.03.2017)
Published in Acta tropica (01.03.2017)
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Journal Article
Distribution of Haemagogus and Sabethes Species in Relation to Forest Cover and Climatic Factors in the Chapada Dos Guimarães National Park, State of Mato Grosso, Brazil
Alencar, Jeronimo, Mello, Cecilia Ferreira de, Morone, Fernanda, Albuquerque, Hermano Gomes, Serra-Freire, Nicolau Maués, Gleiser, Raquel M, Silva, Shayenne Olsson Freitas, Guimarães, Anthony Érico
Published in Journal of the American Mosquito Control Association (01.06.2018)
Published in Journal of the American Mosquito Control Association (01.06.2018)
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Journal Article