The Most Common Functional Groups in Bioactive Molecules and How Their Popularity Has Evolved over Time
Ertl, Peter, Altmann, Eva, McKenna, Jeffrey M
Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
Get full text
Journal Article
Discovery of a Covalent FEM1B Recruiter for Targeted Protein Degradation Applications
Henning, Nathaniel J, Manford, Andrew G, Spradlin, Jessica N, Brittain, Scott M, Zhang, Erika, McKenna, Jeffrey M, Tallarico, John A, Schirle, Markus, Rape, Michael, Nomura, Daniel K
Published in Journal of the American Chemical Society (19.01.2022)
Published in Journal of the American Chemical Society (19.01.2022)
Get full text
Journal Article
Harnessing the anti-cancer natural product nimbolide for targeted protein degradation
Spradlin, Jessica N., Hu, Xirui, Ward, Carl C., Brittain, Scott M., Jones, Michael D., Ou, Lisha, To, Milton, Proudfoot, Andrew, Ornelas, Elizabeth, Woldegiorgis, Mikias, Olzmann, James A., Bussiere, Dirksen E., Thomas, Jason R., Tallarico, John A., McKenna, Jeffrey M., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
Published in Nature Chemical Biology (01.07.2019)
Published in Nature Chemical Biology (01.07.2019)
Get full text
Journal Article
Covalent Ligand Screening Uncovers a RNF4 E3 Ligase Recruiter for Targeted Protein Degradation Applications
Ward, Carl C, Kleinman, Jordan I, Brittain, Scott M, Lee, Patrick S, Chung, Clive Yik Sham, Kim, Kenneth, Petri, Yana, Thomas, Jason R, Tallarico, John A, McKenna, Jeffrey M, Schirle, Markus, Nomura, Daniel K
Published in ACS Chemical Biology (15.11.2019)
Published in ACS Chemical Biology (15.11.2019)
Get full text
Journal Article
Bardoxolone conjugation enables targeted protein degradation of BRD4
Tong, Bingqi, Luo, Mai, Xie, Yi, Spradlin, Jessica N., Tallarico, John A., McKenna, Jeffrey M., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
Published in Scientific Reports (23.09.2020)
Published in Scientific Reports (23.09.2020)
Get full text
Journal Article
Discovery of a Functional Covalent Ligand Targeting an Intrinsically Disordered Cysteine within MYC
Boike, Lydia, Cioffi, Alexander G., Majewski, Felix C., Co, Jennifer, Henning, Nathaniel J., Jones, Michael D., Liu, Gang, McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Nomura, Daniel K.
Published in Cell Chemical Biology (21.01.2021)
Published in Cell Chemical Biology (21.01.2021)
Get full text
Journal Article
Chiral Diaryliodonium Phosphate Enables Light Driven Diastereoselective α‑C(sp3)–H Acetalization
Ye, Baihua, Zhao, Jie, Zhao, Ke, McKenna, Jeffrey M, Toste, F. Dean
Published in Journal of the American Chemical Society (05.07.2018)
Published in Journal of the American Chemical Society (05.07.2018)
Get full text
Journal Article
Chemoproteomics-enabled discovery of covalent RNF114-based degraders that mimic natural product function
Luo, Mai, Spradlin, Jessica N., Boike, Lydia, Tong, Bingqi, Brittain, Scott M., McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
Published in Cell chemical biology (15.04.2021)
Published in Cell chemical biology (15.04.2021)
Get full text
Journal Article
Manumycin polyketides act as molecular glues between UBR7 and P53
Isobe, Yosuke, Okumura, Mikiko, McGregor, Lynn M., Brittain, Scott M., Jones, Michael D., Liang, Xiaoyou, White, Ross, Forrester, William, McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
Published in Nature chemical biology (01.11.2020)
Published in Nature chemical biology (01.11.2020)
Get full text
Journal Article
Chemoproteomics-enabled discovery of a covalent molecular glue degrader targeting NF-κB
King, Elizabeth A., Cho, Yoojin, Hsu, Nathan S., Dovala, Dustin, McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Nomura, Daniel K.
Published in Cell chemical biology (20.04.2023)
Published in Cell chemical biology (20.04.2023)
Get full text
Journal Article
Deubiquitinase-targeting chimeras for targeted protein stabilization
Henning, Nathaniel J., Boike, Lydia, Spradlin, Jessica N., Ward, Carl C., Liu, Gang, Zhang, Erika, Belcher, Bridget P., Brittain, Scott M., Hesse, Matthew J., Dovala, Dustin, McGregor, Lynn M., Valdez Misiolek, Rachel, Plasschaert, Lindsey W., Rowlands, David J., Wang, Feng, Frank, Andreas O., Fuller, Daniel, Estes, Abigail R., Randal, Katelyn L., Panidapu, Anoohya, McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Nomura, Daniel K.
Published in Nature chemical biology (01.04.2022)
Published in Nature chemical biology (01.04.2022)
Get full text
Journal Article
A Nimbolide-Based Kinase Degrader Preferentially Degrades Oncogenic BCR-ABL
Tong, Bingqi, Spradlin, Jessica N, Novaes, Luiz F. T, Zhang, Erika, Hu, Xirui, Moeller, Malte, Brittain, Scott M, McGregor, Lynn M, McKenna, Jeffrey M, Tallarico, John A, Schirle, Markus, Maimone, Thomas J, Nomura, Daniel K
Published in ACS chemical biology (17.07.2020)
Published in ACS chemical biology (17.07.2020)
Get full text
Journal Article
The development and mechanistic investigation of a palladium-catalyzed 1,3-arylfluorination of chromenes
Thornbury, Richard T., Saini, Vaneet, Fernandes, Talita de A., Santiago, Celine B., Talbot, Eric P. A., Sigman, Matthew S., McKenna, Jeffrey M., Toste, F. Dean
Published in Chemical Science (01.04.2017)
Published in Chemical Science (01.04.2017)
Get full text
Journal Article
Targeted Protein Degradation through E2 Recruitment
Forte, Nafsika, Dovala, Dustin, Hesse, Matthew J., McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Nomura, Daniel K.
Published in ACS chemical biology (21.04.2023)
Published in ACS chemical biology (21.04.2023)
Get full text
Journal Article
Oxidative cyclization reagents reveal tryptophan cation–π interactions
Xie, Xiao, Moon, Patrick J., Crossley, Steven W. M., Bischoff, Amanda J., He, Dan, Li, Gen, Dao, Nam, Gonzalez-Valero, Angel, Reeves, Audrey G., McKenna, Jeffrey M., Elledge, Susanna K., Wells, James A., Toste, F. Dean, Chang, Christopher J.
Published in Nature (London) (21.03.2024)
Published in Nature (London) (21.03.2024)
Get full text
Journal Article
An Activity-Based Oxaziridine Platform for Identifying and Developing Covalent Ligands for Functional Allosteric Methionine Sites: Redox-Dependent Inhibition of Cyclin-Dependent Kinase 4
Gonzalez-Valero, Angel, Reeves, Audrey G., Page, Annika C. S., Moon, Patrick J., Miller, Edward, Coulonval, Katia, Crossley, Steven W. M., Xie, Xiao, He, Dan, Musacchio, Patricia Z., Christian, Alec H., McKenna, Jeffrey M., Lewis, Richard A., Fang, Eric, Dovala, Dustin, Lu, Yipin, McGregor, Lynn M., Schirle, Markus, Tallarico, John A., Roger, Pierre P., Toste, F. Dean, Chang, Christopher J.
Published in Journal of the American Chemical Society (21.12.2022)
Published in Journal of the American Chemical Society (21.12.2022)
Get full text
Journal Article