Fragment Screening and Assembly: A Highly Efficient Approach to a Selective and Cell Active Protein Tyrosine Phosphatase 1B Inhibitor
Liu, Gang, Xin, Zhili, Pei, Zhonghua, Hajduk, Philip J, Abad-Zapatero, Cele, Hutchins, Charles W, Zhao, Hongyu, Lubben, Thomas H, Ballaron, Stephen J, Haasch, Deanna L, Kaszubska, Wiweka, Rondinone, Cristina M, Trevillyan, James M, Jirousek, Michael R
Published in Journal of Medicinal Chemistry (25.09.2003)
Published in Journal of Medicinal Chemistry (25.09.2003)
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Discovery of Potent, Highly Selective, and Orally Bioavailable Pyridine Carboxamide c-Jun NH2-Terminal Kinase Inhibitors
Zhao, Hongyu, Serby, Michael D, Xin, Zhili, Szczepankiewicz, Bruce G, Liu, Mei, Kosogof, Christi, Liu, Bo, Nelson, Lissa T. J, Johnson, Eric F, Wang, Sanyi, Pederson, Terry, Gum, Rebecca J, Clampit, Jill E, Haasch, Deanna L, Abad-Zapatero, Cele, Fry, Elizabeth H, Rondinone, Cristina, Trevillyan, James M, Sham, Hing L, Liu, Gang
Published in Journal of Medicinal Chemistry (27.07.2006)
Published in Journal of Medicinal Chemistry (27.07.2006)
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Discovery of a new class of 4-anilinopyrimidines as potent c-Jun N-terminal kinase inhibitors: Synthesis and SAR studies
Liu, Mei, Wang, Sanyi, Clampit, Jill E., Gum, Rebecca J., Haasch, Deanna L., Rondinone, Cristina M., Trevillyan, James M., Abad-Zapatero, Cele, Fry, Elizabeth H., Sham, Hing L., Liu, Gang
Published in Bioorganic & Medicinal Chemistry Letters (01.02.2007)
Published in Bioorganic & Medicinal Chemistry Letters (01.02.2007)
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ABT-165, a Dual Variable Domain Immunoglobulin (DVD-Ig) Targeting DLL4 and VEGF, Demonstrates Superior Efficacy and Favorable Safety Profiles in Preclinical Models
Li, Yingchun, Hickson, Jonathan A, Ambrosi, Dominic J, Haasch, Deanna L, Foster-Duke, Kelly D, Eaton, Lucia J, DiGiammarino, Enrico L, Panchal, Sanjay C, Jiang, Fang, Mudd, Sarah R, Zhang, Catherine, Akella, Surekha S, Gao, Wenqing, Ralston, Sherry L, Naumovski, Louie, Gu, Jijie, Morgan-Lappe, Susan E
Published in Molecular cancer therapeutics (01.05.2018)
Published in Molecular cancer therapeutics (01.05.2018)
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Synthesis and SAR of 1,9-dihydro-9-hydroxypyrazolo[3,4-b]quinolin-4-ones as novel, selective c-Jun N-terminal kinase inhibitors
Liu, Mei, Xin, Zhili, Clampit, Jill E., Wang, Sanyi, Gum, Rebecca J., Haasch, Deanna L., Trevillyan, James M., Abad-Zapatero, Cele, Fry, Elizabeth H., Sham, Hing L., Liu, Gang
Published in Bioorganic & Medicinal Chemistry Letters (15.05.2006)
Published in Bioorganic & Medicinal Chemistry Letters (15.05.2006)
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Journal Article
Aminopyridine-Based c-Jun N-Terminal Kinase Inhibitors with Cellular Activity and Minimal Cross-Kinase Activity
Szczepankiewicz, Bruce G, Kosogof, Christi, Nelson, Lissa T. J, Liu, Gang, Liu, Bo, Zhao, Hongyu, Serby, Michael D, Xin, Zhili, Liu, Mei, Gum, Rebecca J, Haasch, Deanna L, Wang, Sanyi, Clampit, Jill E, Johnson, Eric F, Lubben, Thomas H, Stashko, Michael A, Olejniczak, Edward T, Sun, Chaohong, Dorwin, Sarah A, Haskins, Kristi, Abad-Zapatero, Cele, Fry, Elizabeth H, Hutchins, Charles W, Sham, Hing L, Rondinone, Cristina M, Trevillyan, James M
Published in Journal of medicinal chemistry (15.06.2006)
Published in Journal of medicinal chemistry (15.06.2006)
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Journal Article
Discovery and Characterization of Non-ATP Site Inhibitors of the Mitogen Activated Protein (MAP) Kinases
Comess, Kenneth M, Sun, Chaohong, Abad-Zapatero, Cele, Goedken, Eric R, Gum, Rebecca J, Borhani, David W, Argiriadi, Maria, Groebe, Duncan R, Jia, Yong, Clampit, Jill E, Haasch, Deanna L, Smith, Harriet T, Wang, Sanyi, Song, Danying, Coen, Michael L, Cloutier, Timothy E, Tang, Hua, Cheng, Xueheng, Quinn, Christopher, Liu, Bo, Xin, Zhili, Liu, Gang, Fry, Elizabeth H, Stoll, Vincent, Ng, Teresa I, Banach, David, Marcotte, Doug, Burns, David J, Calderwood, David J, Hajduk, Philip J
Published in ACS Chem. Biol (18.03.2011)
Published in ACS Chem. Biol (18.03.2011)
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Journal Article
Liver-specific Knockdown of JNK1 Up-regulates Proliferator-activated Receptor γ Coactivator 1β and Increases Plasma Triglyceride despite Reduced Glucose and Insulin Levels in Diet-induced Obese Mice
Yang, Ruojing, Wilcox, Denise M., Haasch, Deanna L., Jung, Paul M., Nguyen, Phong T., Voorbach, Martin J., Doktor, Stella, Brodjian, Sevan, Bush, Eugene N., Lin, Emily, Jacobson, Peer B., Collins, Christine A., Landschulz, Katherine T., Trevillyan, James M., Rondinone, Cristina M., Surowy, Terry K.
Published in Journal of biological chemistry/The Journal of biological chemistry (03.08.2007)
Published in Journal of biological chemistry/The Journal of biological chemistry (03.08.2007)
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Isoxazole carboxylic acids as protein tyrosine phosphatase 1B (PTP1B) inhibitors
Zhao, Hongyu, Liu, Gang, Xin, Zhili, Serby, Michael D., Pei, Zhonghua, Szczepankiewicz, Bruce G., Hajduk, Philip J., Abad-Zapatero, Cele, Hutchins, Charles W., Lubben, Thomas H., Ballaron, Stephen J., Haasch, Deanna L., Kaszubska, Wiweka, Rondinone, Cristina M., Trevillyan, James M., Jirousek, Michael R.
Published in Bioorganic & medicinal chemistry letters (15.11.2004)
Published in Bioorganic & medicinal chemistry letters (15.11.2004)
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Journal Article
Aminopyridine carboxamides as c-Jun N-terminal kinase inhibitors: Targeting the gatekeeper residue and beyond
Liu, Gang, Zhao, Hongyu, Liu, Bo, Xin, Zhili, Liu, Mei, Kosogof, Christi, Szczepankiewicz, Bruce G., Wang, Sanyi, Clampit, Jill E., Gum, Rebecca J., Haasch, Deanna L., Trevillyan, James M., Sham, Hing L.
Published in Bioorganic & medicinal chemistry letters (15.11.2006)
Published in Bioorganic & medicinal chemistry letters (15.11.2006)
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4 ANTI-VEGF/DLL4 DUAL VARIABLE DOMAIN IMMUNOGLOBULINS AND USES THEREOF
HAASCH DEANNA L, LAPPE SUSAN E, CHARI RAVI, LI YINGCHUN, AMBROSI DOMINIC J, GU JIJIE, NAUMOVSKI LOUIE, GUPTA SUPRIYA, CAO XIANHUA, HICKSON JONATHAN A, ZAMIRI CAMELLIA
Year of Publication 10.09.2021
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Year of Publication 10.09.2021
Patent
4 ANTI-VEGF/DLL4 DUAL VARIABLE DOMAIN IMMUNOGLOBULINS AND USES THEREOF
HAASCH DEANNA L, LAPPE SUSAN E, CHARI RAVI, LI YINGCHUN, AMBROSI DOMINIC J, GU JIJIE, NAUMOVSKI LOUIE, GUPTA SUPRIYA, CAO XIANHUA, HICKSON JONATHAN A, ZAMIRI CAMELLIA
Year of Publication 18.09.2019
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Year of Publication 18.09.2019
Patent
4 ANTI-VEGF/DLL4 DUAL VARIABLE DOMAIN IMMUNOGLOBULINS AND USES THEREOF
HAASCH DEANNA L, LAPPE SUSAN E, CHARI RAVI, LI YINGCHUN, AMBROSI DOMINIC J, GU JIJIE, NAUMOVSKI LOUIE, GUPTA SUPRIYA, CAO XIANHUA, HICKSON JONATHAN A, ZAMIRI CAMELLIA
Year of Publication 19.08.2019
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Year of Publication 19.08.2019
Patent
4 ANTI-VEGF/DLL4 DUAL VARIABLE DOMAIN IMMUNOGLOBULINS AND USES THEREOF
HAASCH DEANNA L, LAPPE SUSAN E, CHARI RAVI, LI YINGCHUN, AMBROSI DOMINIC J, GU JIJIE, NAUMOVSKI LOUIE, GUPTA SUPRIYA, CAO XIANHUA, HICKSON JONATHAN A, ZAMIRI CAMELLIA
Year of Publication 24.01.2018
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Year of Publication 24.01.2018
Patent
ANTI-VEGF/DLL4 DUAL VARIABLE DOMAIN IMMUNOGLOBULINS AND USES THEREOF
HAASCH DEANNA L, LAPPE SUSAN E, CHARI RAVI, LI YINGCHUN, AMBROSI DOMINIC J, GU JIJIE, NAUMOVSKI LOUIE, GUPTA SUPRIYA, CAO XIANHUA, HICKSON JONATHAN A, ZAMIRI CAMELLIA
Year of Publication 13.07.2015
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Year of Publication 13.07.2015
Patent
Differential Roles of JNK1 and JNK2 in Liver and Fat Cells
Gum, Rebecca J, Haasch, Deanna L, Clampit, Jill E, Carlson, Christian J
Published in Diabetes (New York, N.Y.) (01.06.2005)
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Published in Diabetes (New York, N.Y.) (01.06.2005)
Journal Article
Liver-specific Knockdown of JNK1 Up-regulates Proliferator-activated Receptor γ Coactivator 1β and Increases Plasma Triglyceride despite Reduced Glucose and Insulin Levels in Diet-induced Obese Mice
Ruojing Yang, Denise M. Wilcox, Deanna L. Haasch, Paul M. Jung, Phong T. Nguyen, Martin J. Voorbach, Stella Doktor, Sevan Brodjian, Eugene N. Bush, Emily Lin, Peer B. Jacobson, Christine A. Collins, Katherine T. Landschulz, James M. Trevillyan, Cristina M. Rondinone, Terry K. Surowy
Published in The Journal of biological chemistry (03.08.2007)
Published in The Journal of biological chemistry (03.08.2007)
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Journal Article
Discovery of Potent, Highly Selective, and Orally Bioavailable Pyridine Carboxamide c-Jun NH 2 -Terminal Kinase Inhibitors
Zhao, Hongyu, Serby, Michael D., Xin, Zhili, Szczepankiewicz, Bruce G., Liu, Mei, Kosogof, Christi, Liu, Bo, Nelson, Lissa T. J., Johnson, Eric F., Wang, Sanyi, Pederson, Terry, Gum, Rebecca J., Clampit, Jill E., Haasch, Deanna L., Abad-Zapatero, Cele, Fry, Elizabeth H., Rondinone, Cristina, Trevillyan, James M., Sham, Hing L., Liu, Gang
Published in Journal of medicinal chemistry (01.07.2006)
Published in Journal of medicinal chemistry (01.07.2006)
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Journal Article
ANTI-DLL4/VEGF DUAL VARIABLE DOMAIN IMMMUNOGLOBULIN AND USES THEREOF
Haasch, Deanna L, Cao, Xianhua, Ambrosi, Dominic J, Gu, Jijie, Zamiri, Camellia, Lappe, Susan E, Chari, Ravi, Li, Yingchun, Hickson, Jonathan A, Gupta, Supriya, Naumovski, Louie
Year of Publication 22.12.2022
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Year of Publication 22.12.2022
Patent
ANTI-DLL4/VEGF DUAL VARIABLE DOMAIN IMMUNOGLOBULIN AND USES THEREOF
GU, JIJIE, LI, YINGCHUN, HAASCH, DEANNA L, AMBROSI, DOMINIC J, LAPPE, SUSAN E, CAO, XIANHUA, CHARI, RAVI, ZAMIRI, CAMELLIA, HICKSON, JONATHAN A, GUPTA, SUPRIYA, NAUMOVSKI, LOUIE
Year of Publication 28.11.2022
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Year of Publication 28.11.2022
Patent