Heterocyclic ketones as inhibitors of histone deacetylase
Vasudevan, Anil, Ji, Zhiqin, Frey, Robin R., Wada, Carol K., Steinman, Douglas, Heyman, H.Robin, Guo, Yan, Curtin, Michael L., Guo, Jun, Li, Junling, Pease, Lori, Glaser, Keith B., Marcotte, Patrick A., Bouska, Jennifer J., Davidsen, Steven K., Michaelides, Michael R.
Published in Bioorganic & Medicinal Chemistry Letters (17.11.2003)
Published in Bioorganic & Medicinal Chemistry Letters (17.11.2003)
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Methylpyrrole inhibitors of BET bromodomains
Hasvold, Lisa A., Sheppard, George S., Wang, Le, Fidanze, Steven D., Liu, Dachun, Pratt, John K., Mantei, Robert A., Wada, Carol K., Hubbard, Robbert, Shen, Yu, Lin, Xiaoyu, Huang, Xiaoli, Warder, Scott E., Wilcox, Denise, Li, Leiming, Buchanan, F. Greg, Smithee, Lauren, Albert, Daniel H., Magoc, Terrance J., Park, Chang H., Petros, Andrew M., Panchal, Sanjay C., Sun, Chaohong, Kovar, Peter, Soni, Nirupama B., Elmore, Steven W., Kati, Warren M., McDaniel, Keith F.
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
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Trifluoromethyl ketones as inhibitors of histone deacetylase
Frey, Robin R., Wada, Carol K., Garland, Robert B., Curtin, Michael L., Michaelides, Michael R., Li, Junling, Pease, Lori J., Glaser, Keith B., Marcotte, Patrick A., Bouska, Jennifer J., Murphy, Shannon S., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
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α-Keto amides as inhibitors of histone deacetylase
Wada, Carol K., Frey, Robin R., Ji, Zhiqin, Curtin, Michael L., Garland, Robert B., Holms, James H., Li, Junling, Pease, Lori J., Guo, Jun, Glaser, Keith B., Marcotte, Patrick A., Richardson, Paul L., Murphy, Shannon S., Bouska, Jennifer J., Tapang, Paul, Magoc, Terrance J., Albert, Daniel H., Davidsen, Steven K., Michaelides, Michael R.
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
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Phenoxyphenyl Sulfone N-Formylhydroxylamines (Retrohydroxamates) as Potent, Selective, Orally Bioavailable Matrix Metalloproteinase Inhibitors
Wada, Carol K, Holms, James H, Curtin, Michael L, Dai, Yujia, Florjancic, Alan S, Garland, Robert B, Guo, Yan, Heyman, H. Robin, Stacey, Jamie R, Steinman, Douglas H, Albert, Daniel H, Bouska, Jennifer J, Elmore, Ildiko N, Goodfellow, Carole L, Marcotte, Patrick A, Tapang, Paul, Morgan, Douglas W, Michaelides, Michael R, Davidsen, Steven K
Published in Journal of medicinal chemistry (03.01.2002)
Published in Journal of medicinal chemistry (03.01.2002)
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Integrin ανβ3 Targeted Gene Delivery Using RGD Peptidomimetic Conjugates with Copolymers of PEGylated Poly(ethylene imine)
Olivia M. Merkel, Oliver Germershaus, Carol K. Wada, Peter J. Tarcha, Thomas Merdan, Thomas Kissel
Published in Bioconjugate Chemistry (28.05.2009)
Published in Bioconjugate Chemistry (28.05.2009)
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Biaryl Ether Retrohydroxamates as Potent, Long-lived, Orally Bioavailable MMP Inhibitors
Michaelides, Michael R., Dellaria, Joseph F., Gong, Jane, Holms, James H., Bouska, Jennifer J., Stacey, Jamie, Wada, Carol K., Heyman, H.Robin, Curtin, Michael L., Guo, Yan, Goodfellow, Carole L., Elmore, Ildiko B., Albert, Daniel H., Magoc, Terrance J., Marcotte, Patrick A., Morgan, Douglas W., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
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BROMODOMAIN INHIBITORS
WILLIAM J MCCLELLAN, ROBERT A MANTEI, JOHN H HOLMS, GEORGE S SHEPPARD, DAI YUJIA, CAROL K WADA, WARREN M KATI, LE WANG, LISA HASVOLD, LIU DACHUN, STEVEN D FIDANZE, MCDANIEL KEITH F, JOHN K PRATT
Year of Publication 08.11.2018
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Year of Publication 08.11.2018
Patent
BROMODOMAIN INHIBITORS
WILLIAM J MCCLELLAN, ROBERT A MANTEI, JOHN H HOLMS, GEORGE S SHEPPARD, DAI YUJIA, CAROL K WADA, WARREN M KATI, LE WANG, LISA HASVOLD, LIU DACHUN, STEVEN D FIDANZE, MCDANIEL KEITH F, JOHN K PRATT
Year of Publication 27.07.2017
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Year of Publication 27.07.2017
Patent
Discovery and characterization of the potent, selective and orally bioavailable MMP inhibitor ABT-770
Curtin, Michael L., Florjancic, Alan S., Heyman, H.Robin, Michaelides, Michael R., Garland, Robert B., Holms, James H., Steinman, Douglas H., Dellaria, Joseph F., Gong, Jane, Wada, Carol K., Guo, Yan, Elmore, Ildiko B., Tapang, Paul, Albert, Daniel H., Magoc, Terrance J., Marcotte, Patrick A., Bouska, Jennifer J., Goodfellow, Carole L., Bauch, Joy L., Marsh, Kennan C., Morgan, Douglas W., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
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Trifluoromethyl ketones as inhibitors of histone deacetylase
Robin R. Frey, Carol K. Wada, Robert B. Garland, Michael L. Curtin, Michael R. Michaelides, Junling Li, Lori J. Pease, Keith B. Glaser, Patrick A. Marcotte, Jennifer J. Bouska, Shannon S. Murphy, Steven K. Davidsen
Published in Bioorganic & Medicinal Chemistry Letters (01.12.2002)
Published in Bioorganic & Medicinal Chemistry Letters (01.12.2002)
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Triple‐Helix Formation by Pyrimidine Oligonucleotides Containing Nonnatural Nucleosides with Extended Aromatic Nucleobases: Intercalation from the major groove as a method for recognizing C·G and T · A base pairs
Thomas E. Lehmann, William A. Greenberg, David A. Liberles, Carol K. Wada, Peter B. Dervan
Published in Helvetica Chimica Acta (22.09.1997)
Published in Helvetica Chimica Acta (22.09.1997)
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Journal Article
Phenoxyphenyl SulfoneN-Formylhydroxylamines (Retrohydroxamates) as Potent, Selective, Orally Bioavailable Matrix Metalloproteinase Inhibitors
Carol K. Wada, James H. Holms, Michael L. Curtin, Yujia Dai, Alan S. Florjancic, Robert B. Garland, Yan Guo, H. Robin Heyman, Jamie R. Stacey, Douglas H. Steinman, Daniel H. Albert, Jennifer J. Bouska, Ildiko N. Elmore, Carole L. Goodfellow, Patrick A. Marcotte, Paul Tapang, Douglas W. Morgan, Michael R. Michaelides, Steven K. Davidsen
Published in Journal of Medicinal Chemistry (06.12.2001)
Published in Journal of Medicinal Chemistry (06.12.2001)
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Journal Article
Methylpyrrole inhibitors of BET bromodomains
Hasvold, Lisa A., Sheppard, George S., Wang, Le, Fidanze, Steven D., Liu, Dachun, Pratt, John K., Mantei, Robert A., Wada, Carol K., Hubbard, Robbert, Shen, Yu, Lin, Xiaoyu, Huang, Xiaoli, Warder, Scott E., Wilcox, Denise, Li, Leiming, Buchanan, F. Greg, Smithee, Lauren, Albert, Daniel H., Magoc, Terrance J., Park, Chang H., Petros, Andrew M., Panchal, Sanjay C., Sun, Chaohong, Kovar, Peter, Soni, Nirupama B., Elmore, Steven W., Kati, Warren M., McDaniel, Keith F.
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
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Published in Bioorganic & medicinal chemistry letters (01.05.2017)
Journal Article
Integrin α ν β 3 Targeted Gene Delivery Using RGD Peptidomimetic Conjugates with Copolymers of PEGylated Poly(ethylene imine)
Merkel, Olivia M., Germershaus, Oliver, Wada, Carol K., Tarcha, Peter J., Merdan, Thomas, Kissel, Thomas
Published in Bioconjugate chemistry (17.06.2009)
Published in Bioconjugate chemistry (17.06.2009)
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Integrin [alpha]^sub v^[beta]^sub 3^ Targeted Gene Delivery Using RGD Peptidomimetic Conjugates with Copolymers of PEGylated Poly(ethylene imine)
Merkel, Olivia M, Germershaus, Oliver, Wada, Carol K, Tarcha, Peter J, Merdan, Thomas, Kissel, Thomas
Published in Bioconjugate chemistry (17.06.2009)
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Published in Bioconjugate chemistry (17.06.2009)
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