Pharmacology of JNJ-42314415, a centrally active phosphodiesterase 10A (PDE10A) inhibitor: a comparison of PDE10A inhibitors with D2 receptor blockers as potential antipsychotic drugs
Megens, Anton A H P, Hendrickx, Herman M R, Hens, Koen A, Fonteyn, Ineke, Langlois, Xavier, Lenaerts, Ilse, Somers, Marijke V F, de Boer, Peter, Vanhoof, Greet
Published in The Journal of pharmacology and experimental therapeutics (01.04.2014)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2014)
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Using “big data” to describe the effect of seasonal variation in thyroid-stimulating hormone
De Grande, Linde A.C., Goossens, Kenneth, Van Uytfanghe, Katleen, Halsall, Ian, Yoshimura Noh, Jaeduk, Hens, Koen, Thienpont, Linda M.
Published in Clinical chemistry and laboratory medicine (01.02.2017)
Published in Clinical chemistry and laboratory medicine (01.02.2017)
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Discovery of a New Series of Centrally Active Tricyclic Isoxazoles Combining Serotonin (5-HT) Reuptake Inhibition with α2-Adrenoceptor Blocking Activity
Andrés, J. Ignacio, Alcázar, Jesús, Alonso, José M, Alvarez, Rosa M, Bakker, Margot H, Biesmans, Ilse, Cid, José M, De Lucas, Ana I, Fernández, Javier, Font, Luis M, Hens, Koen A, Iturrino, Laura, Lenaerts, Ilse, Martínez, Sonia, Megens, Anton A, Pastor, Joaquín, Vermote, Patrick C. M, Steckler, Thomas
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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Pharmacology of JNJ-42314415, a Centrally Active Phosphodiesterase 10A (PDE10A) Inhibitor: A Comparison of PDE10A Inhibitors with D 2 Receptor Blockers as Potential Antipsychotic Drugs
Megens, Anton A. H. P., Hendrickx, Herman M. R., Hens, Koen A., Fonteyn, Ineke, Langlois, Xavier, Lenaerts, Ilse, Somers, Marijke V. F., de Boer, Peter, Vanhoof, Greet
Published in The Journal of pharmacology and experimental therapeutics (01.04.2014)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2014)
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JNJ-40255293, a Novel Adenosine A2A/A1 Antagonist with Efficacy in Preclinical Models of Parkinson’s Disease
Atack, John R, Shook, Brian C, Rassnick, Stefanie, Jackson, Paul F, Rhodes, Kenneth, Drinkenburg, Wilhelmus H, Ahnaou, Abdallah, te Riele, Paula, Langlois, Xavier, Hrupka, Brian, De Haes, Patrick, Hendrickx, Herman, Aerts, Nancy, Hens, Koen, Wellens, Annemie, Vermeire, Jef, Megens, Anton A. H. P
Published in ACS chemical neuroscience (15.10.2014)
Published in ACS chemical neuroscience (15.10.2014)
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Journal Article
JNJ-40255293, a Novel Adenosine A 2A /A 1 Antagonist with Efficacy in Preclinical Models of Parkinson’s Disease
Atack, John R., Shook, Brian C., Rassnick, Stefanie, Jackson, Paul F., Rhodes, Kenneth, Drinkenburg, Wilhelmus H., Ahnaou, Abdallah, te Riele, Paula, Langlois, Xavier, Hrupka, Brian, De Haes, Patrick, Hendrickx, Herman, Aerts, Nancy, Hens, Koen, Wellens, Annemie, Vermeire, Jef, Megens, Anton A. H. P.
Published in ACS chemical neuroscience (15.10.2014)
Published in ACS chemical neuroscience (15.10.2014)
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Discovery of a new series of centrally active tricyclic isoxazoles combining serotonin (5-HT) reuptake inhibition with alpha2-adrenoceptor blocking activity
Andrés, J Ignacio, Alcázar, Jesús, Alonso, José M, Alvarez, Rosa M, Bakker, Margot H, Biesmans, Ilse, Cid, José M, De Lucas, Ana I, Fernández, Javier, Font, Luis M, Hens, Koen A, Iturrino, Laura, Lenaerts, Ilse, Martínez, Sonia, Megens, Anton A, Pastor, Joaquín, Vermote, Patrick C M, Steckler, Thomas
Published in Journal of medicinal chemistry (24.03.2005)
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Published in Journal of medicinal chemistry (24.03.2005)
Journal Article
Discovery of a New Series of Centrally Active Tricyclic Isoxazoles Combining Serotonin (5-HT) Reuptake Inhibition with α 2 -Adrenoceptor Blocking Activity
Andrés, J. Ignacio, Alcázar, Jesús, Alonso, José M., Alvarez, Rosa M., Bakker, Margot H., Biesmans, Ilse, Cid, José M., De Lucas, Ana I., Fernández, Javier, Font, Luis M., Hens, Koen A., Iturrino, Laura, Lenaerts, Ilse, Martínez, Sonia, Megens, Anton A., Pastor, Joaquín, Vermote, Patrick C. M., Steckler, Thomas
Published in Journal of medicinal chemistry (01.03.2005)
Published in Journal of medicinal chemistry (01.03.2005)
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Journal Article