Microwave assisted synthesis: a new technology in drug discovery
Santagada, V, Frecentese, F, Perissutti, E, Fiorino, F, Severino, B, Caliendo, G
Published in Mini reviews in medicinal chemistry (01.03.2009)
Published in Mini reviews in medicinal chemistry (01.03.2009)
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Journal Article
Synthesis of phenylpyrimidinones as guanylyl cyclase C inhibitors
Magli, E., Fiorino, F., Severino, B., Corvino, A., Perissutti, E., Frecentese, F., Giordano, F., Saccone, Luciano, P., Zaminelli, T., Santagada, Caliendo, G., de Nucci, G.
Published in Pharmazie (01.01.2019)
Published in Pharmazie (01.01.2019)
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Racemic synthesis and solid phase peptide synthesis application of the chimeric valine/leucine derivative 2-amino-3,3,4-trimethyl-pentanoic acid
Pelà, Zoppo, L. Del, Allegri, Marzola, Trapella, Ruzza, Calo, Perissutti, Frecentese, Salvadori, Guerrini
Published in Pharmazie (01.07.2014)
Published in Pharmazie (01.07.2014)
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Journal Article
Recent advances in synthesis of PAR ligands as therapeutic strategy for inflammatory diseases
Severino, B, Santagada, V, Perissutti, E, Fiorino, F, Frecentese, F, De Angelis, F, Esposito, A, Caliendo, G
Published in Mini reviews in medicinal chemistry (01.06.2009)
Published in Mini reviews in medicinal chemistry (01.06.2009)
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Journal Article
Synthesis and in vitro pharmacological evaluation of a new series of 5-HT1A 5-HT2A and 5-HT2C receptor ligands containing a norbornene nucleus
Fiorino, F., Severino, B., De Angelis, F., Perissutti, E., Magli, E., Frecentese, F., Esposito, A., Massarelli, P., Nencini, C., Viti, B., Santagada, V., Caliendo, G.
Published in Pharmazie (01.09.2009)
Published in Pharmazie (01.09.2009)
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Journal Article
In vitro mutagenicity of anti-inflammatory parsalmide analogues PA7, PA10, and PA31 triggered by biotransformation into hydroxy derivatives
Cardoso, H.S., Bicalho, B., Genari, P., Santagada, V., Caliendo, G., Perissutti, E., Donato, J.L., De Nucci, G.
Published in European journal of medicinal chemistry (01.03.2006)
Published in European journal of medicinal chemistry (01.03.2006)
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Journal Article
Comparative bioavailability of two losartan formulations in healthy human volunteers after a single dose administration
Oliveira, C H, Medeiros Silva, R, Santagada, V, Caliendo, G, Perissutti, E, Prado Galuppo, M, Marcondes Rezende, V, Barrientos-Astigarraga, R E, Mendes, G Duarte, De Nucci, G
Published in International journal of clinical pharmacology and therapeutics (01.03.2006)
Published in International journal of clinical pharmacology and therapeutics (01.03.2006)
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Journal Article
Structure—affinity relationship studies on benzotriazole derivatives binding to 5-HT receptor subtypes
Caliendo, G, Greco, G, Grieco, P, Novellino, E, Perissutti, E, Santagada, V, Barbarulo, D, Esposito, E, De Blasi, A
Published in European journal of medicinal chemistry (1996)
Published in European journal of medicinal chemistry (1996)
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Journal Article
Synthesis, local anesthetic activity and QSAR studies for a set of N-[2-(alkylamino)ethyl]benzotriazol- x-yl acetamides
Caliendo, G, Di Carlo, R, Greco, G, Grieco, P, Meli, R, Novellino, E, Perissutti, E, Santagada, V
Published in European journal of medicinal chemistry (1995)
Published in European journal of medicinal chemistry (1995)
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Journal Article
Synthesis and pharmacological evaluation of a set of N-[2-(alkylamino)ethyl]benzotriazol- X-yl isobutyramides acting as local anesthetics
Caliendo, G, Greco, G, Grieco, P, Raso, G Mattace, Meli, R, Novellino, E, Perissutti, E, Santagada, V
Published in European journal of medicinal chemistry (1996)
Published in European journal of medicinal chemistry (1996)
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Journal Article
Synthesis and structure-activity relationships of antiinflammatory 1-methyl-2-(4- X-benzoyl)imidazole-5-acetic acids
Caliendo, G, Cirino, G, Greco, G, Novellino, E, Perissutti, E, Pinto, A, Santagada, V, Silipo, C, Sorrentino, L
Published in European journal of medicinal chemistry (1994)
Published in European journal of medicinal chemistry (1994)
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Journal Article
Synthesis and in vitro activities of NK-1 antagonists derived from L-tryptophan
Caliendo, G, Fiorino, F, Grieco, P, Perissutti, E, Santagada, Calignano, A, Mancuso, F, Albrizio, S
Published in Farmaco (Società chimica italiana : 1989) (01.10.1997)
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Published in Farmaco (Società chimica italiana : 1989) (01.10.1997)
Journal Article
New 5-hydroxytryptamine(1A) receptor ligands containing a norbornene nucleus: Synthesis and in vitro pharmacological evaluation
Fiorino, F, Perissutti, E, Severino, B, Santagada, Cirillo, D, Terracciano, S, Massarelli, P, Bruni, G, Collavoli, E, Renner, C, Caliendo, G
Published in Journal of medicinal chemistry (25.08.2005)
Published in Journal of medicinal chemistry (25.08.2005)
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