Synthetically modified methoxsalen for enhanced cytotoxicity in light and dark reactions
Guillon, Christophe D., Jan, Yi-Hua, Foster, Natalie, Ressner, Joel, Heck, Diane E., Laskin, Jeffrey D., Heindel, Ned D.
Published in Bioorganic & medicinal chemistry letters (15.02.2019)
Published in Bioorganic & medicinal chemistry letters (15.02.2019)
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Derivatives of 1,2,4-triazole imines acting as dual iNOS and tumor cell growth inhibitors
Guillon, Christophe, Vetrano, Anna M., Saxena, Jaya, Hunter, Angela, Verderone, Geraldine, Finetti, Thomas M., Wisnoski, Jeffrey, DeMatteo, Peter W., Rapp, Robert D., Heindel, Ned D., Joseph, Laurie B., Heck, Diane E., Laskin, Jeffrey D.
Published in Bioorganic chemistry (01.10.2020)
Published in Bioorganic chemistry (01.10.2020)
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Journal Article
Ethynylphenyl carbonates and carbamates as dual-action acetylcholinesterase inhibitors and anti-inflammatory agents
Saxena, Jaya, Meloni, David, Huang, Mou-Tuan, Heck, Diane E., Laskin, Jeffrey D., Heindel, Ned D., Young, Sherri C.
Published in Bioorganic & medicinal chemistry letters (01.12.2015)
Published in Bioorganic & medicinal chemistry letters (01.12.2015)
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Journal Article
Multi-inhibitor prodrug constructs for simultaneous delivery of anti-inflammatory agents to mustard-induced skin injury
Lacey, Carl J., Wohlman, Irene, Guillon, Christophe, Saxena, Jaya, Fianu-Velgus, Cynthia, Aponte, Erik, Young, Sherri C., Heck, Diane E., Joseph, Laurie B., Laskin, Jeffrey D., Heindel, Ned D.
Published in Annals of the New York Academy of Sciences (01.08.2016)
Published in Annals of the New York Academy of Sciences (01.08.2016)
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Journal Article
Phototoxicity of 7-oxycoumarins with keratinocytes in culture
Guillon, Christophe, Jan, Yi-Hua, Heck, Diane E., Mariano, Thomas M., Rapp, Robert D., Jetter, Michele, Kardos, Keith, Whittemore, Marilyn, Akyea, Eric, Jabin, Ivan, Laskin, Jeffrey D., Heindel, Ned D.
Published in Bioorganic chemistry (01.08.2019)
Published in Bioorganic chemistry (01.08.2019)
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Journal Article
Pharmacokinetics and Metabolism of SRX246: A Potent and Selective Vasopressin 1a Antagonist
Fabio, Karine M., Guillon, Christophe D., Lu, Shi-Fang, Heindel, Ned D., Brownstein, Michael J., Lacey, Carl J., Garippa, Carrie, Simon, Neal G.
Published in Journal of pharmaceutical sciences (01.06.2013)
Published in Journal of pharmaceutical sciences (01.06.2013)
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Back-Scattering Interferometry: An Ultrasensitive Method for the Unperturbed Detection of Acetylcholinesterase-Inhibitor Interactions
Haddad, Gabrielle L., Young, Sherri C., Heindel, Ned D., Bornhop, Darryl J., Flowers II, Robert A.
Published in Angewandte Chemie (International ed.) (29.10.2012)
Published in Angewandte Chemie (International ed.) (29.10.2012)
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Synthesis and evaluation of potent and selective human V1a receptor antagonists as potential ligands for PET or SPECT imaging
Fabio, Karine, Guillon, Christophe, Lacey, Carl J., Lu, Shi-fang, Heindel, Ned D., Ferris, Craig F., Placzek, Michael, Jones, Graham, Brownstein, Michael J., Simon, Neal G.
Published in Bioorganic & medicinal chemistry (01.02.2012)
Published in Bioorganic & medicinal chemistry (01.02.2012)
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Journal Article
SYNTHESIS AND EVALUATION OF WATER-SOLUBLE DIMETHYLAMINOETHYL ETHERS OF METHOXSALEN FOR PROLIFERATIVE SKIN DISORDERS
Guillon, Christophe D, Jan, Yi-Hua, Foster, Natalie, Choudhuri, Mridula, Saxena, Jaya, Mariano, Thomas M, Heck, Diane E, Laskin, Jeffrey D, Heindel, Ned D
Published in Heterocyclic letters (01.08.2018)
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Published in Heterocyclic letters (01.08.2018)
Journal Article
Azetidinones as vasopressin V1a antagonists
Guillon, Christophe D., Koppel, Gary A., Brownstein, Michael J., Chaney, Michael O., Ferris, Craig F., Lu, Shi-fang, Fabio, Karine M., Miller, Marvin J., Heindel, Ned D., Hunden, David C., Cooper, Robin D.G., Kaldor, Stephen W., Skelton, Jeffrey J., Dressman, Bruce A., Clay, Michael P., Steinberg, Mitchell I., Bruns, Robert F., Simon, Neal G.
Published in Bioorganic & medicinal chemistry (01.03.2007)
Published in Bioorganic & medicinal chemistry (01.03.2007)
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Journal Article
Peripheral site acetylcholinesterase inhibitors targeting both inflammation and cholinergic dysfunction
Young, Sherri, Fabio, Karine, Guillon, Christophe, Mohanta, Pramod, Halton, Timothy A., Heck, Diane E., Flowers, Robert A., Laskin, Jeffrey D., Heindel, Ned D.
Published in Bioorganic & medicinal chemistry letters (01.05.2010)
Published in Bioorganic & medicinal chemistry letters (01.05.2010)
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Journal Article
Hydrazide pharmaceuticals as conjugates to polyaldehyde dextran: syntheses, characterization, and stability
Heindel, Ned D, Zhao, Huiru, Leiby, Jeffrey, VanDongen, Jacobus M, Lacey, C. Jeffrey, Lima, Daniel A, Shabsoug, Barakat, Buzby, John H
Published in Bioconjugate chemistry (01.01.1990)
Published in Bioconjugate chemistry (01.01.1990)
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Journal Article
A novel heterobifunctional linker for formyl to thiol coupling
Heindel, Ned D, Zhao, Huiru, Egolf, Roger A, Chang, Chien Hsing, Schray, Keith J, Emrich, Jacqueline G, McLaughlin, Joanne P, Woo, David V
Published in Bioconjugate chemistry (01.11.1991)
Published in Bioconjugate chemistry (01.11.1991)
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Journal Article
Misonidazole conjugates of the colorectal tumor-associated monoclonal antibody 17-1A
Pierce, D. L, Heindel, Ned D, Schray, K. J, Jetter, M. M, Emrich, J. G, Woo, D. V
Published in Bioconjugate chemistry (01.09.1990)
Published in Bioconjugate chemistry (01.09.1990)
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